Molecular structure of Fananserin, CAS Number: 127625-29-0
Fananserin (CAS 127625-29-0)
Alternate Names:
RP 62203
Application:
Fananserin is an antagonist of 5-HT2A
CAS Number:
127625-29-0
Purity:
≥99%
Molecular Weight:
425.52
Molecular Formula:
C23H24FN3O2S
For Research Use Only. Not Intended for Diagnostic or Therapeutic Use.
* Refer to Certificate of Analysis for lot specific data.
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SDS & Certificate of Analysis
Fananserin is a potent 5-HT2A and D4 receptor (dopamine D4) antagonist, with efficacy against histamine H1, α1 and 5HT having Ki values of 0.26, 2.93, 25, 38, 70, and 726 nM, respectively. Fananserin shows very modest efficacy towards Dopamine D2 receptors with a Ki value of 726 nM.
Fananserin (CAS 127625-29-0) References
1. Malleron, J.L., et al. 1991. J. Med. Chem. 34: 2477-2483.2. Doble, A., et al. 1992. Br. J. Pharmacol. 105: 27-36.
3. Heuillet, E., et al. 1996. Eur. J. Pharmacol. 314: 229-233.
Inhibitor of:
D4DR, and SR-2A.Ordering Information
| Product Name | Catalog # | UNIT | Price | Qty | FAVORITES | |
Fananserin, 10 mg | sc-203951 | 10 mg | $155.00 | |||
Fananserin, 50 mg | sc-203951A | 50 mg | $620.00 |