Items 1 to 10 of 13 total
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| Product Name | CAS # | Catalog # | QUANTITY | Price | Citations | RATING |
|---|---|---|---|---|---|---|
MLN8237 | 1028486-01-2 | sc-394162 | 5 mg | $220.00 | ||
A highly selective Aurora A kinase inhibitor, commonly studied for its potential in affecting various cancers. Aurora A kinase is a crucial regulator in various cellular processes, including centrosome maturation and mitotic entry. Small molecule inhibitors of Aurora A kinase can indirectly disrupt centrin function due to centrins' role in centrosome dynamics. | ||||||
2-APB | 524-95-8 | sc-201487 sc-201487A | 20 mg 100 mg | $27.00 $52.00 | 37 | |
2-APB can modulate intracellular calcium levels. By altering calcium concentrations, it can affect Centrin activity. | ||||||
Thapsigargin | 67526-95-8 | sc-24017 sc-24017A | 1 mg 5 mg | $94.00 $349.00 | 114 | |
Thapsigargin depletes intracellular calcium stores, which can indirectly modulate Centrin function. | ||||||
Tozasertib | 639089-54-6 | sc-358750 sc-358750A | 25 mg 50 mg | $61.00 $85.00 | 4 | |
A pan-Aurora kinase inhibitor with strong activity against Aurora A, also showing potential in cancer research. Aurora A kinase is a crucial regulator in various cellular processes, including centrosome maturation and mitotic entry. Small molecule inhibitors of Aurora A kinase can indirectly disrupt centrin function due to centrins' role in centrosome dynamics. | ||||||
Nifedipine | 21829-25-4 | sc-3589 sc-3589A | 1 g 5 g | $58.00 $170.00 | 15 | |
Nifedipine is an L-type calcium channel blocker; by inhibiting calcium influx, it can impact Centrin activity. | ||||||
AZD1152-HQPA | 722544-51-6 | sc-265334 | 10 mg | $375.00 | ||
Primarily an Aurora B inhibitor, but also exhibits inhibitory activity against Aurora A kinase at higher concentrations. Aurora A kinase is a crucial regulator in various cellular processes, including centrosome maturation and mitotic entry. Small molecule inhibitors of Aurora A kinase can indirectly disrupt centrin function due to centrins' role in centrosome dynamics. | ||||||
EGTA | 67-42-5 | sc-3593 sc-3593A sc-3593B sc-3593C sc-3593D | 1 g 10 g 100 g 250 g 1 kg | $20.00 $62.00 $116.00 $246.00 $799.00 | 23 | |
EGTA is a calcium chelator, and by binding free calcium, it can potentially influence Centrin's function. | ||||||
TMB-8 • HCl | 53464-72-5 | sc-3522 sc-3522A | 10 mg 50 mg | $42.00 $126.00 | 10 | |
TMB-8 inhibits intracellular calcium release, potentially affecting Centrin's calcium-binding role. | ||||||
BAPTA, Free Acid | 85233-19-8 | sc-201508 sc-201508A | 100 mg 500 mg | $67.00 $262.00 | 10 | |
BAPTA acts as a calcium chelator, and its capacity to bind free calcium can have an effect on Centrin's function. | ||||||
Ryanodine | 15662-33-6 | sc-201523 sc-201523A | 1 mg 5 mg | $219.00 $765.00 | 19 | |
Ryanodine modifies calcium release from intracellular stores, potentially influencing Centrin activity. | ||||||