Molecular structure of JMV3002, CAS Number: 925239-03-8
JMV3002 (CAS 925239-03-8)
Application:
JMV3002 is a strong ghrelin receptor antagonist
CAS Number:
925239-03-8
Molecular Weight:
586.70
Molecular Formula:
C35H34N6O3
Supplemental Information:
This is classified as a Dangerous Good for transport and may be subject to additional shipping charges.
For Research Use Only. Not Intended for Diagnostic or Therapeutic Use.
* Refer to Certificate of Analysis for lot specific data.
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SDS & Certificate of Analysis
JMV3002 is a strong ghrelin receptor antagonist with an IC50 value of 1.1 nM in vitro.1 At 80 µg/kg, JMV3002 inhibits hexarelin-stimulated food intake by as much as 98% in rats.1 JMV3002 alone does not elicit growth hormone release nor does it inhibit hexarelin-stimulated growth hormone secretion when tested in infant rats at a dose of 160 µg/kg.1
JMV3002 (CAS 925239-03-8) References
1 Moulin, A., Demange, L., Ryan, J., et al. New trisubstituted 1,2,4-triazole derivatives as potent ghrelin receptor antagonists. 3. Synthesis and pharmacological in vitro and in vivo evaluations. J Med Chem 51 689-693 (2008).Inhibitor of:
Ghrelin.Ordering Information
| Product Name | Catalog # | UNIT | Price | Qty | FAVORITES | |
JMV3002, 100 µg | sc-221780 | 100 µg | $47.00 | |||
JMV3002, 500 µg | sc-221780A | 500 µg | $210.00 |