B-HT 920 CAS: 36085-73-1
MF: C10H15N3S•2HCl
MW: 282.23
A dopamine D2 receptor agonist, SR-3 antagonist and α2-adrenoceptor agonist.

B-HT 920 (CAS 36085-73-1)

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Alternate Names: Talipexole; 5,6,7,8-Tetrahydro-6-(2-propen-1-yl)-4H-thiazolo[4,5-d]azepin-2-amine dihydrochloride
Application: B-HT 920 is a dopamine D2 receptor agonist, SR-3 antagonist and α2-adrenoceptor agonist
CAS Number: 36085-73-1
Purity: ≥99%
Molecular Weight: 282.23
Molecular Formula: C10H15N3S•2HCl
For Research Use Only. Not Intended for Diagnostic or Therapeutic Use.
* Refer to Certificate of Analysis for lot specific data (including water content).

B-HT 920 is a D2DR (dopamine D2 receptor) agonist, SR-3 antagonist and AR (α2-adrenoceptor) agonist. B-HT 920 also displays antiparkinsonian activity.


References

1. Robertson, C.S., et al. 1993. J. Pharmacol. Exp. her. 264: 1344-1351. PMID: 8095550
2. Nishio, H., et al. 1996. Gen. Pharmacol. 27: 779-785. PMID: 8842679
3. Ricci, D. and Taira, C.A. 1999. Gen. Pharmacol. 32: 29-34. PMID: 9888250

Physical State :
Solid
Solubility :
Soluble in water (100 mM), and DMSO (100 mM).
Storage :
Desiccate at room temperature
Melting Point :
243-246° C
Refractive Index :
n20D 1.60 (Predicted)
IC50 :
Adrenergic receptor α-2: IC50 = 25 nM (rat); Adrenergic receptor α-1: IC50 = 500 µM (rat)
Ki Data :
Dopamine D2 receptor: Ki= 5.8 nM (rat)
For Research Use Only. Not Intended for Diagnostic or Therapeutic Use.
WGK Germany :
3
RTECS :
XJ7050340
PubChem CID :
104870
MDL Number :
MFCD00274573
SMILES :
C=CCN1CCC2=C(CC1)SC(=N2)N.Cl.Cl

Download SDS (MSDS)

Certificate of Analysis

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