Peptide Receptor Ligands

Santa Cruz Biotechnology now offers a broad range of Peptide Receptor Ligands. Peptide Receptors are transmembrane proteins that can be activated or inhibited by peptide ligands. Dysfunction in these contribute to certain cardiovascular, endocrine, and metabolic disorders. Our popular products such as TNF-α Antagonist, SLIGRL-NH2, and 2-Furoyl-LIGRLO-amide trifluoroacetate salt are typically available for immediate shipment. View detailed information on our Peptide Receptor Ligands by clicking on the product name.

indicates a highly recommended product based on customer preference.

PRODUCT NAME/Application CAS Catalog # QUANTITY Price Citations RATING
SU 4312
A potent and selective VEGFR (Flk/Flt) inhibitor
5812-07-7 sc-200637
sc-200637A
5 mg
25 mg
$87.00
$312.00
1
PGE1 (Prostaglandin E1)
A major prostaglandin that affects protein kinase C (PKC), calcium movement, and adenylate cyclase
745-65-3 sc-201223
sc-201223A
1 mg
10 mg
$22.00
$135.00
0
CCR2 Antagonist
A highly potent CKR-2B (CCR2) receptor antagonist
445479-97-0 sc-202525
5 mg
$254.00
14
VEGFR2 Kinase Inhibitor III
A VEGFR2, Met, RET, PDGFR, and ALK inhibitor
204005-46-9 sc-202851
5 mg
$77.00
4
L-732,138
A selective competitive antagonist of the tachykinin NK1 receptors
148451-96-1 sc-203437
sc-203437A
10 mg
50 mg
$85.00
$415.00
0
A-71623
A potent CCK agonist with 1200-fold selectivity over the CCK2 receptor
130408-77-4 sc-203487
1 mg
$279.00
1
(+/-)-AC 7954 hydrochloride
A potent agonist of the GPR14 (urotensin II receptor)
477313-09-0 sc-203491
5 mg
$141.00
0
AG 045572
A selective gonadotropin-releasing hormone (GnRH) receptor antagonist
263847-55-8 sc-203499
sc-203499A
1 mg
10 mg
$105.00
$164.00
0
APC 366
An elective inhibitor of the mast cell tryptase
158921-85-8 sc-203516
5 mg
$229.00
0
AQ-RA 741
A high affinity selective mAChR M2 antagonist
123548-16-3 sc-203517
sc-203517A
10 mg
50 mg
$135.00
$575.00
0
BIIE 0246
A selective and competitive NPY2-R antagonist
246146-55-4 sc-203530
sc-203530A
1 mg
10 mg
$155.00
$329.00
1
BQ 788 sodium salt
A selective Endothelin receptor B (ETBR) antagonist
156161-89-6 sc-203534
1 mg
$214.00
1
Devazepide
A potent CCK (cholecystokinin) inhibitor
103420-77-5 sc-203562
sc-203562A
10 mg
50 mg
$172.00
$970.00
0
L-152,804
A potent, selective non-peptide NPY5-R receptor antagonist
6508-43-6 sc-203618
sc-203618A
10 mg
50 mg
$185.00
$781.00
0
L-803,087 trifluoroacetate
A potent and selective sst4 agonist
217480-26-7 sc-203619
10 mg
$279.00
0
NTNCB hydrochloride
A competitive non-peptidic NPY5-R antagonist
486453-65-0 sc-203655
sc-203655A
10 mg
50 mg
$185.00
$781.00
0
SCH 79797 dihydrochloride
A strong, selective non-peptide Thrombin R inhibitor
1216720-69-2 sc-203693
sc-203693A
10 mg
50 mg
$205.00
$865.00
3
ST 91
An α2-adrenoceptor agonist
4749-61-5 sc-203703
sc-203703A
10 mg
50 mg
$129.00
$548.00
0
SUN-B 8155
A selective calcitonin receptor agonist
345893-91-6 sc-203704
sc-203704A
10 mg
50 mg
$181.00
$681.00
0
(1R,1primeS,3primeR/1R,1primeR,3primeS)-L-054,264
A selective somatostatin sst2 receptor agonist
208706-12-1 sc-203766
sc-203766A
1 mg
10 mg
$115.00
$245.00
0
AC 55541
A selective protease-activated receptor 2 agonist
916170-19-9 sc-203799
sc-203799A
5 mg
25 mg
$132.00
$520.00
0
Antalarmin hydrochloride
A non-peptide CRF-RI receptor antagonist
220953-69-5 sc-203820
sc-203820A
10 mg
50 mg
$186.00
$640.00
0
BAY-u 3405
A suppresor PGD2-induced migration of human eosinophils
116649-85-5 sc-203834
sc-203834A
10 mg
50 mg
$185.00
$781.00
0
BIBO 3304 trifluoroacetate
A high affinity NPY1-R antagonist
191868-14-1 sc-203841
sc-203841A
10 mg
50 mg
$295.00
$1,215.00
1
BIBP 3226 trifluoroacetate
An NPY1-R & NPFF2 receptor inhibitor
1068148-47-9 sc-203842
sc-203842A
1 mg
10 mg
$130.00
$299.00
0
BMS 193885
A competitive NPY1-R antagonist
186185-03-5 sc-203848
sc-203848A
10 mg
50 mg
$235.00
$906.00
0
BU 239 hydrochloride
A potent, selective imidazoline I2 receptor ligand
1217041-98-9 sc-203859
sc-203859A
10 mg
50 mg
$139.00
$585.00
0
CGP 71683 hydrochloride
A potent non-peptide NPY5-R antagonist
192322-50-2 sc-203881
sc-203881A
sc-203881B
10 mg
50 mg
1 g
$199.00
$825.00
$1,185.00
0
EMD 66684
A potent non-peptidic antagonist of the AT1 receptor
187683-79-0 sc-203941
sc-203941A
10 mg
50 mg
$179.00
$760.00
0
IRL-2500
Potent endothelin receptor antagonist
169545-27-1 sc-204018
sc-204018A
10 mg
50 mg
$225.00
$772.00
0
L-168,049
A non-peptidyl human glucagon receptor antagonist
191034-25-0 sc-204034
sc-204034A
10 mg
50 mg
$165.00
$700.00
0
L-368,899 hydrochloride
A non-peptide Oxytocin Receptor Inhibitor
148927-60-0 sc-204037
sc-204037A
1 mg
10 mg
$139.00
$299.00
0
L-371,257
A potent oxytocin receptor inhibitor
162042-44-6 sc-204038
10 mg
$239.00
0
L-692,585
A non-peptidyl GHS R1 acticvator
145455-35-2 sc-204043
10 mg
$245.00
0
L-817,818
A non-peptide somatostatin subtype-5 receptor agonist
217480-27-8 sc-204048
10 mg
$279.00
0
MDL 72832 hydrochloride
A post-synaptic 5-HT1A agonist
113777-33-6 sc-204070
sc-204070A
10 mg
50 mg
$145.00
$605.00
0
NBI 27914 hydrochloride
A selective corticotropin-releasing factor 1 (CRF-RI) inhibitor
184241-44-9 sc-204119
sc-204119A
10 mg
50 mg
$115.00
$510.00
0
Nebivolol hydrochloride
A highly selective β1-adrenoceptor antagonist
152520-56-4 sc-204122
sc-204122A
10 mg
50 mg
$139.00
$224.00
0
PD 135158
A selective CCK-BR antagonist used for research purposes
130325-35-8 sc-204163
sc-204163A
10 mg
50 mg
$235.00
$992.00
0
PD 168368
A NMBR (Neuromedin B) antagonist
204066-82-0 sc-204166
sc-204166A
1 mg
10 mg
$140.00
$300.00
1
PD 176252
A GRPR and NMBR inhibitor
204067-01-6 sc-204171
10 mg
$245.00
0
SDZ NKT 343
A human tachykinin NK1 antagonist receptor
180046-99-5 sc-204274
10 mg
$255.00
0
SR 12813
A PXR agonist that activates the farnesoid X receptor (FXR) at μM concentrations
126411-39-0 sc-204296
sc-204296A
10 mg
50 mg
$87.00
$331.00
0
SR 142948
A potent non-peptidic neurotensin receptor inhibitor
184162-64-9 sc-204297
sc-204297A
1 mg
10 mg
$119.00
$255.00
0
SR 27897
An effective non-peptide antagonist of CCK
136381-85-6 sc-204298
sc-204298A
10 mg
50 mg
$179.00
$7,335.00
0
SR 49059
A potent and selective AVP Receptor V1a antagonist
150375-75-0 sc-204300
10 mg
$305.00
0
Sulfisoxazole
An ETAR antagonist
127-69-5 sc-204313
50 mg
$65.00
0
T 98475
A GnRH receptor antagonist
192887-28-8 sc-204318
1 mg
$199.00
0
Taltirelin
A synthetic thyrotropin-releasing hormone analog
103300-74-9 sc-204319
sc-204319A
1 mg
10 mg
$105.00
$225.00
0
TCS OX2 29
An inhibitor of the orexin R-2 receptor
372523-75-6 sc-204329
sc-204329A
10 mg
50 mg
$185.00
$781.00
0
THIQ
A selective melanocortin 4 receptor agonist
312637-48-2 sc-204343
1 mg
$205.00
0
Tramiprosate
A sulfated glycosaminoglycan mimic that targets amyloid β
3687-18-1 sc-204353
50 mg
$37.00
0
UBP 296
A selective GluR5-subunit containing kainate receptor antagonist
745055-86-1 sc-204366
sc-204366A
10 mg
50 mg
$179.00
$825.00
0
WIN 64338 hydrochloride
A bradykinin B2 R Inhibitor
163727-74-0 sc-204398
sc-204398A
10 mg
50 mg
$134.00
$756.00
0
YM 022
A highly potent and selective non-peptide CCK-BR silent antagonist
145084-28-2 sc-204409
sc-204409A
10 mg
50 mg
$175.00
$739.00
0
PD 160170
A potent and selective non-peptide NPY1-R antagonist
181468-88-2 sc-204836
sc-204836A
10 mg
50 mg
$155.00
$660.00
0
RO 90-7501
An inhibitor of amyloid β42 fibril assembly
293762-45-5 sc-204891
sc-204891A
10 mg
50 mg
$155.00
$660.00
0
RP 67580
A selective antagonist of the tachykinin NK1 receptor
135911-02-3 sc-204894
sc-204894A
10 mg
50 mg
$209.00
$880.00
3
CI 988
A selective and effective antagonist of CCK-BR
130332-27-3 sc-205244
sc-205244A
10 mg
50 mg
$199.00
$1,120.00
0
CP 154526
A non-peptidic selectiveCRF-RI (CRF1 receptor) antagonist
257639-98-8 sc-205268
sc-205268A
10 mg
50 mg
$179.00
$555.00
0
CP 376395 hydrochloride
A CRF-RI receptor antagonist
1013933-37-3 sc-205271
sc-205271A
10 mg
50 mg
$189.00
$781.00
0
Cyclosomatostatin
A non-selective somatostatin receptor antagonist
84211-54-1 sc-205280
1 mg
$227.00
0
MK 0524 sodium salt
A potent, selective DP1 receptor antagonist
572874-50-1 sc-205391
sc-205391A
1 mg
5 mg
$102.00
$284.00
4
N-Cyclohexanecarbonylpentadecylamine
A selective inhibitor of acidic palmitoyl ethanolamidase
702638-84-4 sc-205403
sc-205403A
5 mg
10 mg
$41.00
$77.00
0
Roxatidine Acetate Hydrochloride
An antagonist of the histamine H2-receptor
93793-83-0 sc-205844
sc-205844A
100 mg
500 mg
$80.00
$240.00
0
Yangonin
One of the major components of kava extract
500-62-9 sc-205889
sc-205889A
5 mg
10 mg
$263.00
$500.00
0
Linvanil
A TRPV1 ligand
104899-01-6 sc-205951
5 mg
$288.00
0
Bosentan
A mixed endothelin receptor antagonist
147536-97-8 sc-210957
10 mg
$187.00
3
2-Furoyl-LIGRLO-amide trifluoroacetate salt
A potent, selective PAR2 agonist
729589-58-6 (non-salt) sc-213814
1 mg
$121.00
0
Creatine, anhydrous
Involved in the rapid production of ATP in skeletal muscle tissue
57-00-1 sc-214774
sc-214774A
10 mg
50 g
$20.00
$58.00
0
L-Aminobutyric Acid
A receptor antagonist
1492-24-6 sc-218628
5 g
$60.00
0
Nortriptyline-d3 Hydrochloride
A deuterium labeled tricyclic compound
203784-52-5 sc-219415
1 mg
$250.00
0
(R)-2-Isopropyl-3,6-dimethoxy-2,5-dihydropyrazine
An inhibitor with antitumor activity
109838-85-9 sc-219735
1 g
$180.00
0
BQ-610
A highly selective ETA receptor antagonist
141595-53-1 sc-221380
500 µg
$320.00
0
D-Cycloserine
Antibiotic and a partial agonist of NMDA receptors at the glycine modulatory site
68-41-7 sc-221470
sc-221470A
sc-221470B
sc-221470C
200 mg
1 g
5 g
25 g
$21.00
$59.00
$109.00
$500.00
4
GSK-3 Inhibitor IX, Control, MeBIO
A cell-permeable N-methylated kinase inactive analog of GSK-3 Inhibitor IX
710323-61-8 sc-221688
1 mg
$135.00
0
NBI-31772
An insulin-like growth factor-I binding protein (IGFBP) ligand
374620-70-9 sc-222047
5 mg
$232.00
0
L-alpha-Phosphatidylinositol-3,4,5-trisphosphate, Dipalmitoyl-, Heptaammonium Salt
A Ca2+-insensitive PKCδ, PKCε, and PKCη activator
sc-222174
100 µg
$348.00
1
SB-366791
A potent and selective vanilloid receptor (TRPV1) antagonist
472981-92-3 sc-222293
sc-222293A
5 mg
25 mg
$62.00
$259.00
0
t-CAA
A kainate receptor agonist and glutamate uptake inhibitor
sc-222334
1 mg
$200.00
0
trans-Zeatin
A member of cytokinin family of plant growth regulators
1637-39-4 sc-222365
sc-222365A
5 mg
10 mg
$52.00
$89.00
0
SB 218795
A potent and selective NK3 antagonist
174635-53-1 sc-224280
sc-224280A
10 mg
50 mg
$185.00
$825.00
0
SB 222200
A potent, selective non-peptide NK3 antagonist
174635-69-9 sc-224282
sc-224282A
10 mg
50 mg
$205.00
$800.00
1
Oxytocin acetate salt
An Oxytocin receptor activator
50-56-6 sc-279938
sc-279938A
1 mg
5 mg
$52.00
$167.00
0
4-(Aminomethyl)-L-phenylalanine
A noncanonical aminomethyl derivative of phenylalanine
150338-20-8 sc-284056
sc-284056A
250 mg
1 g
$124.00
$228.00
0
Wang resin
An excellent resin for the synthesis of peptide acids using Fmoc strategy
201058-08-4 sc-286858
sc-286858A
5 g
25 g
$40.00
$72.00
0
FPR A14
An agonist of the formyl peptide receptor (FPR)
sc-294992
sc-294992A
10 mg
50 mg
$149.00
$645.00
0
LU AA33810
A potent NPY5-R antagonist
304008-29-5 sc-295367
sc-295367A
10 mg
50 mg
$145.00
$638.00
0
NPY 5RA972
A potent and selective NPY5-R antagonist
439861-56-0 sc-295945
sc-295945A
10 mg
50 mg
$169.00
$712.00
0
TrkA Inhibitor
A cell-permeable, reversible, potent, and highly selective TrkA inhibitor
388626-12-8 sc-311553
1 mg
$165.00
0
SU1498
An Flk-1 kinase inhibitor
sc-355982
5 mg
$350.00
0
AC 264613
A potent and selective protease-activated receptor 2 agonist
1051487-82-1 sc-358026
sc-358026A
10 mg
50 mg
$170.00
$709.00
0
TNF-alpha Antagonist
A cyclic peptide that mimics the most critical TNF recognition loop on TNF-R1
199999-60-5 sc-358755
1 mg
$272.00
4
ATC 0065
A selective and potent antagonist of the MCH1
510732-84-0 sc-358785
sc-358785A
10 mg
50 mg
$179.00
$825.00
0
(Glp1)-Apelin-13
A potent Apelin receptor (APJ) peptide agonist
217082-60-5 sc-359030
1 mg
$155.00
0
SLIGRL-NH2
A PAR2-activating agonist peptide
171436-38-7 sc-359903
1 mg
$75.00
0
CP 96345
A selective and potent non-peptide NK1receptor antagonist
132746-60-2 sc-361160
sc-361160A
5 mg
25 mg
$110.00
$420.00
0
[D-Arg1,D-Phe5,D-Trp7,9,Leu11]-Substance P
A broad spectrum neuropeptide antagonist and inverse agonist
96736-12-8 sc-361166
1 mg
$94.00
0
GR 159897
A compound that acts as an effective and selective NK2 receptor antagonist
158848-32-9 sc-361193
sc-361193A
5 mg
25 mg
$182.00
$620.00
2
GR 231118
A potent NPY1-R antagonist and NPY4-R agonist
158859-98-4 sc-361194
500 µg
$345.00
0
ICI 216,140
An effective antagonist of the bombesin/gastrin releasing peptide
124001-41-8 sc-361211
1 mg
$295.00
0
LY 225910
A potent CCK-BR antagonist
133040-77-4 sc-361237
sc-361237A
5 mg
25 mg
$139.00
$585.00
0
NNC 26-9100
A somatostatin sst4 receptor agonist
199522-35-5 sc-361276
10 mg
$240.00
0
S 25585
A potent antagonist of the neuropeptide Y (NPY) Y5 receptor
263849-50-9 sc-361325
sc-361325A
10 mg
50 mg
$179.00
$760.00
0
SB 408124
A selective non-peptide orexin R-1 receptor inhibitor
288150-92-5 sc-361345
5 mg
$135.00
0
SN 003
A corticotropin releasing factor receptor 1 (CRF-RI) reversible antagonist
197801-88-0 sc-361361
10 mg
$175.00
0
SSR 146977 hydrochloride
A selective and potent NK3 receptor antagonist
264618-44-2 sc-361366
sc-361366A
10 mg
50 mg
$209.00
$875.00
0
TCS 1102
N effective antagonist of the dual orexin receptor
916141-36-1 sc-361375
sc-361375A
10 mg
50 mg
$145.00
$615.00
0
YIL 781
A (GHS-R1) antagonist that improves glucose tolerance
875258-85-8 sc-361410
sc-361410A
10 mg
50 mg
$179.00
$825.00
0
LRGILS-NH2
245329-01-5 sc-361979
1 mg
$129.00
0
L 760735
A high affinity NK1 receptor antagonist
188923-01-5 sc-362760
sc-362760A
10 mg
50 mg
$161.00
$906.00
0
SB 268262
A calcitonin inhibitor
217438-17-0 sc-362793
sc-362793A
10 mg
50 mg
$199.00
$849.00
0
GW 803430
A melanin-concentrating hormone receptor 1 antagonist
515141-51-2 sc-363281
sc-363281A
10 mg
50 mg
$199.00
$849.00
0
Exendin-3 (9-39)
A potent and selecive GLP-1 receptor antagonist.
133514-43-9 sc-364387
500 µg
$310.00
3
Ghrelin (human)
An endogenous peptide GHS-R agonist
258279-04-8 sc-364689
0.5 mg
$168.00
0
Seglitide
Peptide agonist for SSTR2 and SSTR5 receptor
81377-02-8 sc-391008
1 mg
$146.00
0
Alytesin
Stimulates gastric acid, intestinal contraction and hypertension
31078-12-3 sc-391186
1 mg
$175.00
0
GIP (HUMAN)
A hormone that induces insulin secretion in response to glucose.
100040-31-1 sc-396673
1 mg
$492.00
0
Neuromedin (Porcine)
81608-30-2 sc-396716
1 mg
$169.00
0
4-Carboxymethylphenylalanine Hydrocholoride
An aromatic compound with high affinity for CCK-B receptor
140233-60-9 sc-397458
1 g
$700.00
0
Kinetensin
A neurotensin-related peptide that increases vascular permeability
103131-69-7 sc-397563
1 mg
$100.00
0
GRP
74815-57-9 sc-495870
1 mg
$215.00
0

Santa Cruz Biotechnology, Inc. is a world leader in the development of products for the biomedical research market. Call us Toll Free at 1-800-457-3801.
Copyright © 2007-2019 Santa Cruz Biotechnology, Inc. All Rights Reserved. "Santa Cruz Biotechnology", and the Santa Cruz Biotechnology, Inc. logo, "Santa Cruz Animal Health", "San Juan Ranch", "Supplement of Champions", the San Juan Ranch logo, "Ultracruz", "Chemcruz", "Immunocruz", "Exactacruz", and "EZ Touch" are registered trademarks of Santa Cruz Biotechnology, Inc.
All trademarks are the property of their respective owners.