Date published: 2026-3-31

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Endophilin I Inhibitors

Endophilin I inhibitors constitute a diverse group of compounds that either directly target Endophilin I or indirectly modulate its activity by influencing key cellular pathways involved in membrane remodeling and endocytosis. Dynasore, a small molecule inhibitor of dynamin, indirectly modulates Endophilin I by disrupting endocytosis processes. Dynasore-induced dynamin inhibition leads to impaired endocytosis, influencing the recruitment and function of Endophilin I in membrane remodeling and vesicle formation. Ionomycin, a calcium ionophore, indirectly modulates Endophilin I by influencing calcium-dependent cellular processes. Ionomycin-induced calcium influx leads to altered calcium signaling, affecting the recruitment and function of Endophilin I in membrane remodeling and vesicle formation. ML141, a Cdc42 inhibitor, indirectly influences Endophilin I by disrupting Rho GTPase signaling. Dyngo-4a, a dynamin inhibitor, indirectly modulates Endophilin I by disrupting clathrin-mediated endocytosis. Dyngo-4a-induced dynamin inhibition leads to impaired endocytosis, influencing the recruitment and function of Endophilin I in membrane remodeling and vesicle formation. NSC23766, a Rac1 inhibitor, indirectly influences Endophilin I by disrupting Rho GTPase signaling. CK666, an Arp2/3 complex inhibitor, indirectly modulates Endophilin I by disrupting actin polymerization. CK666-induced Arp2/3 complex inhibition leads to altered actin dynamics, affecting the recruitment and function of Endophilin I in membrane remodeling and endocytosis processes. SMIFH2, an inhibitor of formin homology 2 (FH2) domains, indirectly influences Endophilin I by disrupting actin dynamics. Jasplakinolide, an actin polymerization stabilizer, indirectly modulates Endophilin I by influencing actin dynamics. Jasplakinolide-induced actin stabilization leads to altered actin polymerization, affecting the recruitment and function of Endophilin I in membrane remodeling and endocytosis processes. Wiskostatin, an N-WASP inhibitor, indirectly influences Endophilin I by disrupting actin polymerization. CK869, a myosin II inhibitor, indirectly modulates Endophilin I by disrupting actin dynamics. CK869-induced myosin II inhibition leads to altered actin polymerization, affecting the recruitment and function of Endophilin I in membrane remodeling and endocytosis processes. ML7, a myosin light chain kinase (MLCK) inhibitor, indirectly influences Endophilin I by disrupting actin dynamics.

Items 1 to 10 of 11 total

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Product NameCAS #Catalog #QUANTITYPriceCitationsRATING

Dynamin Inhibitor I, Dynasore

304448-55-3sc-202592
10 mg
$89.00
44
(2)

Dynasore is a small molecule inhibitor of dynamin, which indirectly modulates Endophilin I by disrupting endocytosis. Dynasore-induced dynamin inhibition leads to impaired endocytosis processes, influencing the recruitment and function of Endophilin I in membrane remodeling and vesicle formation.

Dynamin Inhibitor II

1119-97-7sc-203931
sc-203931A
sc-203931B
sc-203931C
25 g
250 g
500 g
1 kg
$47.00
$84.00
$124.00
$198.00
(1)

Dynamin Inhibitor II is a myosin inhibitor that indirectly influences Endophilin I by disrupting actin dynamics. MiTMAB-induced myosin inhibition leads to altered actin polymerization, affecting the recruitment and function of Endophilin I in membrane remodeling and endocytosis processes.

Ionomycin, free acid

56092-81-0sc-263405
sc-263405A
1 mg
5 mg
$96.00
$264.00
2
(2)

Ionomycin is a calcium ionophore that indirectly modulates Endophilin I by influencing calcium-dependent cellular processes. Ionomycin-induced calcium influx leads to altered calcium signaling, affecting the recruitment and function of Endophilin I in membrane remodeling and vesicle formation.

ML 141

71203-35-5sc-362768
sc-362768A
5 mg
25 mg
$137.00
$512.00
7
(1)

ML141 is a Cdc42 inhibitor that indirectly influences Endophilin I by disrupting Rho GTPase signaling. ML141-induced Cdc42 inhibition leads to altered actin dynamics, affecting the recruitment and function of Endophilin I in membrane remodeling and endocytosis processes.

Hydroxy-Dynasore

1256493-34-1sc-364678
10 mg
$255.00
(0)

Hydroxy-Dynasore is a dynamin inhibitor that indirectly modulates Endophilin I by disrupting clathrin-mediated endocytosis. Hydroxy-Dynasore-induced dynamin inhibition leads to impaired endocytosis processes, influencing the recruitment and function of Endophilin I in membrane remodeling and vesicle formation.

CK 666

442633-00-3sc-361151
sc-361151A
10 mg
50 mg
$321.00
$1040.00
5
(0)

CK666 is an Arp2/3 complex inhibitor that indirectly modulates Endophilin I by disrupting actin polymerization. CK666-induced Arp2/3 complex inhibition leads to altered actin dynamics, affecting the recruitment and function of Endophilin I in membrane remodeling and endocytosis processes.

SMIFH2

340316-62-3sc-507273
5 mg
$140.00
(0)

SMIFH2 is an inhibitor of formin homology 2 (FH2) domains that indirectly influences Endophilin I by disrupting actin dynamics. SMIFH2-induced FH2 domain inhibition leads to altered actin polymerization, affecting the recruitment and function of Endophilin I in membrane remodeling and endocytosis processes.

Jasplakinolide

102396-24-7sc-202191
sc-202191A
50 µg
100 µg
$184.00
$305.00
59
(1)

Jasplakinolide is an actin polymerization stabilizer that indirectly modulates Endophilin I by influencing actin dynamics. Jasplakinolide-induced actin stabilization leads to altered actin polymerization, affecting the recruitment and function of Endophilin I in membrane remodeling and endocytosis processes.

Wiskostatin

253449-04-6sc-204399
sc-204399A
sc-204399B
sc-204399C
1 mg
5 mg
25 mg
50 mg
$49.00
$124.00
$441.00
$828.00
4
(1)

Wiskostatin is an N-WASP inhibitor that indirectly influences Endophilin I by disrupting actin polymerization. Wiskostatin-induced N-WASP inhibition leads to altered actin dynamics, affecting the recruitment and function of Endophilin I in membrane remodeling and endocytosis processes.

CK-869

388592-44-7sc-507274
5 mg
$163.00
(0)

CK869 is a myosin II inhibitor that indirectly modulates Endophilin I by disrupting actin dynamics. CK869-induced myosin II inhibition leads to altered actin polymerization, affecting the recruitment and function of Endophilin I in membrane remodeling and endocytosis processes.