Date published: 2026-4-24

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A1 Inhibitors

A1 inhibitors belong to a class of chemical compounds specifically developed to target and suppress the activity of the A1 receptor, which is a subtype of adenosine receptors. These inhibitors are carefully designed to interact with the A1 receptor and modulate its function, thereby influencing the cellular signaling pathways it regulates. By inhibiting the A1 receptor, these compounds have the ability to alter the cellular responses mediated by adenosine signaling, leading to downstream effects on various physiological processes within the body. The research and development of A1 inhibitors are driven by the desire to gain a deeper understanding of the A1 receptor's role in cellular signaling and its involvement in different biological functions. The identification and characterization of A1 inhibitors provide valuable tools for studying adenosine receptor pharmacology and offer insights into the intricate mechanisms of adenosine signaling in health and disease. Through rigorous investigation and experimentation, A1 inhibitors have the ability to shed light on adenosine receptor biology, unveiling new perspectives on the complexities of adenosine-mediated cellular responses. By elucidating the intricate interactions between A1 inhibitors and their target receptor, researchers can further refine their understanding of adenosine signaling pathways and their impact on various physiological processes.
Product NameCAS #Catalog #QUANTITYPriceCitationsRATING

Gambogic Acid

2752-65-0sc-200137
sc-200137A
sc-200137B
sc-200137C
sc-200137D
5 mg
25 mg
100 mg
500 mg
1 g
$87.00
$248.00
$427.00
$734.00
$1255.00
5
(1)

Gambogic Acid (CAS 2752-65-0) is a natural compound known for its inhibitory effect on A1, a subtype of adenosine receptors. It interacts with the A1 receptor, modulating its activity and potentially impacting cellular signaling pathways. This compound's ability to inhibit A1 makes it a valuable tool in studying A1 receptor function and its role in various physiological processes.

PD 116,948

102146-07-6sc-200115
sc-200115A
25 mg
100 mg
$124.00
$228.00
6
(0)

Also called DPCPX, this compound is a selective A1 receptor antagonist that has been widely used in experimental studies to block A1 receptor activation.

8-Cyclopentyl-1,3-dimethylxanthine

35873-49-5sc-210676
100 mg
$230.00
(0)

CPX is a non-selective adenosine receptor antagonist that includes A1 receptor inhibition.

GR 79236

124555-18-6sc-361197
sc-361197A
10 mg
50 mg
$235.00
$999.00
(0)

GR79236 is a potent and selective A1 receptor antagonist that has been studied for its potential as an analgesic and anti-inflammatory agent.