Harada M, Yamashita A, Aburada M. J Pharm Soc Japan 92:750-756 (1972). Hirai A, Terano T, Hamazaki T et al. Throm Res. 31:29-40 (1983). Zhang WG, Zhang ZS. Acta Pharm Sinica 29:145-148 (1994).
抑制剂:
HSF3, LITAF, 和 TIMP-3.
激活剂:
TCP-1 ζ2.
外观 :
Crystalline
物理状态 :
Solid
溶解度 :
Soluble in water (<1 mg/ml at 25° C), methanol, DMSO (33 mg/ml at 25° C), and ethanol (33 mg/ml at 25° C).
保存 :
Store at room temperature
熔点 :
48-50° C (lit.)
沸点 :
154° C (lit.) at 20 mmHg
密度 :
~1.2 g/cm3 (Predicted)
折射率 :
n20D 1.54 (Predicted)
IC50 :
Sprague-Dawley rat lens alodse reductase : IC50 = >50 µM; Formation of advanced glycation end product : IC50 = >5 mM