1. Malleron, J.L., et al. 1991. J. Med. Chem. 34: 2477-2483. 2. Doble, A., et al. 1992. Br. J. Pharmacol. 105: 27-36. 3. Heuillet, E., et al. 1996. Eur. J. Pharmacol. 314: 229-233.
抑制剂:
D4DR, 和 SR-2A.
物理状态 :
Solid
溶解度 :
Soluble in DMSO (100 mM).
保存 :
Store at room temperature
熔点 :
238.16° C (Predicted)
沸点 :
~641.1° C at 760 mmHg (Predicted)
密度 :
~1.3 g/cm3 (Predicted)
折射率 :
n20D 1.66 (Predicted)
IC50 :
Inositol phosphate formation evoked by 5-HT: IC50 = 7.76 nM