CYP3A4 Inhibitors

Cytochrome P450 (CYP) proteins are heme-thiolate monooxygenases that mediate NADPH-dependent electron transport and function to oxidize a variety of structurally unrelated compounds, including steroids, fatty acids and xenobiotics. Biochemicals that inhibit CYP3A4 have many applications in biochemical and physiological research. Click on the product name to view detailed information such as the chemical structure and specific chemical properties for each of our CYP3A4 Inhibitors. In stock CYP3A4 Inhibitors are available for immediate shipping.

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PRODUCT NAME/ApplicationCASCatalog #QUANTITYPriceCitationsRATING
Metyrapone
An inhibitor of cytochrome P450-mediated ω/ω-1 hydroxylase activity and CYP11B1
54-36-4sc-200597
sc-200597A
sc-200597B
200 mg
500 mg
1 g
$20.00
$50.00
$79.00
0
(3)
Erythromycin
A macrolide antibiotic protein synthesis inhibitor
114-07-8sc-204742
5 g
$44.00
1
(2)
Ketoconazole
An inhibitor of CYP proteins, thromboxane synthetase, and 5-LO
65277-42-1sc-200496
sc-200496A
50 mg
500 mg
$54.00
$249.00
13
(1)
Isoniazid
An antituberculosis agent and an inhibitor/activator of CYP isoenzymes
54-85-3sc-205722
sc-205722A
sc-205722B
5 g
50 g
100 g
$20.00
$25.00
$36.00
0
(1)
Itraconazole
A triazole antifungal agent
84625-61-6sc-205724
sc-205724A
50 mg
100 mg
$70.00
$131.00
10
(1)
Myricetin
An ATP-competitive inhibitor of various casein kinases and protein kinases
529-44-2sc-203147
sc-203147A
sc-203147B
sc-203147C
sc-203147D
25 mg
100 mg
1 g
25 g
100 g
$93.00
$180.00
$250.00
$490.00
$982.00
0
(1)
Naringin
A citrus bioflavonoid reported to inhibit cytochrom P450 monooxygenase activity
10236-47-2sc-203443
sc-203443A
25 g
50 g
$38.00
$92.00
1
(1)
Clotrimazole
An antifungal compound and CYP inhibitor
23593-75-1sc-3583
sc-3583A
100 mg
1 g
$35.00
$50.00
4
(2)
Fluconazole
A triazole broad-spectrum antifungal agent particularly for candida species
86386-73-4sc-205698
sc-205698A
500 mg
1 g
$52.00
$82.00
1
(1)
6prime,7prime-dihydroxy Bergamottin
A potent CYP3A4 inhibitor
145414-76-2sc-205162
sc-205162A
1 mg
10 mg
$100.00
$600.00
0
(1)
Clarithromycin
A macrolide antibiotic and protein synthesis inhibitor
81103-11-9sc-205634
sc-205634A
100 mg
250 mg
$69.00
$113.00
0
(1)
Desacetyl diltiazem
A metabolite of Diltiazem
42399-40-6sc-207527
10 mg
$250.00
1
(0)
Stiripentol
An inhibitor of CYP1A2, CYP2C19 and CYP3A4
49763-96-4sc-208402
100 mg
$300.00
0
(0)
Omeprazole
A selective proton pump and CYP inhibitor
73590-58-6sc-202265
50 mg
$65.00
3
(1)
Azamulin
A highly selective CYP3A4 inhibitor & a mutilin derivative
76530-44-4sc-207310
5 mg
$188.00
0
(1)
Clarithromycin-N-methyl-d3 (contains 2% d0)
A deuterium-labeled clarithromycin derivative and a CYP4A inhibitor and substrate
sc-217926
5 mg
$280.00
0
(0)
Ritonavir-d6
A deuterated selective HIV-1 protease inhibitor
155213-67-5 (unlabeled)sc-355967
10 mg
$3,125.00
0
(0)
alpha-Asarone
An inhibitor of HMG-CoA reductase and CYP isoenzymes
2883-98-9sc-239153
1 g
$55.00
0
(0)
Ritonavir
An inhibitor of HIV-1 protease
155213-67-5sc-208310
10 mg
$120.00
5
(1)
Fluconazole-d4
A deuterium labeled fluconazole used to study the antifungal effects of this compound
1124197-58-5sc-218490
1 mg
$300.00
0
(1)
Isoniazid-d4
An inhibitor and an inducer of various isoforms of CYP450
774596-24-6sc-218611
1 mg
$300.00
0
(0)
N-Desmethyl Diltiazem Hydrochloride
A calcium channel blocker
130606-60-9sc-219119
sc-219119A
sc-219119B
sc-219119C
10 mg
25 mg
50 mg
100 mg
$300.00
$700.00
$1,300.00
$2,250.00
0
(0)

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