Molecular structure of Fluvoxamine maleate, CAS Number: 61718-82-9
Fluvoxamine maleate (CAS 61718-82-9)
Alternate Names:
(E)-5-Methoxy-1-[4-(trifluoromethyl)phenyl]-1-pentanone-O-(2-aminoethyl)oxime maleate
Application:
Fluvoxamine maleate is a SR inhibitor which binds to the 5-HT transporter
CAS Number:
61718-82-9
Purity:
≥99%
Molecular Weight:
434.41
Molecular Formula:
C15H21F3N2O2•C4H4O4
For Research Use Only. Not Intended for Diagnostic or Therapeutic Use.
* Refer to Certificate of Analysis for lot specific data.
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Description
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SDS & Certificate of Analysis
Fluvoxamine maleate is a selective SR (serotonin reputake) inhibitor. It binds to the 5-HT transporter protein with high affinity (Ki = 1.6 nM) and demonstrates very low affinity at the norepinephrine transporter (Ki = 2,950 nM). Fluvoxamine maleate is a Sigma Receptor agonist. It has been in a number of in vitro experiments, including studies of its effects on serotonin and norepinephrine reuptake, the release of neurotransmitters, the expression of various proteins, cell viability, and the production of various cytokines.
Fluvoxamine maleate (CAS 61718-82-9) References
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- Use of acetylacetone for nano-level assay of fluvoxamine maleate in pure form and pharmaceutical formulation. | Abu-Hassan, AA., et al. 2020. Luminescence. 35: 1360-1365. PMID: 32519373
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Inhibitor of:
SR.Activator of:
Sigma Receptor.Ordering Information
| Product Name | Catalog # | UNIT | Price | Qty | FAVORITES | |
Fluvoxamine maleate, 10 mg | sc-203582 | 10 mg | $51.00 | |||
Fluvoxamine maleate, 50 mg | sc-203582A | 50 mg | $224.00 |