Molecular structure of E4CPG, CAS Number: 170846-89-6
E4CPG (CAS 170846-89-6)
Alternate Names:
(RS)-α-Ethyl-4-carboxyphenylglycine; 4-(2-amino-1-hydroxy-1-oxobutan-2-yl)benzoic acid
Application:
E4CPG is A group I/group II metabotropic glutamate receptor antagonist
CAS Number:
170846-89-6
Molecular Weight:
223.23
Molecular Formula:
C11H13NO4
For Research Use Only. Not Intended for Diagnostic or Therapeutic Use.
* Refer to Certificate of Analysis for lot specific data.
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Description
Technical Information
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SDS & Certificate of Analysis
E4CPG is a group I/group II metabotropic glutamate receptor antagonist which is more potent than (RS)-MCPG (sc-202325).
E4CPG (CAS 170846-89-6) References
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- Dendritic calcium nonlinearities switch the direction of synaptic plasticity in fast-spiking interneurons. | Camiré, O. and Topolnik, L. 2014. J Neurosci. 34: 3864-77. PMID: 24623765
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- Long-term potentiation of glycinergic synapses by semi-natural stimulation patterns during tonotopic map refinement. | Bach, EC. and Kandler, K. 2020. Sci Rep. 10: 16899. PMID: 33037263
- Structure-activity relationships for a series of phenylglycine derivatives acting at metabotropic glutamate receptors (mGluRs). | Bedingfield, JS., et al. 1995. Br J Pharmacol. 116: 3323-9. PMID: 8719814
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Inhibitor of:
mGluR-1a, mGluR-1b, mGluR-2, mGluR-3, and mGluR-5.Ordering Information
| Product Name | Catalog # | UNIT | Price | Qty | FAVORITES | |
E4CPG, 10 mg | sc-205943 | 10 mg | $129.00 | |||
E4CPG, 50 mg | sc-205943A | 50 mg | $548.00 |