GT 2016 is a high affinity H3 receptor antagonist (Ki = 43.8 nM). GT 2016 displays selectivity against H1 and H2 (IC50 > 10 μM). This compound displays no activity at histamine methyltransferase in vitro at concentrations up to 3 μM.
Soluble in DMSO (100 mM), and ethanol (100 mM).
Store at -20° C
H3 receptor : Ki= 43.8 nM
For Research Use Only. Not Intended for Diagnostic or Therapeutic Use.