rac O-Desmethyl venlafaxine β-D-glucuronide (CAS 1021933-98-1)
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rac O-Desmethyl Venlafaxine β-D-Glucuronide is a metabolite of Venlafaxine (sc-201102). Venlafaxine is a derivative of phenylethylamine which is reported to facilitate neurotransmission within the central nervous system via blocking the presynaptic reuptake of neuroamines such as serotonin (5-hydroxytryptamine 5-HT) and noradrenaline (norepinephrine). Velanfaxine is also reported to be a weak inhibitor of dopamine reuptake. In vitro studies indicate that Venlafaxine does not demonstrate significant activity for muscarinic, histaminergic or alpha-1 adrenergic receptors. The metabolism of venlafaxine is reported to occur by cytochrome P450 (CYP) enzyme CYP2D6 yielding O-desmethylvenlafaxine. A lesser metabolite, N-desmethylvenlafaxine is produced by CYP3A4.
rac O-Desmethyl venlafaxine β-D-glucuronide (CAS 1021933-98-1) References
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Ordering Information
| Product Name | Catalog # | UNIT | Price | Qty | FAVORITES | |
rac O-Desmethyl venlafaxine β-D-glucuronide, 1 mg | sc-208279 | 1 mg | $360.00 |