Bufuralol hydrochloride (CAS 60398-91-6)
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Bufuralol hydrochloride, a benzofuran derivative, exhibits its biological activities primarily through beta-adrenergic blockade coupled with peripheral vasodilation mechanisms, implicating a multifaceted role in modulating cardiovascular dynamics. This compound′s interaction with the beta-adrenergic system demonstrates its capability to influence heart rate and vascular tone, which are pivotal in the study of cardiovascular function and its regulatory mechanisms. Furthermore, the metabolic processing of Bufuralol hydrochloride highlights its diastereomer selective metabolism, involving the cytochrome P450 enzymes CYP2D6 and CYP2C19, in the formation of 1-OH-Bufuralol. This selective metabolic pathway provides an insightful model for understanding the intricacies of cytochrome P450 enzyme-mediated metabolism and its implications in the stereoselective formation of metabolites, making Bufuralol hydrochloride a valuable compound for research in enzymology and pharmacokinetics within the realm of biochemical and cardiovascular studies.
Bufuralol hydrochloride (CAS 60398-91-6) References
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Ordering Information
| Product Name | Catalog # | UNIT | Price | Qty | FAVORITES | |
Bufuralol hydrochloride, 1 mg | sc-207384A | 1 mg | $176.00 | |||
Bufuralol hydrochloride, 2.5 mg | sc-207384B | 2.5 mg | $306.00 | |||
Bufuralol hydrochloride, 10 mg | sc-207384 | 10 mg | $849.00 | |||
Bufuralol hydrochloride, 25 mg | sc-207384C | 25 mg | $1799.00 | |||
Bufuralol hydrochloride, 100 mg | sc-207384D | 100 mg | $3689.00 |