Histamine Receptor Inhibitors

Histamine is an inflammatory mediator that is ubiquitously expressed and has a broad range of pharmacologic effects. The effects of histamine are mediated by a family of G protein-coupled receptors, the Histamine H1, H2, H3 and H4 Receptors. Histamine Receptor Inhibitors offered by Santa Cruz inhibit Histamine Receptor and, in some cases, other inflammation and immune response related proteins. View detailed Histamine Receptor Inhibitor specifications, including Histamine Receptor Inhibitor CAS number, molecular weight, molecular formula and chemical structure, by clicking on the product name.

PRODUCT NAME/Application CAS Catalog # QUANTITY Price Citations RATING
Astemizole
A potent and selective H1-receptor antagonist that displays antihistamine and antimalarial activity
68844-77-9 sc-201088
sc-201088A
10 mg
50 mg
$69.00
$275.00
0
Thioperamide dot maleate
A potent and selective histamine H3 receptor antagonist shown to cross the blood-brain barrier
148440-81-7 sc-201092
sc-201092A
10 mg
50 mg
$100.00
$440.00
0
Ketotifen fumarate
A histamine H1 antagonist and mast cell growth inhibitor
34580-14-8 sc-201094
sc-201094A
1 g
100 mg
$62.00
$39.00
0
Cetirizine Dihydrochloride
A Histamine H1 receptor inverse agonist
83881-52-1 sc-202992
50 mg
$59.00
0
Cimetidine
An inhibitor of histamine binding to histamine H2 receptors
51481-61-9 sc-202996
sc-202996A
5 g
10 g
$62.00
$86.00
1
Dimebolin dihydrochloride
A histamine, AR, and Ca channel inhibitor
97657-92-6 sc-294348
sc-294348A
sc-294348B
1 mg
5 mg
50 mg
$37.00
$96.00
$384.00
0
Clobenpropit Dihydrobromide, VUF 9153
A histamine H3 receptor antagonist
145231-45-4 sc-202999
sc-202999A
10 mg
50 mg
$155.00
$620.00
0
Burimamide oxalate
A mixed H2/H3 antagonist
34970-69-9 sc-203535
sc-203535A
10 mg
50 mg
$200.00
$825.00
0
Conessine
A selective antagonist at the histamine H3-receptor
546-06-5 sc-203554
50 mg
$125.00
0
Impentamine dihydrobromide
A selective H3 receptor antagonist
34973-91-6 sc-203604
sc-203604A
10 mg
50 mg
$125.00
$525.00
0
JNJ 10191584 maleate
A selective histamine H4 receptor silent antagonist
869497-75-6 sc-203613
sc-203613A
10 mg
50 mg
$125.00
$525.00
0
Mepyramine maleate
A histamine H1 receptor antagonist
59-33-6 sc-203629
sc-203629A
100 mg
1 g
$65.00
$220.00
1
Ranitidine
A selective and competitive histamine H2 receptor inhibitor
66357-35-5 sc-203679
1 g
$180.00
0
Aminopotentidine
A histamine H2-receptor antagonist
140873-26-3 sc-203817
10 mg
$175.00
0
Clemastine fumarate
A selective histamine H1 antagonist
14976-57-9 sc-203897
100 mg
$95.00
0
Doxepin hydrochloride
A highly potent histamine H1 antagonist with affinity to H4 receptor
1229-29-4 sc-203930
1 g
$32.00
0
Deschloro Cetirizine Dihydrochloride
A Cetirizine impurity
83881-54-3 sc-391929
50 mg
$280.00
0
Fananserin
An antagonist of 5-HT2A
127625-29-0 sc-203951
sc-203951A
10 mg
50 mg
$129.00
$548.00
0
Lidocaine
A selective inverse peripheral histamine H1-receptor agonist
137-58-6 sc-204056
sc-204056A
50 mg
1 g
$49.00
$125.00
0
Mirtazapine
A potent SR-2, SR-3, and Histamine H1 receptor antagonist
85650-52-8 sc-204088
sc-204088A
10 mg
50 mg
$105.00
$409.00
0
trans-Triprolidine hydrochloride
A potent H1 receptor antagonist
6138-79-0 sc-204354
1 g
$35.00
0
VUF 5681 dihydrobromide
A potent histamine H3-receptor silent antagonist
639089-06-8 sc-204389
sc-204389A
10 mg
50 mg
$165.00
$700.00
0
Desloratadine N-Hydroxypiperidine
A related compound of Desloratadine
1193725-73-3 sc-391888
10 mg
$280.00
0
Diphenhydramine hydrochloride
A histamine H1-receptor antagonist
147-24-0 sc-204729
sc-204729A
sc-204729B
10 g
25 g
100 g
$50.00
$80.00
$120.00
0
ROS 234 dioxalate
A potent H3 antagonist
184576-87-2 sc-204893
sc-204893A
10 mg
50 mg
$140.00
$585.00
0
Clobenpropit hydrobromide
A histamine H3 receptor antagonist
145231-35-2 sc-205258
sc-205258A
1 mg
10 mg
$36.00
$288.00
0
2prime-O-(tert-Butyldimethylsilyl)-6,7-dehydropaclitaxel
165065-02-1 sc-206548
1 mg
$250.00
0
Terfenadine
A histamine H1-receptor antagonist, which blocks HERG and KIR6 channels
50679-08-8 sc-208421
5 g
$85.00
0
Embramine Hydrochloride
An antihistamine for proteomics research
13977-28-1 sc-396124
sc-396124A
100 mg
5 mg
$280.00
$20.00
0
Brompheniramine Maleate
A histamine H1 receptors antagonist
980-71-2 sc-210967
sc-210967A
25 mg
250 mg
$60.00
$200.00
1
Meclizine Dihydrochloride
A histamine H1 receptor antagonist and pregnane X receptor (PXR) agonist
1104-22-9 sc-211779
sc-211779A
10 g
5 g
$150.00
$85.00
1
Olopatadine Hydrochloride
A dual acting histamine H1-receptor antagonist and mast cell stabilizer
140462-76-6 sc-212473
25 mg
$140.00
0
A 943931 dihydrochloride
A potent and selective H4 receptor antagonist
1227675-50-4 sc-291775
sc-291775A
10 mg
50 mg
$205.00
$849.00
0
Azaperone
An α-adrenergic, dopamine and histamine receptor inhibitor
1649-18-9 sc-210851
100 mg
$284.00
0
A 987306
A potent and selective histamine H4 receptor antagonist
1082954-71-9 sc-291776
sc-291776A
10 mg
50 mg
$209.00
$875.00
0
Zotepine
An SR-2A and D2DR inhibitor and Histamine H1 receptor antagonist
26615-21-4 sc-360895
sc-360895A
10 mg
50 mg
$66.00
$246.00
0
Asenapine maleate
An antagonist of noradrenalin, dopamine, 5-HT and receptors
65576-45-6 sc-361110
sc-361110A
10 mg
50 mg
$145.00
$615.00
0
BF 2649
A histamine H3 receptor antagonist and inverse agonist
903576-44-3 sc-361119
sc-361119A
sc-361119B
sc-361119C
10 mg
50 mg
100 mg
1 g
$159.00
$585.00
$1,000.00
$3,600.00
0
Carcinine ditrifluoroacetate
A selective H3 receptor antagonist
56897-53-1 sc-361133
50 mg
$159.00
0
ICI 162,846
A potent histamine H2 receptor antagonist
84545-30-2 sc-361207
50 mg
$200.00
0
Iodophenpropit dihydrobromide
An antagonist of histamine H3
143407-29-8 sc-361213
sc-361213A
10 mg
50 mg
$149.00
$630.00
0
JNJ 10181457 dihydrochloride
A membrane permeable histamine H3 receptor antagonist
544707-19-9 sc-361216
sc-361216A
10 mg
50 mg
$169.00
$793.00
0
(S)-(+)-Dimethindene maleate
A subtype-selective mAChR M2 antagonist and histamine H1 receptor antagonist
121367-05-3 sc-361329
sc-361329A
10 mg
50 mg
$165.00
$700.00
0
GT 2016
A high affinity antagonist of the H3 receptor
152241-24-2 sc-362740
sc-362740A
10 mg
50 mg
$145.00
$645.00
0
Zolantidine dimaleate
A selective and penetrating H2 receptor inhibitor
104076-38-2 sc-364691
25 mg
$522.00
0

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