Molecular structure of 1-(Phenylsulfonyl)-3-indolylboronic acid, CAS Number: 129271-98-3
1-(Phenylsulfonyl)-3-indolylboronic acid (CAS 129271-98-3)
Application:
1-(Phenylsulfonyl)-3-indolylboronic acid is an indole boronic acid building block
CAS Number:
129271-98-3
Molecular Weight:
301.13
Molecular Formula:
C14H12BNO4S
For Research Use Only. Not Intended for Diagnostic or Therapeutic Use.
* Refer to Certificate of Analysis for lot specific data.
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SDS & Certificate of Analysis
1-(Phenylsulfonyl)-3-indolylboronic acid is an indole boronic acid compound useful as an indole building block for cross-coupling protocols. 1-(Phenylsulfonyl)-3-indolylboronic acid was reported to undergo oxidative Heck coupling with tert-butyl acrylate along with a range of different aryl boronic acids. 1-(Phenylsulfonyl)-3-indolylboronic acid was also used as a starting material in the synthesis of novel c-Jun N-terminal kinase inhibitors.
1-(Phenylsulfonyl)-3-indolylboronic acid (CAS 129271-98-3) References
- Oxygen-promoted Pd(II) catalysis for the coupling of organoboron compounds and olefins. | Jung, YC., et al. 2003. Org Lett. 5: 2231-4. PMID: 12816416
- Synthesis and SAR of aminopyrimidines as novel c-Jun N-terminal kinase (JNK) inhibitors. | Alam, M., et al. 2007. Bioorg Med Chem Lett. 17: 3463-7. PMID: 17459703
- The application of formyl group activation of bromopyrrole esters to formal syntheses of lycogarubin C, permethyl storniamide A and lamellarin G trimethyl ether. | Gupton, JT., et al. 2014. Tetrahedron. 70: 9759-9767. PMID: 25584014
- Investigation of chalcogen bioisosteric replacement in a series of heterocyclic inhibitors of tryptophan 2,3-dioxygenase. | Kozlova, A., et al. 2022. Eur J Med Chem. 227: 113892. PMID: 34678572
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| Product Name | Catalog # | UNIT | Price | Qty | FAVORITES | |
1-(Phenylsulfonyl)-3-indolylboronic acid, 1 g | sc-222634 | 1 g | $168.00 |