Protein アクチベーター

Santa Cruz Biotechnology offers an extensive range of biochemicals with protein-interacting properties which are useful for studying protein function, cell signaling pathways and other biological processes. Protein Activators interact with specific proteins to activate or increase their function, thereby affecting cell signaling pathways. Browse our ChemCruz Biochemicals for Protein Activators here. Also see our Protein Inhibitors or Protein Substrates. Not finding the chemical you want? Click here to fill out a Chemical Request form.

製品名/アプリケーション CAS カタログ # 数量 価格 引用文献 レーティング
Batrachotoxin
A neurotoxic voltage-gated Na+ channel activator
23509-16-2 sc-201086
10 µg
$250.00
0
Lyso-PAF (C18)
A substrate for either PAF C-18 formation
74430-89-0 sc-203123
sc-203123A
5 mg
50 mg
$75.00
$342.00
0
Spermidine
A NOS1 inhibitor and NMDA and T4 polynucleotide kinase activator
124-20-9 sc-215900
sc-215900A
1 g
5 g
$32.00
$109.00
0
Camptothecin
A reversible Mitochondrial Topo I inhibitor shown to exhibit antitumor activity
7689-03-4 sc-200871
sc-200871A
50 mg
250 mg
$46.00
$168.00
11
Other image(s) available
MPEP hydrochloride
A selective antagonist of the mGluR5 receptor
96206-92-7 sc-279454
sc-279454A
50 mg
10 mg
$495.00
$125.00
0
CGS 20625
A central benzodiazepine receptor partial agonist
111205-55-1 sc-203545
sc-203545A
10 mg
50 mg
$169.00
$712.00
0
Benzylimidazole
An inducer of various cytochrome P-450 isozymes and inhibitor of thromboxane A2 synthase
4238-71-5 sc-200530
sc-200530A
25 g
5 g
$130.00
$40.00
0
PSY-279
A Transient Receptor Potential Vanilloid 1 agonist and amide based RTX analog
289903-41-9 sc-202780
sc-202780A
1 mg
5 mg
$55.00
$218.00
0
Fumonisin B1
A serine and threonine phosphatase inhibitor
116355-83-0 sc-201395
sc-201395A
1 mg
5 mg
$70.00
$304.00
4
C16 Ceramide (N-Palmitoylsphingosine, D-erythro)
An endogenous ceramide
24696-26-2 sc-201379
sc-201379A
5 mg
25 mg
$62.00
$273.00
1
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Resveratrol
A natural phenolic antioxidant that is a potent activator of SIRT1 and inhibitor of Cox-1
501-36-0 sc-200808
sc-200808A
100 mg
500 mg
$53.00
$175.00
2
Muraglitazar
A peroxisome proliferator-activated receptor agonist
331741-94-7 sc-211931
1 mg
$280.00
1
Taurine
A compound that Inhibits lipid peroxidation
107-35-7 sc-202354
25 g
$30.00
0
R(-)-alpha-Methylhistamine dot 2HBr
A potent and selective histamine H3 agonist
868698-49-1 sc-471364
10 mg
$165.00
0
Diminazene Aceturate
An anti-protozoal and anti-trypanosomal compound
908-54-3 sc-205651
sc-205651A
1 g
5 g
$85.00
$340.00
3
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Tenovin-6
An inhibitor of SIRT1, SIRT2, and SIRT3 and activator of p53
1011557-82-6 sc-224296
sc-224296A
1 mg
5 mg
$262.00
$1,185.00
7
CV 1808
An Adenosine A2-R agonist
53296-10-9 sc-203556
sc-203556A
10 mg
50 mg
$79.00
$299.00
0
Azelaoyl-PAF
A PPARγ agonist
354583-69-0 sc-221278
sc-221278A
1 mg
5 mg
$200.00
$440.00
0
CGS 12066B dimaleate
A selective SR-1B agonist
109028-10-6 sc-201106
sc-201106A
10 mg
50 mg
$113.00
$349.00
0
4-Nitrophenethyl bromide
A GST T1-1 substrate
5339-26-4 sc-238931
sc-238931A
25 g
5 g
$149.00
$47.00
0
PGJ2 (Prostaglandin J2)
A Prostaglandin D2 metabolite that has shown potent anti-neoplastic and antiviral activity
60203-57-8 sc-201248
sc-201248A
1 mg
10 mg
$224.00
$1,821.00
0
Leelamine HCl
A weak CB1 receptor agonist and PDK inhibitor
1446-61-3 sc-200375
sc-200375A
10 mg
50 mg
$162.00
$520.00
0
ZD 7114 hydrochloride
A β1-adrenoceptor agonist
129689-30-1 sc-361417
sc-361417A
5 mg
25 mg
$109.00
$440.00
0
PNU 22394 hydrochloride
A potent SR-2C agonist and partial SR-2A/SR-2B agonist
15923-78-1 sc-204851
sc-204851A
10 mg
50 mg
$125.00
$495.00
0
Pindolol
A SR-1A/SR-1B antagonist
13523-86-9 sc-204847
100 mg
$55.00
0
MDL 72832 hydrochloride
A post-synaptic 5-HT1A agonist
113777-33-6 sc-204070
sc-204070A
10 mg
50 mg
$125.00
$560.00
0
Taprostene
A highly selective agonist of the prostanoid receptor IP1
108945-35-3 sc-215940
sc-215940A
1 mg
5 mg
$179.00
$645.00
0
(2S)-2-Ethyl-8-methyl-1-thia-4,8-diazaspiro[4,5]decan-3-one
A M1 muscarinic agonist
503431-81-0 sc-206582
5 mg
$250.00
0
AM 1172
A potent and selective inhibitor of anandamide uptake and FAAH
251908-92-6 sc-202456
sc-202456A
10 mg
50 mg
$200.00
$650.00
0
Naphtho[1,2-d]thiazol-2-ylamine
CAS: 40172-65-4, MF: C11H8N2S, MW: 200.26
40172-65-4 sc-279906
1 g
$245.00
0
N-(Methyl-d3)-N'-nitrosopiperazine
sc-218973
25 mg
$250.00
0
(+/-)-Anatoxin A Fumarate
A cyanotoxin agonist of AChR
64285-06-9 sc-200185
1 mg
$225.00
0
WAY 200070
A selective ERβ agonist
440122-66-7 sc-301977
sc-301977A
10 mg
50 mg
$111.00
$435.00
0
Lobeline hydrochloride
An AChR agonist
134-63-4 sc-203114
sc-203114A
50 mg
1 g
$20.00
$106.00
0
CX546
An AMPA receptor potentiator and GluR activator
215923-54-9 sc-205278
sc-205278A
10 mg
50 mg
$190.00
$653.00
0
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EB 1089
A vitamin D receptor agonist and potent inhibitor of PTH-rP
134404-52-7 sc-358831
1 mg
$169.00
0
Methyl Phytoprostane B1 (Type I) (racemic)
An inducer of GST (glutathione-S-transferase)
sc-221931
5 mg
$267.00
0
Corticotropin
16960-16-0 sc-278882
sc-278882A
250 µg
1 mg
$68.00
$195.00
0
Adenosine 5prime-Monophosphate, Disodium Salt
A nucleotide involved in the reactions of cellular energy transfers
4578-31-8 sc-202444
5 g
$64.00
0
PK 11195
A peripheral benzodiazepine antagonist
85532-75-8 sc-203199
sc-203199A
10 mg
50 mg
$79.00
$304.00
0
Indoxyl sulfate potassium salt
An agonist for the human aryl hydrocarbon receptor (AHR)
2642-37-7 sc-255218
sc-255218A
250 mg
1 g
$68.00
$137.00
0
ET-18-OCH3
An inhibitor of phosphatidylinositol specific PLC & PKC
77286-66-9 sc-201021
sc-201021A
sc-201021B
5 mg
25 mg
50 mg
$50.00
$100.00
$150.00
1
rac-2-Ethoxy-3-octadecanamido-1-propylphosphocholine
A protein kinase C inhibitor
163702-18-9 sc-215787
25 mg
$480.00
0
PHA 568487
An agonist of AChR α7
527680-56-4 sc-204186
sc-204186A
10 mg
50 mg
$135.00
$575.00
0
SC9
A Protein kinase C (PKC) activator in the presence of Ca2+
102649-78-5 sc-202336
sc-202336A
sc-202336B
1 mg
5 mg
50 mg
$30.00
$64.00
$560.00
0
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(S)-Pramipexole Dihydrochloride
A D2DR and D3DR agonist
104632-25-9 sc-212895
10 mg
$84.00
0
Vidarabine
A neurotransmitter that acts as the preferred endogenous agonist at all adenosine receptor subtypes
5536-17-4 sc-205881
sc-205881A
100 mg
500 mg
$46.00
$129.00
1
Resiniferatoxin
A diterpenoid stimulator of substance P release
57444-62-9 sc-24015
sc-24015A
1 mg
5 mg
$122.00
$450.00
12
PAF C-16
A PAF-R, MAP kinase, and MAP kinase kinase activator
74389-68-7 sc-201009
sc-201009A
5 mg
25 mg
$58.00
$224.00
0
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Oleylethanolamide
An activator of Neu/ErbB2 receptors and a mediator of p38 and JNK kinases
111-58-0 sc-201400
sc-201400A
10 mg
50 mg
$55.00
$219.00
0
Bromocriptine mesylate
A selective D2 and D3 dopamine receptor agonist and NOS1 inhibitor
22260-51-1 sc-200395
sc-200395A
100 mg
500 mg
$72.00
$295.00
0
PETCM
A caspace-3 activator in cell extracts
10129-56-3 sc-202279
sc-202279A
10 mg
50 mg
$30.00
$82.00
0
L-694,247
A highly potent and selective SR-1D agonist
137403-12-4 sc-361223
sc-361223A
10 mg
50 mg
$179.00
$756.00
0
R(+)-7-Hydroxy-DPAT hydrobromide
Is a selective D3DR agonist
82730-72-1 sc-253356
5 mg
$115.00
0
PB 28 dihydrochloride
A high affinity selective σ2 receptor agonist
172906-90-0 sc-204834
sc-204834A
10 mg
50 mg
$129.00
$548.00
0
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SAG
A potent agonist of Hedgehog (Hh) signalling
912545-86-9 sc-212905
sc-212905A
1 mg
5 mg
$150.00
$525.00
3
Oxotremorine Sesquifumarate
An M2 and M4 Muscarinic acetylcholine receptor agonist
17360-35-9 sc-200170
sc-200170A
100 mg
500 mg
$52.00
$207.00
0
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Zaprinast (MB 22948)
An inhibitor of cGMP-specific phosphodiesterase
37762-06-4 sc-201206
sc-201206A
25 mg
100 mg
$59.00
$192.00
6
PEPA
An allosteric potentiator of AMPA desensitization
141286-78-4 sc-204178
sc-204178A
10 mg
50 mg
$125.00
$560.00
0
Quercetin
A PI 3-kinase inhibitor, GPR30 activator, and apoptosis inducer
117-39-5 sc-206089
sc-206089A
sc-206089B
100 mg
500 mg
25 g
$10.00
$15.00
$39.00
3
Kahweol acetate
An inducer of glutathione S-transferase (GST)
81760-47-6 sc-228383
sc-228383A
10 mg
25 mg
$276.00
$451.00
1
(+/-)-Epibatidine
A particularly potent AChR agonist
140111-52-0 sc-200177
sc-200177A
1 mg
5 mg
$62.00
$251.00
0
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Calpeptin
A calpain-2, cathepsin L, and calpain-1 inhibitor
117591-20-5 sc-202516
sc-202516A
10 mg
50 mg
$107.00
$428.00
10
(2S,4R)-gamma-Hydroxyglutamic acid
A glutamate derivative
2485-33-8 sc-283521
sc-283521A
10 mg
50 mg
$143.00
$568.00
0
Mirabegron
A β3 adrenergic receptor agonist of bladder muscles
223673-61-8 sc-211912
500 mg
$350.00
0
PBDA
A mGluR3-selective agonist and an inhibitor of glutamate carboxypeptidase II
229472-51-9 sc-222128
sc-222128A
1 mg
5 mg
$38.00
$150.00
0
Y-27152
A prodrug of the KATP (Kir6) channel opener Y-26763
127408-30-4 sc-204407
sc-204407A
10 mg
50 mg
$189.00
$796.00
0
alpha-Carboline-15N2 N-Oxide
sc-220428
1 mg
$300.00
0
Cotinine N-beta-D-Glucuronide
A major metabolite of Nicotine derivative
139427-57-9 sc-211139
1 mg
$300.00
1
PNU-282987 hydrate
A highly selective AChR α7 agonist
123464-89-1 (anhydrous) sc-301554
10 mg
$133.00
0
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CTPB
A potent p300 HAT activator
586976-24-1 sc-202558
sc-202558A
1 mg
5 mg
$46.00
$134.00
2
Ser-Leu-Ile-Gly-Arg-Leu-amide trifluoroacetate salt
A selective PAR2 peptide agonist
171436-38-7 (non-salt) sc-301799
1 mg
$77.00
0
R-(-)-Glucoraphanin potassium salt
A modulator of hepatic cytochrome P450 and phase II conjugation activity
21414-41-5 (non-salt) sc-359618
10 mg
$263.00
0
Neuromedin B, porcine
An endogenous activator for the NMBR (neuromedin B receptor)
87096-84-2 sc-394391
1 mg
$160.00
0
1-Methyl-4-imidazoleacetic acid hydrochloride
A metabolite
35454-39-8 sc-222712
sc-222712A
10 mg
250 mg
$60.00
$600.00
0
Paeoniflorin
A glycoside that activates Adenosine A1-R
23180-57-6 sc-204827
sc-204827A
sc-204827B
1 mg
5 mg
100 mg
$20.00
$80.00
$300.00
0
PGI2 dot Na (Prostaglandin I2 dot Na, Prostacyclin)
An eiconasoid shown to induce vasodilation and inhibit platelet aggregation
61849-14-7 sc-201231
sc-201231A
1 mg
10 mg
$79.00
$615.00
2
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Ghrelin (human)
An endogenous peptide GHS-R agonist
258279-04-8 sc-364689
0.5 mg
$168.00
0
12-epi Leukotriene B4
A leukotriene with less affinity than LTB4 at LTB4 receptors
83709-73-3 sc-204980
sc-204980A
25 µg
50 µg
$176.00
$334.00
0
Hyperforin dicyclohexylammonium salt
An inhibitor of monoamine uptake and TRPC6 agonsit
238074-03-8 sc-202178
sc-202178A
500 µg
1 mg
$134.00
$235.00
0
Uridine-5prime-diphosphoglucose, disodium salt
A biosynthetic product from the reaction of UTP and glucose-1-phosphate catalyzed by the enzyme uridyl transferase
117756-22-6 sc-296687
sc-296687A
100 mg
1 g
$70.00
$248.00
0
Dihydrolipoic acid
The reduced form of lipoic acid, increases ROS and NO levels and activates caspase-9 and caspase-3
462-20-4 sc-207581
sc-207581A
25 mg
100 mg
$30.00
$75.00
3
(-)-Indolactam V
A protein kinase C activator; also can direct the differentiation of human ESCs
90365-57-4 sc-202182
300 µg
$163.00
1
Linoleic Acid
A fatty acid with cytotoxic activity that influences the inflammatory process
60-33-3 sc-200788
sc-200788A
100 mg
1 g
$23.00
$52.00
1
CB 65
A high affinity and selective cannabinoid CB2 receptor agonist
913534-05-1 sc-361134
sc-361134A
10 mg
50 mg
$185.00
$781.00
0
Betulinic Acid
A cytotoxic, cell apoptosis causing agent that upregulates caspase-8
472-15-1 sc-200132
sc-200132A
25 mg
100 mg
$108.00
$325.00
0
Lonidamine
It elicits cell apoptosis and blocks CFTR Cl- channel
50264-69-2 sc-203115
sc-203115A
5 mg
25 mg
$101.00
$350.00
0
Deltorphin I
A δ opioid receptor agonist.
122752-15-2 sc-396073
1 mg
$85.00
0
Varenicline Tartrate
An AChR α4β2 partial agonist
375815-87-5 sc-208481
sc-208481A
sc-208481B
10 mg
50 mg
100 mg
$179.00
$825.00
$1,200.00
0
CBiPES hydrochloride
A selective positive allosteric modulator of the mGluR-2
856702-40-4 sc-358830
sc-358830A
10 mg
50 mg
$145.00
$645.00
0
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5-Nonyloxytryptamine oxalate
A selective agonist for SR-1B
157798-13-5 sc-203480
sc-203480A
10 mg
50 mg
$145.00
$615.00
0
Adenosine 5prime-Diphosphate Potassium Salt
A nucleotide that is widely distributed in nature
72696-48-1 sc-202443
sc-202443A
1 g
5 g
$50.00
$190.00
0
WAY 629 hydrochloride
A selective SR-2C agonist
57756-45-3 sc-204393
sc-204393A
10 mg
50 mg
$129.00
$548.00
0
1-Acetyl-4-methylpiperazine hydrochloride
An AChR agonist acetylcholine analog
60787-05-5 sc-203759
sc-203759A
10 mg
50 mg
$115.00
$473.00
0
Aceclidine Hydrochloride
A non-selective muscarinic acetylcholine receptor partial agonist
6109-70-2 sc-210735
1 g
$300.00
0
Naratriptan Hydrochloride
143388-64-1 sc-212362
10 mg
$56.00
0
DMAB-anabaseine dihydrochloride
A neuronal AChR partial agonist
32013-69-7 sc-203568
10 mg
$155.00
0
PNU 142633
A high affinity SR-1D agonist
187665-65-2 sc-204204
10 mg
$205.00
0
Adenosine 3prime,5prime-cyclic monophosphate sodium salt monohydrate
A PKA (protein kinase A) activator
37839-81-9 sc-291840
sc-291840A
25 mg
100 mg
$26.00
$62.00
0
Lipopolysaccharide, E. coli J5
An E. coli mutant that stimulates the activity of inducible NO synthase
sc-221854
5 mg
$159.00
0
(+)-15-epi Cloprostenol
A synthetic analog of prostaglandin F2α
54276-22-1 sc-205019
sc-205019A
1 mg
5 mg
$78.00
$352.00
0
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BEC, Hydrochloride
A competitive transition state inhibitor of arginases I and II
sc-221291
5 mg
$345.00
0
SC10
A protein kinase C (PKC) activator
102649-79-6 sc-202335
sc-202335A
1 mg
5 mg
$20.00
$50.00
0
Prostaglandin F2alpha
A potent smooth muscle contricting prostaglandin shown to inhibit adipocyte differentiation
551-11-1 sc-203219
1 mg
$81.00
0
Isatin
An endogenous monoamine oxidase inhibitor
91-56-5 sc-205721
sc-205721A
100 g
500 g
$63.00
$276.00
0
GW 3965 hydrochloride
A liver X receptor (LXR) activator
405911-17-3 sc-224011
sc-224011A
5 mg
25 mg
$134.00
$465.00
0
9-Nitrooleate
An activator of PPARγ
875685-44-2 sc-204632
sc-204632A
50 µg
100 µg
$50.00
$80.00
0
IB-MECA
A potent and selective Adenosine A3-R agonist
152918-18-8 sc-224020
sc-224020A
5 mg
25 mg
$266.00
$1,095.00
0
Fluprostenol isopropyl ester
A prodrug PGFR agonist
157283-68-6 sc-205327
sc-205327A
1 mg
5 mg
$106.00
$465.00
0
JYL-273
A potent TRPV1 agonist with reported high potency over capsaicin
289902-71-2 sc-202678
sc-202678A
1 mg
5 mg
$48.00
$192.00
0
Bourgeonal
A potent hOR17-4 receptor agonist
18127-01-0 sc-210959
10 mg
$220.00
0
Other image(s) available
CL 316243 disodium salt
A β3-AR agonist
151126-84-0 sc-203895
sc-203895A
10 mg
50 mg
$220.00
$720.00
2
Other image(s) available
Proxyfan oxalate
A high affinity histamine H3 receptor ligand
177708-09-7 sc-204867
sc-204867A
10 mg
50 mg
$139.00
$585.00
0