Cantharidin is a potent small molecule inhibitor of PP2A (protein phosphatase 2A), used as an herbicide and a known toxin to animals. Cantharidin shows strong inhibition of PP2A (IC50=40 nM) compared to the analog Endothall (sc-201325), with Cantharidin displaying near complete inhibition of phosphatase activity.
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See how others have used Cantharidin. Click on the entry to view the PubMed entry .
PMID: # 14993658
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