Date published: 2026-4-25

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Carbetapentane citrate (CAS 23142-01-0)

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Application:
Carbetapentane citrate is a compound shown to increase effectiveness of diphenylhydantoin
CAS Number:
23142-01-0
Purity:
99%
Molecular Weight:
525.59
Molecular Formula:
C20H31NO3•C6H8O7
For Research Use Only. Not Intended for Diagnostic or Therapeutic Use.
* Refer to Certificate of Analysis for lot specific data.

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Carbetapentane citrate is a synthetic compound extensively employed in scientific research for its diverse applications. It is a structural analog of the alkaloid pentoxyverine, which naturally occurs in the Peruvian bark tree. Carbetapentane citrate is characterized by its citrate salt form, which enhances its solubility in water compared to the base compound. Understanding how carbetapentane citrate interacts with the body, including its absorption, distribution, metabolism, and excretion (ADME), can provide valuable information.


Carbetapentane citrate (CAS 23142-01-0) References

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  8. Simultaneous determination of potassium guaiacolsulfonate, guaifenesin, diphenhydramine HCl and carbetapentane citrate in syrups by using HPLC-DAD coupled with partial least squares multivariate calibration.  |  Dönmez, OA., et al. 2011. Talanta. 83: 1601-5. PMID: 21238758
  9. The use of carbetapentane for spinal anesthesia and use-dependent block of sodium currents.  |  Leung, YM., et al. 2013. Eur J Pharmacol. 714: 366-72. PMID: 23872380
  10. Carbetapentane citrate.  |  Abo Dena, AS., et al. 2020. Profiles Drug Subst Excip Relat Methodol. 45: 41-53. PMID: 32164969
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  12. Cloning and functional comparison of kappa and delta opioid receptors from mouse brain.  |  Yasuda, K., et al. 1993. Proc Natl Acad Sci U S A. 90: 6736-40. PMID: 8393575
  13. Are high-affinity progesterone binding site(s) from porcine liver microsomes members of the sigma receptor family?  |  Meyer, C., et al. 1998. Eur J Pharmacol. 347: 293-9. PMID: 9653896

Ordering Information

Product NameCatalog #UNITPriceQtyFAVORITES

Carbetapentane citrate, 100 mg

sc-203538
100 mg
$116.00