ICI-199,441 hydrochloride (CAS 115199-84-3)

ICI-199,441 hydrochloride (CAS 115199-84-3) References

1. Characterization of the antinociceptive effects of TRK-820 in the rat.  |  Endoh, T., et al. 2000. Eur J Pharmacol. 387: 133-40. PMID: 10650153
2. Arylacetamides as peripherally restricted kappa opioid receptor agonists.  |  Kumar, V., et al. 2000. Bioorg Med Chem Lett. 10: 2567-70. PMID: 11086731
3. Modulation of myofilament Ca2+ densitivity by delta- and kappa-opioid agonists in intact guinea pig hearts.  |  Nakae, Y., et al. 2003. Anesth Analg. 96: 733-739. PMID: 12598254
4. Effect of repeated administration of TRK-820, a kappa-opioid receptor agonist, on tolerance to its antinociceptive and sedative actions.  |  Suzuki, T., et al. 2004. Brain Res. 995: 167-75. PMID: 14672806
5. Differential properties between TRK-820 and U-50,488H on the discriminative stimulus effects in rats.  |  Mori, T., et al. 2004. Life Sci. 75: 2473-82. PMID: 15350822
6. A bivalent ligand (KDAN-18) containing delta-antagonist and kappa-agonist pharmacophores bridges delta2 and kappa1 opioid receptor phenotypes.  |  Daniels, DJ., et al. 2005. J Med Chem. 48: 1713-6. PMID: 15771416
7. Structure/activity studies related to 2-(3,4-dichlorophenyl)-N-methyl-N-[2-(1-pyrrolidinyl)-1-substituted- ethyl]acetamides: a novel series of potent and selective kappa-opioid agonists.  |  Barlow, JJ., et al. 1991. J Med Chem. 34: 3149-58. PMID: 1659636
8. Comparative pharmacological profiles of morphine and oxycodone under a neuropathic pain-like state in mice: evidence for less sensitivity to morphine.  |  Narita, M., et al. 2008. Neuropsychopharmacology. 33: 1097-112. PMID: 17593930
9. Opioid modulation of ferret vagal afferent mechanosensitivity.  |  Page, AJ., et al. 2008. Am J Physiol Gastrointest Liver Physiol. 294: G963-70. PMID: 18258789
10. Chemical function-based pharmacophore development for novel, selective kappa opioid receptor agonists.  |  Singh, N., et al. 2008. J Mol Graph Model. 27: 131-9. PMID: 18456526
11. 2-(3,4-Dichlorophenyl)-N-methyl-N-[2-(1-pyrrolidinyl)-1-substituted- ethyl]-acetamides: the use of conformational analysis in the development of a novel series of potent opioid kappa agonists.  |  Costello, GF., et al. 1991. J Med Chem. 34: 181-9. PMID: 1846918
12. Prospects of Using of κ-Opioid Receptor Agonists U-50,488 and ICI 199,441 for Improving Heart Resistance to Ischemia/Reperfusion.  |  Tsibulnikov, SY., et al. 2015. Bull Exp Biol Med. 159: 718-21. PMID: 26519268
13. A novel series of potent and selective agonists at the opioid kappa-receptor.  |  Costello, GF., et al. 1988. Eur J Pharmacol. 151: 475-8. PMID: 2850924
14. Fundamental features of receptor-mediated Gαi/o activation in human prefrontal cortical membranes: A postmortem study.  |  Odagaki, Y., et al. 2020. Brain Res. 1747: 147032. PMID: 32745659
15. Activation of Peripheral Opioid Kappa1 Receptor Prevents Cardiac Reperfusion Injury.  |  Popov, SV., et al. 2021. Physiol Res. 70: 523-531. PMID: 34062075