Molecular structure of Azaperol, CAS Number: 2804-05-9
Azaperol (CAS 2804-05-9)
Alternate Names:
Dihydroazaperone; α-(4-Fluorophenyl)-4-(2-pyridinyl)-1-piperazinebutanol
CAS Number:
2804-05-9
Molecular Weight:
329.41
Molecular Formula:
C19H24FN3O
For Research Use Only. Not Intended for Diagnostic or Therapeutic Use.
* Refer to Certificate of Analysis for lot specific data.
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Azaperol operates through its interaction with the benzodiazepine receptor. By binding to this receptor, Azaperol triggers its activation, resulting in a reduction of anxiety levels and an enhancement of sleep. The influence of Azaperol extends beyond the benzodiazepine receptor, as it has demonstrated the capacity to modulate the activity of additional neurotransmitters, including serotonin and dopamine. This modulation of neurotransmitter function reinforces the reduction of anxiety and the promotion of sleep induced by Azaperol, contributing to its overall effect.
Azaperol (CAS 2804-05-9) References
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- Determination of a method for detecting and quantifying azaperone, azaperol and carazolol in pig tissues by liquid chromatography-tandem mass spectrometry. | Fluchard, D., et al. 2000. J Chromatogr B Biomed Sci Appl. 744: 139-47. PMID: 10985575
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- Simultaneous determination of azaperone and azaperol in animal tissues by HPLC with confirmation by electrospray ionization mass spectrometry. | Aoki, Y., et al. 2009. J Chromatogr B Analyt Technol Biomed Life Sci. 877: 166-72. PMID: 19111512
- Rapid method for the determination of tranquilizers and a beta-blocker in porcine and bovine kidney by liquid chromatography with tandem mass spectrometry. | Mitrowska, K., et al. 2009. Anal Chim Acta. 637: 185-92. PMID: 19286028
- Development and validation of a confirmatory method for the determination of tranquilisers and a β-blocker in porcine and bovine kidney by LC-MS/MS. | Bock, C. and Stachel, CS. 2013. Food Addit Contam Part A Chem Anal Control Expo Risk Assess. 30: 1000-11. PMID: 23767920
- Integrated Risk Index of Chemical Aquatic Pollution (IRICAP): case studies in Iberian rivers. | Fàbrega, F., et al. 2013. J Hazard Mater. 263 Pt 1: 187-96. PMID: 23810233
- Thin-layer chromatographic screening method for the tranquillizers azaperone, propiopromazine and carazolol in pig tissues. | Haagsma, N., et al. 1988. J Chromatogr. 436: 73-9. PMID: 2897377
- Highly sensitive immunochromatographic assay for simultaneous determination of azaperone and azaperol in pork. | Chen, L., et al. 2023. Food Chem X. 17: 100525. PMID: 36478711
- Development of the Chromatographic Method for Simultaneous Determination of Azaperone and Azaperol in Animal Kidneys and Livers. | Kośka, I. and Kubalczyk, P. 2022. Int J Mol Sci. 24: PMID: 36613536
- Evaluation of the effects of the enantiomers of reduced haloperidol, azaperol, and related 4-amino-1-arylbutanols on dopamine and sigma receptors. | Jaen, JC., et al. 1993. J Med Chem. 36: 3929-36. PMID: 7902870
- Investigation of the metabolism of azaperone in the horse. | Chui, YC., et al. 1994. J Chromatogr. 652: 23-33. PMID: 8014224
Ordering Information
| Product Name | Catalog # | UNIT | Price | Qty | FAVORITES | |
Azaperol, 25 mg | sc-503181 | 25 mg | $367.00 |