Molecular structure of Rilmenidine hemifumarate, CAS Number: 207572-68-7
Rilmenidine hemifumarate (CAS 207572-68-7)
Alternate Names:
N-(Dicyclopropylmethyl)-4,5-dihydro-2-oxazolamine hemifumarate salt
Application:
Rilmenidine hemifumarate is a selective ligand for I1-imidazoline and α2-AR agonist
CAS Number:
207572-68-7
Molecular Weight:
238.29
Molecular Formula:
C10H16N2O•1/2C4H4O4
For Research Use Only. Not Intended for Diagnostic or Therapeutic Use.
* Refer to Certificate of Analysis for lot specific data.
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SDS & Certificate of Analysis
Rilmenidine hemifumarate is an imidazoline I1 binding site (I1BS)-selective ligand (Ki = 7.1 nM), with much weaker affinity for I2BS (Ki = 5.2 μM). Rilmenidine hemifumarate also acts as an α2-adrenoceptor (α2-AR) agonist. Unlike clonidine (sc-203002), rilmenidine hemifumarate has greater selectivity for I1BS relative to α2-AR.
Rilmenidine hemifumarate (CAS 207572-68-7) References
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AR, and Nischarin.Ordering Information
| Product Name | Catalog # | UNIT | Price | Qty | FAVORITES | |
Rilmenidine hemifumarate, 5 mg | sc-203680 | 5 mg | $110.00 | |||
Rilmenidine hemifumarate, 25 mg | sc-203680A | 25 mg | $550.00 |