Date published: 2026-10-24

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MRP2 抗体 (6D564): sc-71603

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说明书
  • MRP2 抗体 6D564 是小鼠单克隆 IgG1, 在3篇文献中引用,提供 500 µl supernatant
  • 免疫human物种的MRP2的氨基酸215-310
  • 推荐用于 human 来源的MRP2 WB, IP 和 IF检测; 不会与 MDR1, MRP1, MRP3 or MRP5产生交联反应
  • 目前,我们还没有完成MRP2 抗体 (6D564)的首选二抗检测试剂的鉴定。这项工作正在进行中。
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MRP2抗体(6D564)是一种IgG1小鼠单克隆MRP2抗体,通过WB、IP和IF检测人类来源的MRP2。MRP2抗体可以是非偶联的抗MRP2抗体形式。已知在人类癌症细胞中赋予多药耐药性的ABC转运蛋白大家族的两个成员是Mdr-1 P-糖蛋白和多药耐药蛋白MRP1。MRP1是一种完整的膜蛋白,包含MDR样核心、N端膜结合区和细胞质连接体,在各种脑细胞、肺、睾丸和外周血中表达。MRP基因家族还包括MRP2和MRP3,它们都是主要在肝细胞中表达的缀合物输出泵,MRP2也被命名为cMOAT(用于小管多特异性有机阴离子转运蛋白)。MRP2仅定位于心尖膜,并在正常肝细胞中以高水平组成性表达。相反,MRP3定位于基底外侧膜,在那里它还介导有机阴离子S-(2,4-二硝基苯基-)谷胱甘肽向膜的基底外侧的转运。MRP3通常以相对低于MRP2的水平表达,并且仅当MRP2通过顶膜的分泌受损时才增加。MRP6在肝脏和肾脏中高表达,而MRP4和MRP5在各种组织中检测到,但表达水平要低得多。

仅限研究使用。不适用于诊断和治疗用途。

Alexa Fluor® 是Molecular Probes Inc., OR., USA的商标

LI-COR®和 Odyssey® 是LI-COR Biosciences的注册商标

MRP2 抗体 (6D564) 参考文献:

  1. ABC药物转运蛋白:MDR1、MRP1和MRP2的遗传多态性和药理影响。  |  Kerb, R., et al. 2001. Pharmacogenomics. 2: 51-64. PMID: 11258197
  2. 黄酮类化合物和药物反应对ABC转运蛋白(P-糖蛋白、MRP2、BCRP)活性的调节。  |  Alvarez, AI., et al. 2010. J Pharm Sci. 99: 598-617. PMID: 19544374
  3. 药物对MRP2/Mrp2介导的雌二醇-17beta-葡萄糖醛酸苷转运的增强作用--简明综述。  |  Herédi-Szabó, K., et al. 2009. Chem Biodivers. 6: 1970-4. PMID: 19937833
  4. 4-苯丁酸调节肝小管MRP2的泛素化,降低血清总胆红素浓度。  |  Hayashi, H., et al. 2012. J Hepatol. 56: 1136-1144. PMID: 22245901
  5. 人鼠MRP2/Mrp2对他汀类药物的ATP依赖性转运。  |  Ellis, LC., et al. 2013. Toxicol Appl Pharmacol. 269: 187-94. PMID: 23562342
  6. CFTR 相关配体是 Mrp2 表达的负调控因子。  |  Li, M., et al. 2017. Am J Physiol Cell Physiol. 312: C40-C46. PMID: 27834195
  7. 肝移植后MRP2表达的改变和移植结果。  |  Yi, NJ., et al. 2018. Ann Surg Treat Res. 95: 249-257. PMID: 30402443
  8. 昼夜节律基因Bmal1控制肠道转运蛋白MRP2和药物处置。  |  Yu, F., et al. 2019. Theranostics. 9: 2754-2767. PMID: 31244920
  9. 环孢菌素A通过抑制PXR介导的CYP3A4/CYP3A5/MRP2途径诱导HepG2细胞内的细胞毒性。  |  Shang, S., et al. 2024. Drug Chem Toxicol. 47: 739-747. PMID: 38166548
  10. MRP1和cMOAT/MRP2介导的GSSG和谷胱甘肽结合物的排泄。  |  Suzuki, H. and Sugiyama, Y. 1998. Semin Liver Dis. 18: 359-76. PMID: 9875554

订购信息

产品名称产品编号规格价格数量收藏夹

MRP2 抗体 (6D564)

sc-71603
500 µl supernatant
$322.00

For Western Blot, is it recommended to use denatured or non-denatured conditions with MRP2 (6D564): sc-71603 antibody?

Asked by: TinTin
Thank you for your question. We recommend this antibody for use in denatured Western Blot conditions. It has not been validated for use in non-denatured conditions. Please contact our Technical Service Department for further details or inquiries.
Answered by: Technical Support
Date published: 2017-03-27
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Rated 5 out of 5 by dolphin11065 from greatgreat antibody work well in WB at 1:300, bladder cancer
Date published: 2017-07-06
Rated 5 out of 5 by DDanae from superbStrong band in WB in A-431 whole cell lysates, I'll continue to use it.
Date published: 2017-03-18
Rated 5 out of 5 by jenniferc from Strong and clearStrong and clear band produced with MRP2 Antibody (6D564)
Date published: 2017-01-25
Rated 4 out of 5 by JM from Western blot publication in HepG2Western blot publication in HepG2, SGC7901, HepG2/AS and SGC7901/AS cells. -SCBT Publication Review
Date published: 2015-05-02
Rated 4 out of 5 by CJ from WB: Single strong bands in JAR and AWB: Single strong bands in JAR and A-431 whole cell lysates. -SCBT QC
Date published: 2014-11-14
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MRP2 抗体 (6D564) is rated 4.6 out of 5 by 5.
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