Molecular structure of L-703,606 oxalate, CAS Number: 351351-06-9
L-703,606 oxalate (CAS 351351-06-9)
Alternate Names:
cis-2-(Diphenylmethyl)-N-[(2-iodophenyl)methyl]-1-azabicyclo[2.2.2]octan-3-amine oxalate salt
Application:
L-703,606 oxalate is a selective nonpeptide NK1 tachykinin receptor antagonist
CAS Number:
351351-06-9
Molecular Weight:
598.50
Molecular Formula:
C27H29N2I•C2H2O4
For Research Use Only. Not Intended for Diagnostic or Therapeutic Use.
* Refer to Certificate of Analysis for lot specific data.
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Description
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SDS & Certificate of Analysis
L-703,606 oxalate represents a pivotal chemical entity in the landscape of receptor antagonism, specifically targeting the NK-1R (NK1 tachykinin receptor) with high potency and selectivity. As a non-peptide antagonist, this compound offers a significant advantage in terms of molecular stability and the ability to cross biological barriers, compared to peptide-based antagonists. The NK-1R, integral to the tachykinin system, is predominantly involved in the transmission of pain signals and the modulation of inflammatory responses within the central and peripheral nervous system, making it a target for the investigation of novel therapeutic strategies against pain and inflammation.
L-703,606 oxalate (CAS 351351-06-9) References
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Inhibitor of:
NK-1R.Ordering Information
| Product Name | Catalog # | UNIT | Price | Qty | FAVORITES | |
L-703,606 oxalate, 1 mg | sc-203095 | 1 mg | $107.00 | |||
L-703,606 oxalate, 5 mg | sc-203095A | 5 mg | $194.00 | |||
L-703,606 oxalate, 50 mg | sc-203095B | 50 mg | $1280.00 | |||
L-703,606 oxalate, 100 mg | sc-203095C | 100 mg | $2045.00 | |||
L-703,606 oxalate, 1 g | sc-203095D | 1 g | $9185.00 |