Flt-3 Inhibitor is a cell-permeable thienylcarboxamide compound that acts as a potent, ATP-competitive, and highly selective Flt-3/Flk-2 (Flt-3) inhibitor (IC50 = 42 nM) with little effect against a panel of 22 other kinases (IC50 ≥3 μM).
Patch, R.J., et al. 2006. Bioorg. Med. Chem. Lett. 16, 3282.
Soluble in water (<2 mg/ml), DMSO (15 mg/ml at 25° C), and ethanol (<1 mg/ml at 25° C).
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PatchPatch, RJ. et al. (PubMed 16580199) tested Flt-3 Inhibitor (2-(3,4-Dimethoxy-benzoylamino)-4,5,6,7-tetrahydro-benzo[b]thiophene-3-carboxylic acid amide) against several other derivatives. Found that the inhibitor was both potent and highly selective for Flt-3 at low concentrations (IC50 0.043 M). -SCBT Publication Review
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