Molecular structure of Glucagon Receptor Antagonist, Control, CAS Number: 362482-00-6
Glucagon Receptor Antagonist, Control (CAS 362482-00-6)
Alternate Names:
N-(3-Cyano-6-(1,1-dimethylpropyl)-4,5,6,7-tetrahydro-1-benzothien-2-yl)-4-bromobenzamide
Application:
Glucagon Receptor Antagonist, Control is a compound that serves as an inactive control for Glucagon Receptor Antagonist
CAS Number:
362482-00-6
Molecular Weight:
431.4
Molecular Formula:
C21H23BrN2OS
For Research Use Only. Not Intended for Diagnostic or Therapeutic Use.
* Refer to Certificate of Analysis for lot specific data.
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Description
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SDS & Certificate of Analysis
Glucagon Receptor Antagonist, Control is a cell-permeable thienyl-amide compound that serves as an inactive control for Glucagon Receptor Antagonist. Glucagon Receptor Antagonist, Control displays weak affinity for hGCGR and is ineffective when preventing glucagon binding (20% inhibition at 10 μM in membranes prepared from CHO-hGCGR) and glucagon-, forskolin-, and GIP-induced cAMP production (10% inhibition in CHO-hGCGR cells). Only minimally suppresses glucagon-induced glycogenolysis in human primary hepatocytes.
Glucagon Receptor Antagonist, Control (CAS 362482-00-6) References
- A novel glucagon receptor antagonist inhibits glucagon-mediated biological effects. | Qureshi, SA., et al. 2004. Diabetes. 53: 3267-73. PMID: 15561959
Inhibitor of:
Glucagon Receptor.Ordering Information
| Product Name | Catalog # | UNIT | Price | Qty | FAVORITES | |
Glucagon Receptor Antagonist, Control, 1 mg | sc-203973 | 1 mg | $180.00 | |||
Glucagon Receptor Antagonist, Control, 5 mg | sc-203973A | 5 mg | $902.00 |