CAY10502 (CAS 888320-29-4)
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CAY10502 is a compound that is studied in various research applications, particularly due to its role as a chemical probe and inhibitor in biochemical pathways. It is a potent Calcium-dependent cytosolic PLA2 (cPLA2alpha) inhibitor with an IC50 value of 4.3 nM for the purified enzyme from human platelets. Additionally, it inhibits arachidonic acid mobilization from A23187-stimulated or TPA-stimulated human platelets with IC50 values of 570 and 0.9 nM, respectively. The compound′s effects on protein interactions and gene expression are also areas of interest, as understanding these can provide insights into cellular responses to external stimuli. Also, CAY10502 may be used in the exploration of molecular mechanisms underlying certain cellular functions and in the identification of novel targets for potential intervention strategies in various biological systems.
CAY10502 (CAS 888320-29-4) References
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Ordering Information
| Product Name | Catalog # | UNIT | Price | Qty | FAVORITES | |
CAY10502, 500 µg | sc-223866 | 500 µg | $44.00 | |||
CAY10502, 1 mg | sc-223866A | 1 mg | $81.00 | |||
CAY10502, 5 mg | sc-223866B | 5 mg | $337.00 | |||
CAY10502, 10 mg | sc-223866C | 10 mg | $591.00 |