Molecular structure of Gavestinel, CAS Number: 153436-38-5
Gavestinel (CAS 153436-38-5)
Alternate Names:
4,6-Dichloro-3-[(1E)-3-oxo-3-(phenylamino)-1-propenyl]-1H-indole-2-carboxylic acid sodium salt; Gavestinel sodium
Application:
Gavestinel is a potent, selective, and non competitive NMDA receptor antagonist
CAS Number:
153436-38-5
Purity:
≥98%
Molecular Weight:
397.19
Molecular Formula:
C18H11Cl2N2O3Na
For Research Use Only. Not Intended for Diagnostic or Therapeutic Use.
* Refer to Certificate of Analysis for lot specific data.
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SDS & Certificate of Analysis
Gavestinel is a potent and selective, non competitive antagonist. The compound has been shown to act at the NMDA receptor-channel complexes strychnine insensitive glycine binding site. Gavestinel has been reported to be more selective than AMPA, kainate, and NMDA binding sites.
Gavestinel (CAS 153436-38-5) References
Di Fabio et al (1997) Substituted indole-2-carboxylates as in vivo potent antagonists acting at the strychnine-insensitive glycine binding site. J.Med.Chem. 40 841. Mugnaini et al (2000) Receptor binding characteristics of the novel NMDA receptor glycineInhibitor of:
NMDA.Ordering Information
| Product Name | Catalog # | UNIT | Price | Qty | FAVORITES | |
Gavestinel, 10 mg | sc-361183 | 10 mg | $159.00 | |||
Gavestinel, 50 mg | sc-361183A | 50 mg | $650.00 |