EAT-4 activators represent a unique chemical class with intriguing properties and functions at the molecular level, mainly revolving around their interaction with a specific type of protein transporter. These activators are specially designed to target and modulate the activity of the EAT-4 protein, a type of vesicular glutamate transporter. EAT-4, a crucial component in the nervous system of some organisms, is primarily responsible for the packaging of glutamate into synaptic vesicles. This function is pivotal for the proper transmission of nerve signals, particularly in glutamatergic neurons, where glutamate acts as the primary excitatory neurotransmitter. The unique action mechanism of EAT-4 activators involves the enhancement of EAT-4's natural function, which results in an increased efficiency of glutamate packaging into vesicles. This heightened activity could have significant implications for the overall dynamics of synaptic transmission, influencing the rate and efficacy of nerve signal propagation.
The molecular structure of EAT-4 activators is characterized by their ability to bind selectively to the EAT-4 transporter. This selectivity is a result of their specific chemical composition, which is often tailored to match the binding sites on the EAT-4 protein. These activators typically have high affinity for these sites, ensuring effective modulation of the transporter's activity. In terms of chemical composition, EAT-4 activators are diverse, encompassing a range of structures from simple organic compounds to more complex molecular arrangements. This diversity allows for the fine-tuning of their properties, including solubility, stability, and the strength of interaction with the EAT-4 transporter. The development and study of EAT-4 activators are driven by a keen interest in understanding the fundamental processes governing neurotransmitter storage and release, particularly in relation to the glutamatergic system. By shedding light on these processes, EAT-4 activators contribute to a deeper understanding of the intricate mechanisms that underlie neural communication.
| Nome del prodotto | CAS # | Codice del prodotto | Quantità | Prezzo | CITAZIONI | Valutazione |
|---|---|---|---|---|---|---|
L-Glutamic Acid | 56-86-0 | sc-394004 sc-394004A | 10 g 100 g | $291.00 $566.00 | ||
Essendo il neurotrasmettitore primario che EAT-4 trasporta, un aumento del glutammato extracellulare potrebbe potenzialmente potenziare l'attività di EAT-4. | ||||||
Dihydrokainic acid | 52497-36-6 | sc-200442B sc-200442 sc-200442A | 1 mg 10 mg 50 mg | $108.00 $296.00 $896.00 | 3 | |
Un inibitore di alcuni trasportatori di glutammato; i suoi effetti sull'EAT-4 necessitano di ulteriori studi, ma potrebbe influenzare le dinamiche di segnalazione del glutammato. | ||||||
Riluzole | 1744-22-5 | sc-201081 sc-201081A sc-201081B sc-201081C | 20 mg 100 mg 1 g 25 g | $20.00 $189.00 $209.00 $311.00 | 1 | |
Noto per modulare la neurotrasmissione glutammatergica, il riluzolo potrebbe influenzare indirettamente la funzione dell'EAT-4. | ||||||
Ceftriaxone, Disodium Salt, Hemiheptahydrate | 104376-79-6 | sc-211050 sc-211050A | 1 g 5 g | $175.00 $440.00 | 1 | |
È stato dimostrato che gli antibiotici beta-lattamici regolano alcuni trasportatori di glutammato; il loro effetto sull'EAT-4 richiederebbe ulteriori indagini. | ||||||
Taurine | 107-35-7 | sc-202354 sc-202354A | 25 g 500 g | $47.00 $100.00 | 1 | |
La taurina è stata coinvolta nella modulazione dei sistemi neurotrasmettitoriali e potrebbe influenzare l'attività del trasportatore del glutammato. | ||||||
L-Theanine | 3081-61-6 | sc-204787 sc-204787A | 1 g 5 g | $57.00 $139.00 | 1 | |
La L-teanina, contenuta nel tè, influisce sulla neurotrasmissione glutammatergica, influenzando potenzialmente l'EAT-4 in modo indiretto. | ||||||
Memantine hydrochloride | 41100-52-1 | sc-203628 | 50 mg | $68.00 | 4 | |
Un antagonista dei recettori NMDA che modula la segnalazione glutammatergica, influenzando eventualmente l'attività dell'EAT-4. | ||||||