Naltriben methanesulfonate CAS: 111555-58-9
MF: C26H25NO4•CH4O3S
MW: 511.59
A highly selective δ2 opioid receptor (DOR) antagonist.

Naltriben methanesulfonate (CAS 111555-58-9)

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Alternativa namn: NTB
Ansökan Naltriben methanesulfonate is a highly selective δ2 opioid receptor (DOR) antagonist
CAS Nr: 111555-58-9
Molekylvikt: 511.59
Molekylär formel: C26H25NO4•CH4O3S
For Research Use Only. Not Intended for Diagnostic or Therapeutic Use.
* Refer to Certificate of Analysis for lot specific data (including water content).

Naltriben methanesulfonate is a highly selective DOR (δ2 opioid receptor ) antagonist. Ligand binding assays show biphasic binding of the antagonist to the single receptor type.


Konferenser

Szekeres, P.G., Traynor, J.R., Delta opioid modulation of the binding of guanosine-5′-O-(3-[35S]thio)triphosphate to NG108-15 cell membranes: characterization of agonist and inverse agonist effects. J. Pharmacol. Exp. Ther. 283, 1276, (1997) Abstract Takemori, A.E., et al., Agonist and antagonist activities of ligands derived from naltrexone and oxymorphone. Life Sci. 50, 1491-1495, (1992) Abstract Miyamoto, Y., et al., Involvement of δ2 opioid receptors in the development of morphine dependence in mice. J. Pharmacol. Exp. Ther. 264, 1141-1145, (1993) Abstract

Physical State :
Solid
Solubility :
Soluble in DMSO (14 mg/ml at ~60° C).
LAGRING :
Store at -20° C
Melting Point :
277-278° C
Refractive Index :
n20D ~1.78 (Predicted)
Ki Data :
δ-opioid receptor: Ki= 0.01 nM; μ-opioid receptor: Ki= 19 nM; κ-opioid receptor: Ki= 152 nM
For Research Use Only. Not Intended for Diagnostic or Therapeutic Use.
WGK Germany :
3
RTECS :
PB9175000
PubChem CID :
MDL Number :
MFCD11046015
SMILES :
CS(=O)(=O)O.C1CC1CN2CCC34[[email protected]@H]5C6=C(C[[email protected]]3(C2CC7=C4C(=C(C=C7)O)O5)O)C8=CC=CC=C8O6

Download SDS (MSDS)

Certificate of Analysis

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