CYP3A4 Inhibitors
Cytochrome P450 (CYP) proteins are heme-thiolate monooxygenases that mediate NADPH-dependent electron transport and function to oxidize a variety of structurally unrelated compounds, including steroids, fatty acids and xenobiotics. Biochemicals that inhibit CYP3A4 have many applications in biochemical and physiological research. Click on the product name to view detailed information such as the chemical structure and specific chemical properties for each of our CYP3A4 Inhibitors. In stock CYP3A4 Inhibitors are available for immediate shipping.
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SEE ALSO...
- CYP3A4 Antibodies for 10 µg trial size samples
- ChemCruz™ Chemical CYP3A4 Activators or CYP3A4 Substrates for functional analysis of cellular responses to CYP3A4
| PRODUCT NAME/Application | CAS | Catalog # | QUANTITY | Price | Citations | RATING | |
|---|---|---|---|---|---|---|---|
MetyraponeMetyrapone is an inhibitor of cytochrome P450-mediated ω/ω-1 hydroxylase activity and CYP11B1 |
54-36-4 |
sc-200597 sc-200597A sc-200597B |
200 mg 500 mg 1 g |
$20.00
$50.00 $79.00 |
3 |
| |
ErythromycinErythromycin is a macrolide antibiotic protein synthesis inhibitor |
114-07-8 |
sc-204742 |
5 g |
$44.00
|
3 |
| |
KetoconazoleKetoconazole is an inhibitor of CYP proteins, thromboxane synthetase, and 5-LO |
65277-42-1 |
sc-200496 sc-200496A |
50 mg 500 mg |
$54.00
$249.00 |
20 |
| |
IsoniazidIsoniazid is an antituberculosis agent and an inhibitor/activator of CYP isoenzymes |
54-85-3 |
sc-205722 sc-205722A sc-205722B |
5 g 50 g 100 g |
$20.00
$25.00 $36.00 |
0 |
| |
ItraconazoleItraconazole is a triazole antifungal agent |
84625-61-6 |
sc-205724 sc-205724A |
50 mg 100 mg |
$70.00
$131.00 |
22 |
| |
MyricetinMyricetin is a cell-permeable, ATP-competitive inhibitor of various casein kinases and protein kinases. |
529-44-2 |
sc-203147 sc-203147A sc-203147B sc-203147C sc-203147D |
25 mg 100 mg 1 g 25 g 100 g |
$93.00
$180.00 $250.00 $490.00 $982.00 |
2 |
| |
NaringinNaringin is a citrus bioflavonoid reported to inhibit cytochrom P450 monooxygenase activity |
10236-47-2 |
sc-203443 sc-203443A |
25 g 50 g |
$38.00
$92.00 |
6 |
| |
ClotrimazoleClotrimazole is an antifungal compound and CYP inhibitor |
23593-75-1 |
sc-3583 sc-3583A |
100 mg 1 g |
$35.00
$50.00 |
6 |
| |
FluconazoleFluconazole is a triazole broad-spectrum antifungal agent particularly for candida species |
86386-73-4 |
sc-205698 sc-205698A |
500 mg 1 g |
$52.00
$82.00 |
14 |
| |
6prime,7prime-dihydroxy Bergamottin6′,7′-dihydroxy Bergamottin is a potent CYP3A4 inhibitor |
145414-76-2 |
sc-205162 sc-205162A |
1 mg 10 mg |
$100.00
$600.00 |
1 |
| |
ClarithromycinClarithromycin is a macrolide antibiotic and protein synthesis inhibitor |
81103-11-9 |
sc-205634 sc-205634A |
100 mg 250 mg |
$69.00
$113.00 |
1 |
| |
Desacetyl diltiazemDesacetyl diltiazem is a metabolite of Diltiazem |
42399-40-6 |
sc-207527 |
10 mg |
$290.00
|
1 |
| |
StiripentolStiripentol is an inhibitor of CYP1A2, CYP2C19 and CYP3A4 |
49763-96-4 |
sc-208402 |
100 mg |
$340.00
|
0 |
| |
OmeprazoleOmeprazole is a selective proton pump and CYP inhibitor |
73590-58-6 |
sc-202265 |
50 mg |
$65.00
|
4 |
| |
AzamulinAzamulin is a highly selective CYP3A4 inhibitor & a mutilin derivative |
76530-44-4 |
sc-207310 |
5 mg |
$228.00
|
0 |
| |
Clarithromycin-N-methyl-d3Clarithromycin-N-methyl-d3 (contains 2% d0) is a deuterium-labeled clarithromycin derivative and a CYP4A inhibitor and substrate |
sc-217926 |
5 mg |
$320.00
|
0 |
| ||
Ritonavir-d6Ritonavir-d6 is a deuterated selective HIV-1 protease inhibitor |
155213-67-5 (unlabeled) |
sc-355967 |
10 mg |
$3,125.00
|
0 |
| |
alpha-Asaroneα-Asarone is an inhibitor of HMG-CoA reductase and CYP isoenzymes |
2883-98-9 |
sc-239153 |
1 g |
$55.00
|
0 |
| |
RitonavirRitonavir is an inhibitor of HIV-1 protease |
155213-67-5 |
sc-208310 |
10 mg |
$120.00
|
7 |
| |
Fluconazole-d4Fluconazole-d4 is a deuterium labeled fluconazole used to study the antifungal effects of this compound |
1124197-58-5 |
sc-218490 |
1 mg |
$340.00
|
0 |
| |
Isoniazid-d4Isoniazid-d4 is an inhibitor and an inducer of various isoforms of CYP450 |
774596-24-6 |
sc-218611 |
1 mg |
$340.00
|
1 |
| |
N-Desmethyl Diltiazem HydrochlorideN-Desmethyl Diltiazem Hydrochloride is a calcium channel blocker |
130606-60-9 |
sc-219119 sc-219119A sc-219119B sc-219119C |
10 mg 25 mg 50 mg 100 mg |
$370.00
$850.00 $1,503.00 $2,400.00 |
0 |
|