UNQ9391 (serine protease 55) activators include a range of compounds that indirectly increase the protease's activity by inhibiting other proteases, which would otherwise degrade or negatively regulate UNQ9391. By acting as competitive or irreversible inhibitors of these regulatory proteases, they ensure that UNQ9391 retains its functional integrity and enzymatic activity. Some of these activators are synthetic inhibitors designed to target serine proteases specifically, thereby reducing competition for substrates and preventing inactivation of UNQ9391. Others, while not exclusively specific for serine proteases, provide broad-spectrum protection by binding to the active sites of various enzymes, which might interfere with the activity of UNQ9391. This inhibition strategy sustains the active state of UNQ9391, thus enhancing its overall proteolytic activity.
Further, certain activators are particularly potent in safeguarding UNQ9391 against degradation by inhibiting the proteasomes responsible for protein turnover, including those of serine proteases. Additional activators focus on preserving the activity of UNQ9391 by shielding it from the action of aspartic and cysteine proteases, which could otherwise lead to its inactivation.
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| Product Name | CAS # | Catalog # | QUANTITY | Price | Citations | RATING |
|---|---|---|---|---|---|---|
Benzamidine | 618-39-3 | sc-233933 | 10 g | $292.00 | 1 | |
A reversible inhibitor of trypsin-like proteases and serine proteases. Benzamidine enhances the activity of UNQ9391 by competitively inhibiting proteins that would otherwise inhibit UNQ9391, thereby increasing its functional activity. | ||||||
Phenylmethylsulfonyl Fluoride | 329-98-6 | sc-3597 sc-3597A | 1 g 100 g | $50.00 $697.00 | 92 | |
An irreversible inhibitor of serine proteases. PMSF acts to preserve the functionality of UNQ9391 by inhibiting proteases that would degrade or inactivate UNQ9391, thus indirectly increasing its activity. | ||||||
Aprotinin | 9087-70-1 | sc-3595 sc-3595A sc-3595B | 10 mg 100 mg 1 g | $112.00 $408.00 $3000.00 | 51 | |
A potent serine protease inhibitor that binds to and blocks the active sites of enzymes that could degrade UNQ9391. This inhibition protects UNQ9391 from inactivation, resulting in an overall increase in its activity. | ||||||
Leupeptin hemisulfate | 103476-89-7 | sc-295358 sc-295358A sc-295358D sc-295358E sc-295358B sc-295358C | 5 mg 25 mg 50 mg 100 mg 500 mg 10 mg | $73.00 $148.00 $316.00 $499.00 $1427.00 $101.00 | 19 | |
A reversible inhibitor of serine proteases. By inhibiting the action of serine protease inhibitors, indirectly maintains the active state of UNQ9391. | ||||||
Gabexate mesylate | 56974-61-9 | sc-215066 | 5 mg | $100.00 | ||
A synthetic inhibitor of various serine proteases. Indirectly enhances the activity of UNQ9391 by inhibiting proteases that would normally decrease the activity of UNQ9391. | ||||||
Nafamostat mesylate | 82956-11-4 | sc-201307 sc-201307A | 10 mg 50 mg | $82.00 $306.00 | 4 | |
A synthetic serine protease inhibitor that can indirectly increase the activity of UNQ9391 by inhibiting proteases that degrade or inactivate UNQ9391. | ||||||
Camostat mesylate | 59721-29-8 | sc-203867 sc-203867A sc-203867B sc-203867C sc-203867D sc-203867E | 10 mg 50 mg 500 mg 1 g 10 g 100 g | $43.00 $183.00 $312.00 $624.00 $2081.00 $4474.00 | 5 | |
A synthetic serine protease inhibitor that helps maintain the activity of UNQ9391 by preventing the degradation or inactivation by other proteases. | ||||||
Argatroban | 74863-84-6 | sc-201310 sc-201310A | 10 mg 50 mg | $117.00 $469.00 | 13 | |
A direct thrombin inhibitor that can indirectly increase the activity of UNQ9391 by inhibiting thrombin, a serine protease that may regulate the activity of UNQ9391. | ||||||
Bortezomib | 179324-69-7 | sc-217785 sc-217785A | 2.5 mg 25 mg | $135.00 $1085.00 | 115 | |
A proteasome inhibitor that can prevent the degradation of UNQ9391, thus indirectly increasing its functional activity. | ||||||
E-64 | 66701-25-5 | sc-201276 sc-201276A sc-201276B | 5 mg 25 mg 250 mg | $281.00 $947.00 $1574.00 | 14 | |
An irreversible inhibitor that targets cysteine proteases. By inhibiting cysteine proteases, E-64 indirectly preserves the functional state of UNQ9391. | ||||||