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AQ-RA 741 is a high affinity, selective mAChR M2 antagonist (pKi values are 8.3, 7.7, and 6.82 for mAChR M2, mAChR M1, and mAChR M3 receptors, respectively). AQ-RA 741 displays cardioselectivity over tracheal, intestinal and bladder muscarinic receptors. AQ-RA 741 also inhibits vagally and agonist-induced bradycardia.
Ordering Information
| Product Name | Catalog # | UNIT | Price | Qty | FAVORITES | |
AQ-RA 741, 10 mg | sc-203517 | 10 mg | $135.00 | |||
AQ-RA 741, 50 mg | sc-203517A | 50 mg | $575.00 |