Histamine H1 Receptor Activators
Santa Cruz Biotechnology now offers a broad range of Histamine H1 Receptor Activators. Histamine is an inflammatory mediator that is ubiquitously expressed and has a broad range of pharmacologic effects. The effects of histamine are mediated by a family of G protein-coupled receptors, the Histamine H1, H2, H3 and H4 Receptors. Histamine H1 Receptor Activators offered by Santa Cruz activate Histamine H1 Receptor and, in some cases, other inflammation and immune response related proteins. View detailed Histamine H1 Receptor Activator specifications, including Histamine H1 Receptor Activator CAS number, molecular weight, molecular formula and chemical structure, by clicking on the product name.
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| Product Name | CAS # | Catalog # | QUANTITY | Price | Citations | RATING |
|---|---|---|---|---|---|---|
2-(1,3-thiazol-2-yl)ethanamine dihydrochloride | 18453-07-1 | sc-282443 | 100 mg | $200.00 | ||
Known to be a potent activator of the H1 Receptor, with specificity towards this subtype. | ||||||
Histamine-α,α,β,β-d4 Dihydrochloride | 344299-48-5 | sc-218580 sc-218580A sc-218580B sc-218580C | 1 mg 2.5 mg 5 mg 10 mg | $430.00 $750.00 $1200.00 $2058.00 | ||
Histamine-α,α,β,β-d4 Dihydrochloride is characterized by its deuterated structure, which alters its isotopic composition, impacting its metabolic pathways and reaction kinetics. This compound engages with the Histamine H1 receptor through specific hydrogen bonding and hydrophobic interactions, enhancing its binding affinity. The presence of deuterium may influence the rate of enzymatic degradation, providing insights into receptor dynamics and signaling mechanisms. Its unique isotopic labeling allows for advanced tracking in biochemical studies. | ||||||
Betahistine Hydrochloride | 15430-48-5 | sc-210906 | 50 mg | $2290.00 | ||
Betahistine Hydrochloride exhibits a unique interaction profile with the Histamine H1 receptor, primarily through its ability to mimic histamine's structure, facilitating competitive binding. This compound's distinct molecular conformation enhances its affinity for the receptor, promoting specific conformational changes that influence downstream signaling pathways. Additionally, its solubility characteristics and stability in physiological conditions allow for nuanced studies of receptor activation and modulation, providing valuable insights into histaminergic signaling dynamics. | ||||||