Date published: 2026-4-26

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4′-Dimethylamino 7,8-Dihydroxyflavone (CAS 1205548-00-0)

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Alternate Names:
2-[4-(Dimethylamino)phenyl]-7,8-dihydroxy-4H-1-benzopyran-4-one; 2-[4-(Dimethylamino)phenyl]-7,8-dihydroxy-4H-chromen-4-one; 4′-DMA-7,8-DHF
CAS Number:
1205548-00-0
Molecular Weight:
297.31
Molecular Formula:
C17H15NO4
For Research Use Only. Not Intended for Diagnostic or Therapeutic Use.
* Refer to Certificate of Analysis for lot specific data.

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4′-Dimethylamino 7,8-Dihydroxyflavone is a compound belonging to the flavonoid class. Although the precise mechanism of action of 4′-Dimethylamino 7,8-Dihydroxyflavone is not yet fully identified, current understanding suggests its involvement in the inhibition of specific enzymes and signaling pathways. Experimental evidence demonstrates its ability to inhibit cyclooxygenase-2 (COX-2), an enzyme in prostaglandin production that promotes inflammation. 4′-Dimethylamino 7,8-Dihydroxyflavone exerts inhibitory effects on matrix metalloproteinases (MMPs), enzymes responsible for extracellular matrix breakdown and tissue remodeling. 4′-Dimethylamino 7,8-Dihydroxyflavone activates the nuclear factor erythroid 2-related factor 2 (Nrf2) pathway, which plays a role in regulating the expression of antioxidant genes, thereby guarding against oxidative stress.


4′-Dimethylamino 7,8-Dihydroxyflavone (CAS 1205548-00-0) References

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Ordering Information

Product NameCatalog #UNITPriceQtyFAVORITES

4′-Dimethylamino 7,8-Dihydroxyflavone, 25 mg

sc-497721
25 mg
$396.00