GluR-5 Inhibitors
SEE ALSO...
| Product Name | CAS # | Catalog # | QUANTITY | Price | Citations | RATING |
|---|---|---|---|---|---|---|
Topiramate | 97240-79-4 | sc-204350 sc-204350A | 10 mg 50 mg | $107.00 $369.00 | ||
Topiramate acts as a selective modulator of the GluR5 receptor, engaging in specific hydrogen bonding interactions that stabilize its binding conformation. This interaction leads to a unique alteration in receptor dynamics, promoting a shift in ion permeability. The compound's affinity for the receptor is influenced by its stereochemistry, resulting in distinct kinetic profiles that affect the rate of receptor activation and desensitization, ultimately impacting synaptic plasticity. | ||||||
UBP 310 | 902464-46-4 | sc-361389 sc-361389A | 10 mg 50 mg | $169.00 $615.00 | 1 | |
UBP310 is a potent and selective antagonist of the GluR-5 receptor. It acts by competitively inhibiting glutamate binding, thus reducing receptor activation and subsequent neuronal excitation. | ||||||
UBP 296 | 745055-86-1 | sc-204366 sc-204366A | 1 mg 10 mg | $190.00 $900.00 | ||
UBP 296 functions as a selective antagonist of the GluR5 receptor, exhibiting unique electrostatic interactions that disrupt the receptor's conformational stability. This compound alters the receptor's ion channel kinetics, leading to a pronounced modulation of calcium influx. Its distinct molecular architecture allows for specific binding that influences downstream signaling pathways, thereby affecting neuronal excitability and synaptic transmission dynamics. | ||||||