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2-Formyl-4-methoxyphenylboronic acid (CAS 139962-95-1)

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Alternate Names:
2-Borono-5-methoxybenzaldehyde
CAS Number:
139962-95-1
Molecular Weight:
179.97
Molecular Formula:
C8H9BO4
For Research Use Only. Not Intended for Diagnostic or Therapeutic Use.
* Refer to Certificate of Analysis for lot specific data.

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2-Formyl-4-methoxyphenylboronic acid has found application in diverse scientific studies and research endeavors. In the domain of organic synthesis, it serves as a reagent, enabling the synthesis of various organic compounds. Moreover, in the field of biochemistry, this compound has been instrumental in investigating the effects of boronic acids on the binding of carbohydrates to proteins. Its mechanism of action hinges on its capability to establish a reversible covalent bond with carbohydrates. Specifically, the boron atom within the molecule interacts with the oxygen atoms in carbohydrates, facilitating the formation of a complex in a highly specific manner.


2-Formyl-4-methoxyphenylboronic acid (CAS 139962-95-1) References

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  2. Synthesis of the o-quinones and other oxidized metabolites of polycyclic aromatic hydrocarbons implicated in carcinogenesis.  |  Harvey, RG., et al. 2004. J Org Chem. 69: 2024-32. PMID: 15058949
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  7. Structure-anti-MRSA activity relationship of macrocyclic bis(bibenzyl) derivatives.  |  Sawada, H., et al. 2013. Bioorg Med Chem Lett. 23: 6563-8. PMID: 24239015
  8. Chirality sensing of amines, diamines, amino acids, amino alcohols, and α-hydroxy acids with a single probe.  |  Bentley, KW., et al. 2013. J Am Chem Soc. 135: 18052-5. PMID: 24261969
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  11. TfOH-Catalyzed Intramolecular Annulation of 2-(Aryl)-Phenyl-Substituted p-Quinone Methides under Continuous Flow: Total Syntheses of Selaginpulvilin I and Isoselagintamarlin A.  |  Pankhade, YA., et al. 2022. J Org Chem. 87: 3363-3377. PMID: 35107013
  12. Recent advances in application of intramolecular Suzuki cross-coupling in cyclization and heterocyclization  |  , et al. (2012). Monatshefte für Chemie - Chemical Monthly. volume 143,: pages 861–880.
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Ordering Information

Product NameCatalog #UNITPriceQtyFAVORITES

2-Formyl-4-methoxyphenylboronic acid, 1 g

sc-259910
1 g
$87.00

2-Formyl-4-methoxyphenylboronic acid, 5 g

sc-259910A
5 g
$403.00