SEE ALSO...
| Product Name | CAS # | Catalog # | QUANTITY | Price | Citations | RATING |
|---|---|---|---|---|---|---|
Mifepristone | 84371-65-3 | sc-203134 | 100 mg | $61.00 | 17 | |
Mifepristone acts as a potent antagonist at progesterone receptors, disrupting the typical receptor-ligand interactions. Its unique structural features enable it to form stable complexes that inhibit receptor activation, thereby altering gene expression. The compound's lipophilic nature facilitates its diffusion across cellular membranes, enhancing its bioavailability. Additionally, Mifepristone's kinetic profile reveals rapid receptor binding and dissociation, influencing cellular responses through competitive inhibition. | ||||||
Guggulsterone | 95975-55-6 | sc-203990 sc-203990A | 10 mg 50 mg | $145.00 $615.00 | 1 | |
Guggulsterone functions as a selective modulator of progesterone receptors, exhibiting unique binding dynamics that influence receptor conformation. Its distinct molecular structure allows for specific interactions with the receptor's ligand-binding domain, promoting a nuanced regulatory effect on gene transcription. The compound's hydrophobic characteristics enhance its affinity for lipid membranes, facilitating cellular uptake. Furthermore, Guggulsterone's interaction kinetics suggest a slower dissociation rate, potentially leading to prolonged receptor engagement and sustained biological effects. | ||||||