* Refer to Certificate of Analysis for lot specific data.
クイックリンク
注文情報
参考文献
説明
技術サポート情報
安全情報
SDSと分析証明書
UCM 707 (CAS 390824-20-1) 参考文献
Design, synthesis and biological evaluation of novel arachidonic acid derivatives as highly potent and selective endocannabinoid transporter inhibitors: M.L. Lopez-Rodriguez, et al.; J. Med. Chem. 44, 4505 (2001) UCM707, a potent and selective inhibitor of endocannabinoid uptake, potentiates hypokinetic and antinociceptive effects of anandamide: E. de Lago, et al.; Eur. J. Pharmacol. 449, 99 (2002) Design, synthesis and biological evaluation of new endocannabinoid transporter inhibitors: M.L. Lopez-Rodriguez, et al.; Eur. J. Med. Chem. 38, 403 (2003) Design, synthesis, and biological evaluation of new inhibitors of the endocannabinoid uptake: comparison with effects on fatty acid amidohydrolase: M.L. Lopez-Rodriguez, et al.; J. Med. Chem. 46, 1512 (2003) Selective inhibition of anandamide cellular uptake versus enzymatic hydrolysis-a difficult issue to handle: C.J. Fowler, et al.; Eur. J. Pharmacol. 492, 1 (2004)
の阻害剤である:
FAAH, VR1.
処方 :
Solution in methyl acetate
身体の状態 :
Liquid
溶解度 :
Soluble in water (0.25 mg/ml at 25° C), ethanol, DMSO, DMF, and ethanol: PBS (ph 7.2) (1: 2).