NPY5-R Inhibitors
SEE ALSO...
| Product Name | CAS # | Catalog # | QUANTITY | Price | Citations | RATING |
|---|---|---|---|---|---|---|
L-152,804 | 6508-43-6 | sc-203618 sc-203618A | 10 mg 50 mg | $185.00 $781.00 | ||
L-152,804 functions as a selective antagonist for the NPY5 receptor, exhibiting unique binding characteristics that disrupt receptor-ligand interactions. Its molecular structure allows for specific steric hindrance, effectively blocking receptor activation. The compound's kinetic profile reveals a rapid association and slower dissociation, which alters downstream signaling pathways. Additionally, L-152,804's interactions with membrane microdomains suggest a role in modulating receptor localization and function. | ||||||
CGP 71683 hydrochloride | 192322-50-2 | sc-203881 sc-203881A sc-203881B | 10 mg 50 mg 1 g | $209.00 $862.00 $1320.00 | ||
CGP 71683 hydrochloride acts as a selective antagonist for the NPY5 receptor, characterized by its unique ability to stabilize inactive receptor conformations. This compound exhibits a distinct affinity for specific binding sites, influencing receptor dynamics and altering the conformational landscape. Its interaction with lipid bilayers may affect membrane fluidity, potentially impacting receptor clustering and signaling efficiency. The compound's kinetic behavior indicates a nuanced modulation of receptor activity, contributing to its unique pharmacological profile. | ||||||
NTNCB hydrochloride | 486453-65-0 | sc-203655 sc-203655A | 10 mg 50 mg | $300.00 $781.00 | ||
NTNCB hydrochloride functions as a selective modulator of the NPY5 receptor, distinguished by its capacity to induce conformational changes that favor inactive states. This compound engages in specific hydrogen bonding and hydrophobic interactions, which can alter receptor accessibility and downstream signaling pathways. Its unique electronic properties may influence charge distribution, affecting interaction kinetics and receptor-ligand dynamics, thereby modulating physiological responses. | ||||||
LU AA33810 | 304008-29-5 | sc-295367 sc-295367A | 10 mg 50 mg | $169.00 $638.00 | ||
LU AA33810 functions as a selective NPY5 receptor antagonist, distinguished by its unique ability to induce conformational changes that hinder receptor activation. Its molecular structure allows for specific hydrogen bonding and hydrophobic interactions, which modulate the receptor's signaling pathways. The compound's kinetic profile reveals a slow dissociation rate from the receptor, enhancing its efficacy in altering downstream cellular processes. This specificity in binding dynamics offers valuable insights into receptor behavior and modulation. | ||||||
NPY 5RA972 | 439861-56-0 | sc-295945 sc-295945A | 10 mg 50 mg | $340.00 $850.00 | ||
NPY 5RA972 acts as a potent NPY5 receptor modulator, characterized by its ability to stabilize receptor conformations that inhibit signaling. Its unique molecular architecture facilitates specific electrostatic interactions and steric hindrance, effectively blocking receptor activation. The compound exhibits a distinctive binding affinity, leading to altered kinetics in receptor-ligand interactions, which can influence downstream signaling cascades and cellular responses. | ||||||
SB 408124 | 288150-92-5 | sc-361345 | 5 mg | $135.00 | ||
L-152,804 is an NPY5-R antagonist that can inhibit the function of NPY5-R by blocking the receptor and preventing its activation. | ||||||