Molecular structure of Compound 101, CAS Number: 865608-11-3
Compound 101 (CAS 161125-36-6)
Alternate Names:
3-({[4-Methyl-5-(Pyridin-4-Yl)-4h-1,2,4-Triazol-3-Yl]methyl}amino)-N-[2-(Trifluoromethyl)benzyl]benzamide; CHEMBL1738877
CAS Number:
161125-36-6
Molecular Weight:
466.50
Molecular Formula:
C24H21F3N6O
For Research Use Only. Not Intended for Diagnostic or Therapeutic Use.
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Compound 101 (CAS 161125-36-6) References
- N,N'-Dithiobisphthalimide, a disulfide aromatic compound, is a potent spermicide agent in humans. | Florez, M., et al. 2011. Syst Biol Reprod Med. 57: 309-17. PMID: 21942567
- Small-Molecule G Protein-Coupled Receptor Kinase Inhibitors Attenuate G Protein-Coupled Receptor Kinase 2-Mediated Desensitization of Vasoconstrictor-Induced Arterial Contractions. | Rainbow, RD., et al. 2018. Mol Pharmacol. 94: 1079-1091. PMID: 29980659
- Chronic Treatment with Morphine Disrupts Acute Kinase-Dependent Desensitization of GPCRs. | Leff, ER., et al. 2020. Mol Pharmacol. 98: 497-507. PMID: 32362586
- Regulation of Kappa Opioid Receptor Inactivation Depends on Sex and Cellular Site of Antagonist Action. | Reichard, KL., et al. 2020. Mol Pharmacol. 98: 548-558. PMID: 32913138
- Structure-Activity Relationship Analysis of Potential New Vapor-Active Insect Repellents. | Richoux, GM., et al. 2020. J Agric Food Chem. 68: 13960-13969. PMID: 33147044
- G protein-coupled receptor kinase 2 is essential to enable vasoconstrictor-mediated arterial smooth muscle proliferation. | Alonazi, ASA. and Willets, JM. 2021. Cell Signal. 88: 110152. PMID: 34555505
- Agonist-Specific Regulation of G Protein-Coupled Receptors after Chronic Opioid Treatment. | Adhikary, S., et al. 2022. Mol Pharmacol. 101: 300-308. PMID: 35193934
- Monoacylglycerol Lipase Protects the Presynaptic Cannabinoid 1 Receptor from Desensitization by Endocannabinoids after Persistent Inflammation. | Bouchet, CA., et al. 2023. J Neurosci. 43: 5458-5467. PMID: 37414560
- GRK2 expression and catalytic activity are essential for vasoconstrictor/ERK-stimulated arterial smooth muscle proliferation. | Alonazi, A., et al. 2023. Biochem Pharmacol. 216: 115795. PMID: 37690571
- G Protein-Coupled Receptor Kinase 2 Selectively Enhances β-Arrestin Recruitment to the D2 Dopamine Receptor through Mechanisms That Are Independent of Receptor Phosphorylation. | Sánchez-Soto, M., et al. 2023. Biomolecules. 13: PMID: 37892234
Inhibitor of:
β-Arrestin-2, GRK 2, JAB1, KOR-3, Olfr695, Olfr697, Olfr698, Olfr699, Olfr700, PRL-1, and TC-PTP.Ordering Information
| Product Name | Catalog # | UNIT | Price | Qty | FAVORITES | |
Compound 101, 5 mg | sc-507528 | 5 mg | $108.00 |