BNTX maleate (CAS 864461-31-4)

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Alternativa namn: 7-Benzylidenenaltrexone maleate

Ansökan BNTX maleate is a selective δ₁ opioid receptor (DOR) antagonist

CAS Nr: 864461-31-4

Molekylvikt: 545.59

Molekylär formel: C₂₇H₂₇NO₄•C₄H₄O₄

Kompletterande information: This is classified as a Dangerous Good for transport and may be subject to additional shipping charges.

For Research Use Only. Not Intended for Diagnostic or Therapeutic Use.
Available in US only.

* Refer to Certificate of Analysis for lot specific data (including water content).

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SDS & Certificate of Analysis

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BNTX maleate is a selective DOR (δ₁ opioid receptor ) antagonist. BNTX maleate inhibits neurogenic ion transport in porcine ileal mucosa.

Konferenser

1. Portoghese, P.S., Sultana, M., Nagase, H. and Takemori, A.E. 1992. A highly selective delta 1-opioid receptor antagonist: 7-benzylidenenaltrexone. Eur. J. Pharmacol. 218(1): 195-196. PMID: 1327826 2. Poonyachoti, S., Portoghese, P.S. and Brown, D.R. 20

Physical State :

Solid

Solubility :

Soluble in DMSO (100 mM), and water (10 mM).

LAGRING :

Desiccate at -20° C

Boiling Point :

828.5° C at 760 mmHg (Predicted)

Refractive Index :

n²⁰_D 1.73 (Predicted)

Ki Data :

Delta opioid receptor: K_i= 0.83 nM (rat); MOR-1: K_i= 1.9 nM (human); Kappa opioid receptor: K_i= 66 nM (Cavia porcellus)

For Research Use Only. Not Intended for Diagnostic or Therapeutic Use.
Available in US only.

RTECS :

QD2154700

PubChem CID :

6438353

MDL Number :

MFCD01310504

SMILES :

OC(=O)/C=C\\C(=O)O.Oc1ccc2CC3N(CC[[email protected]]45[[email protected]@H](Oc1c24)C(=O)/C(=C/c1ccccc1)/C[[email protected]]35O)CC1CC1

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Certificate of Analysis

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