L-152,804 CAS: 6508-43-6
MF: C23H26O4
MW: 366.46
A potent, selective non-peptide NPY5-R receptor antagonist.

L-152,804 (CAS 6508-43-6)

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Alternate Names: 9-(2-Hydroxy-4,4-dimethyl-6-oxo-1-cyclohexen-1-yl)-3,3-dimethyl-2,3,4,9-tetrahydro-1H-xanthen-1-one
Application: L-152,804 is a potent, selective non-peptide NPY5-R receptor antagonist
CAS Number: 6508-43-6
Purity: ≥90%
Molecular Weight: 366.46
Molecular Formula: C23H26O4
For Research Use Only. Not Intended for Diagnostic or Therapeutic Use.
* Refer to Certificate of Analysis for lot specific data (including water content).
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L-152,804 is a potent, selective, non-peptide NPY5-R antagonist (neuropeptide Y) (Ki = 26 nM for hNPY5-R). Displays > 300-fold selectivity over hNPY1-R, hNPY2-R, and hNPY4-R.


References

1. Kanatani, A., et al. 2000. Biochem. Biophys. Res. Comm. 272: 169-173.
2. Schroeder, J.P., et al. 2005. Alcohol 36: 179-186.
3. Mashiko, S., et al. 2007. Mol. Pharmacol. 71: 602-608.

Physical State :
Solid
Solubility :
Soluble in DMSO (100 mM).
Storage :
Desiccate at 4° C
Melting Point :
208.79° C (Predicted)
Boiling Point :
513.72° C at 760 mmHg (Predicted)
Density :
1.21 g/cm3 (Predicted)
Refractive Index :
n20D 1.58 (Predicted)
Ki Data :
NPY5-R: Ki= 26 nM
pK Values :
pKa: 4.86 (Predicted)
For Research Use Only. Not Intended for Diagnostic or Therapeutic Use.
PubChem CID :
624746
MDL Number :
MFCD00184132
SMILES :
CC1(CC(=C(C(=O)C1)C2C3=CC=CC=C3OC4=C2C(=O)CC(C4)(C)C)O)C

Download SDS (MSDS)

Certificate of Analysis

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