Methimepip dihydrobromideA selective histamine H3 receptor agonist

Methimepip dihydrobromide (CAS 151070-80-3)

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Application: A selective histamine H3 receptor agonist
CAS Number: 151070-80-3
Purity: ≥98%
Molecular Weight: 341.09
Molecular Formula: C10H17N32HBr
* Refer to Certificate of Analysis for lot specific data (including water content).
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Methimepip dihydrobromide extremely selective histamine H3 receptor agonist [pKi values are 9.0, 5.7, < 5.0 and < 5.0 for Histamine H3 (hH3), Histamine H4 (hH4), Histamine H1(hH1) and Histamine H2(hH2) receptors respectively]. Potently inhibits EFS-evoked contractions of guinea pig ileum (pD2 = 8.26).


References

Kitbunnadaj et al (2005) N-substituted piperidinyl alkyl imidazoles: discovery of methimepip as a potent and selective histamine H3 receptor agonist. J.Med.Chem. 48 2100.

Physical State :
Solid
Solubility :
Soluble in water (100 mM).
Storage :
Desiccate at room temperature
For Research Use Only. Not Intended for Diagnostic or Therapeutic Use.
PubChem CID :
11313836
MDL Number :
MFCD09908999
SMILES :
CN1CCC(CC1)CC2=CN=CN2.Br.Br

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Certificate of Analysis

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