Cholinergics

Santa Cruz Biotechnology now offers a broad range of Cholinergics. Cholinergics are compounds which can stimulate or inhibit the production or release of acetylcholine, mimic the effects of acetylcholine, or activate or inhibit acetylcholine receptors. Due to the variety of compounds encompassed in this group, Cholinergics are useful for studying a wide range of physiological systems. Our popular products such as (±)-Anatoxin A Fumarate and Acetyl-L-carnitine chloride are typically available for immediate shipment.

indicates a highly recommended product based on customer preference.

PRODUCT NAME/Application CAS Catalog # QUANTITY Price Citations RATING
4-DAMP
An antagonist of mAChR M3
1952-15-4 sc-200167
50 mg
$119.00
2
Hydroxytacrine maleate
A cholinesterase inhibitor that exhibits a biochemical profile very similar to tacrine
118909-22-1 sc-200168
sc-200168A
200 mg
1 g
$68.00
$259.00
7
Oxotremorine Sesquifumarate
An M2 and M4 Muscarinic acetylcholine receptor agonist
17360-35-9 sc-200170
sc-200170A
100 mg
500 mg
$52.00
$207.00
0
Tacrine Hydrochloride
An anticholinesterase (AChE) inhibitor
1684-40-8 sc-200172
sc-200172A
1 g
5 g
$40.00
$105.00
0
(+/-)-Vesamicol dot HCl (AH-5183)
A blocker of acetylcholine transfer into nerve terminal vesicles
120447-62-3 sc-200174
200 mg
$120.00
0
Gallamine Triethiodide
A cardioselective mAChR M2 antagonist
65-29-2 sc-200175
sc-200175A
1 g
5 g
$63.00
$91.00
0
(+/-)-Epibatidine
A particularly potent AChR agonist
140111-52-0 sc-200177
sc-200177A
1 mg
5 mg
$62.00
$251.00
0
Galanthamine Hydrobromide
A competitive and reversible acetylcholinesterase inhibitor
1953-04-4 sc-200179
sc-200179A
25 mg
100 mg
$42.00
$94.00
1
Himbacine
An alkaloid muscarinic receptor antagonist
6879-74-9 sc-200181
sc-200181A
1 mg
5 mg
$62.00
$287.00
2
(+/-)-Anatoxin A Fumarate
A cyanotoxin agonist of AChR
64285-06-9 sc-200185
1 mg
$225.00
0
McN-A-343
A selective agonist of mAChR M1
55-45-8 sc-200186A
sc-200186
10 mg
50 mg
$25.00
$75.00
4
PNU-282,987
A highly selective α7 nicotinic acetylcholine receptor agonist
123464-89-1 sc-200187
sc-200187A
10 mg
50 mg
$95.00
$355.00
0
Carbachol
An anti-apoptosis agent and TNF-α inhibitor
51-83-2 sc-202092
sc-202092A
sc-202092B
1 g
10 g
100 g
$82.00
$250.00
$1,200.00
4
5-Methylfurmethide
A potent muscarinic agonist
1197-60-0 sc-202891
sc-202891A
10 mg
50 mg
$42.00
$180.00
0
alpha-Bungarotoxin
An α-neurotoxin which competitively and irreversibly binds and blocks nAChR
11032-79-4 sc-202897
1 mg
$119.00
4
Acetylcholine chloride
A cholinergic neurotransmitter that can induce the opening of calcium channels
60-31-1 sc-202904
sc-202904A
sc-202904B
sc-202904C
sc-202904D
5 g
25 g
100 g
250 g
1 kg
$31.00
$43.00
$172.00
$380.00
$1,400.00
0
Cytisine
An AChR agonist and potent ligand for many AChR subtypes
485-35-8 sc-203015
sc-203015A
5 mg
25 mg
$56.00
$190.00
0
Lobeline hydrochloride
An AChR agonist
134-63-4 sc-203114
sc-203114A
50 mg
1 g
$35.00
$75.00
0
(-)-Nicotine ditartrate
A potent agonist of AChR
65-31-6 sc-203161
sc-203161A
sc-203161B
sc-203161C
1 g
5 g
10 g
25 g
$78.00
$148.00
$192.00
$258.00
0
Pancuronium dibromide
A nicotine neuromuscular antagonist
15500-66-0 sc-203179
sc-203179A
10 mg
50 mg
$49.00
$275.00
1
(+)-Pilocarpine hydrochloride
A nonselective cholinergic agonist
54-71-7 sc-203196
1 g
$41.00
2
PNU 120596
A type II positive allosteric modulator
501925-31-1 sc-203200
sc-203200A
1 mg
5 mg
$30.00
$80.00
0
(-)-Scopolamine hydrobromide
A competitive inhibitor of acetylcholine muscarinic receptors
114-49-8 sc-203259
1 g
$77.00
0
Atropine Sulfate Monohydrate
A chlolinergic receptor antagonist
5908-99-6 sc-203322
5 g
$85.00
0
4-Acetyl-1,1-dimethylpiperazinium iodide
An AChR agonist
75667-84-4 sc-203473
sc-203473A
10 mg
50 mg
$115.00
$473.00
0
5-IODO-A-85380 dihydrochloride
A subtype-selective agonist for AChR
213764-92-2 sc-203478
5 mg
$110.00
0
5-Iodo-A-85380, 5-trimethylstannyl N-BOC derivative
A precursor to 5-iodo-A-85380
213766-21-3 sc-203479
200 µg
$119.00
0
(+/-)-Acetylcarnitine chloride
A weak cholinergic agonist
2504-11-2 sc-203495
100 mg
$44.00
0
AF-DX 384
A potent mAChR M2/mAChR M4 selective antagonist
118290-27-0 sc-203498
sc-203498A
10 mg
50 mg
$129.00
$548.00
0
Ambenonium dichloride
A selective, potent and rapid reversible inhibitor of AChE
52022-31-8 sc-203507
sc-203507A
10 mg
50 mg
$119.00
$510.00
0
AQ-RA 741
A high affinity selective mAChR M2 antagonist
123548-16-3 sc-203517
sc-203517A
10 mg
50 mg
$135.00
$575.00
0
Arecaidine but-2-ynyl ester tosylate
A potent, selective mAChR M2 activator
119630-77-2 sc-203519
sc-203519A
10 mg
50 mg
$285.00
$364.00
0
Arecaidine propargyl ester tosylate
A potent muscarinic receptor agonist
147202-94-6 sc-203520
sc-203520A
10 mg
50 mg
$95.00
$399.00
0
DMAB-anabaseine dihydrochloride
A neuronal AChR partial agonist
32013-69-7 sc-203568
10 mg
$155.00
0
Ipratropium bromide
An N-isopropyl salt of atropine and muscarinic antagonist
22254-24-6 sc-203606
100 mg
$69.00
0
J 104129 fumarate
A mAChR M3 antagonist
244277-89-2 sc-203610
10 mg
$185.00
0
Oxotremorine M
A small molecule agonist of muscarinic receptors
63939-65-1 sc-203656
100 mg
$115.00
0
PD 102807
A selective mAChR M4 antagonist
23062-91-1 sc-203659
sc-203659A
10 mg
50 mg
$195.00
$880.00
0
Physostigmine hemisulfate
A useful analogue of Physostigmine
64-47-1 sc-203661
sc-203661A
10 mg
100 mg
$78.00
$520.00
0
TC 2559 difumarate
A partial agonist for AChR α4β2
212332-35-9 sc-203707
sc-203707A
10 mg
50 mg
$185.00
$781.00
0
1-Acetyl-4-methylpiperazine hydrochloride
An AChR agonist acetylcholine analog
60787-05-5 sc-203759
sc-203759A
10 mg
50 mg
$115.00
$473.00
0
Acephate
An inhibitor of acetylcholinesterase (AChE)
30560-19-1 sc-203800
50 mg
$59.00
0
Benzoquinonium Dibromide
An AChR and ganglion inhibitor
311-09-1 sc-203839
sc-203839A
10 mg
50 mg
$135.00
$560.00
0
Biperiden hydrochloride
A muscarinic receptor antagonist
1235-82-1 sc-203846
sc-203846A
10 mg
50 mg
$105.00
$409.00
0
Chk2 Inhibitor
A checkpoint kinase inhibitor that mediates apoptosis and cell cycle arrest
724708-21-8 sc-203885
500 µg
$458.00
0
DAU 5884 hydrochloride
An mAChR M3 antagonist
131780-47-7 sc-203912
sc-203912A
10 mg
50 mg
$135.00
$575.00
0
(+/-)-Decanoylcarnitine chloride
A homolog of acetylcarnitine chloride and an intermediate in lipid metabolism
14919-36-9 sc-203914
50 mg
$115.00
0
LY 2365109 hydrochloride
A potent and selective glycine transporter 1 (GlyT1) inhibitor
868265-28-5 sc-204063
sc-204063A
10 mg
50 mg
$209.00
$825.00
0
MG 624
An antagonist of neuronal AChR
77257-42-2 sc-204082
sc-204082A
10 mg
50 mg
$145.00
$605.00
1
Milameline hydrochloride
A muscarinic receptor agonist
139886-32-1 sc-204085
sc-204085A
10 mg
50 mg
$129.00
$548.00
0
MR 16728 hydrochloride
A stimulator of acetylcholine release from synaptosomes
207403-36-9 sc-204099
sc-204099A
10 mg
50 mg
$135.00
$595.00
0
(+/-)-Myristoylcarnitine chloride
A homolog of acetylcarnitine chloride, and an intermediate in lipid metabolism
14919-38-1 sc-204108
50 mg
$119.00
0
Nitrocaramiphen hydrochloride
A mAChR M1 selective muscarinic antagonist
98636-73-8 sc-204129
sc-204129A
10 mg
50 mg
$129.00
$535.00
0
NS 1738
A selective a7 nAchR allosteric modulator
501684-93-1 sc-204136
sc-204136A
10 mg
50 mg
$149.00
$620.00
0
(+/-)-Octanoylcarnitine chloride
An ester analog of acetylcarnitine chloride
18822-86-1 sc-204143
50 mg
$109.00
0
PG-9 maleate
A potent analgesic and nootropic agent
sc-204184
sc-204184A
10 mg
50 mg
$115.00
$473.00
0
PHA 568487
An agonist of AChR α7
527680-56-4 sc-204186
sc-204186A
10 mg
50 mg
$101.00
$575.00
0
Phenserine
Inhibitor of amyloid precursor protein (APP)
101246-66-6 sc-204188
50 mg
$129.00
1
Piracetam
A modulator of neurotransmitter-induced ion flux
7491-74-9 sc-204196
sc-204196A
5 g
25 g
$38.00
$66.00
0
Pirenzepine Dihydrochloride
An mAChR M1 selective antagonist
29868-97-1 sc-204197
100 mg
$69.00
2
RJR 2429 dihydrochloride
A potent AChR agonist
91556-75-1 sc-204237
sc-204237A
10 mg
50 mg
$183.00
$681.00
0
SM-21 maleate
Potent and selective σ2 antagonist, increasing release of ACh
155058-71-2 sc-204289
sc-204289A
10 mg
50 mg
$101.00
$550.00
0
TC 1698 dihydrochloride
A selective AChR α7 agonist
700834-58-8 sc-204324
sc-204324A
10 mg
50 mg
$155.00
$620.00
0
Telenzepine dihydrochloride
A potent and selective muscarnic receptor antagonist
147416-96-4 sc-204332
sc-204332A
10 mg
25 mg
$61.00
$125.00
0
VU 10010
A selective allosteric potentiator of M4 acetylcholine receptors
633283-39-3 sc-204387
sc-204387A
5 mg
25 mg
$80.00
$323.00
0
Xanomeline oxalate
A functionally selective mAChR M1 agonist
141064-23-5 sc-204402
10 mg
$155.00
0
Zamifenacin fumarate
A selective antagonist of mAChR M3 (M3 muscarinic receptor)
127308-98-9 sc-204416
sc-204416A
10 mg
50 mg
$175.00
$709.00
0
Darifenacin Hydrobromide
An M3 muscarinic acetylcholine receptor blocker
133099-07-7 sc-204708
sc-204708A
sc-204708B
10 mg
25 mg
50 mg
$85.00
$225.00
$450.00
3
Desoxypeganine hydrochloride
An inhibitor of acetylcholinesterase
61939-05-7 sc-204712
25 mg
$200.00
1
Itopride Hydrochloride
An AChE inhibitor and D2DR inhibitor
122892-31-3 sc-204778
sc-204778A
1 g
5 g
$134.00
$430.00
1
Neostigmine Bromide
An acetylcholine esterase inhibitor
114-80-7 sc-204816
sc-204816A
250 mg
1 g
$48.00
$72.00
0
(+/-)-Propionylcarnitine chloride
A homolog of acetylcarnitine chloride and an important intermediate in lipid metabolism
17298-37-2 sc-204864
50 mg
$82.00
0
Rivastigmine hydrogen tartrate
A parasympathomimetic or cholinergic agent
129101-54-8 sc-204883
sc-204883A
100 mg
250 mg
$152.00
$300.00
0
RJR 2403 oxalate
A selective AChR angonist
183288-99-5 sc-204884
sc-204884A
10 mg
50 mg
$119.00
$510.00
0
Mecamylamine Hydrochloride
A noncompetitive nicotinic AChR inhibitor
826-39-1 sc-205742
sc-205742A
5 mg
25 mg
$43.00
$129.00
1
Nefiracetam
Activator of L/N-type calcium channels, cholinergic, monoaminergic and GABAergic systems
77191-36-7 sc-205766
sc-205766A
100 mg
250 mg
$125.00
$140.00
0
Tropanyl 2-(4-chlorophenylthio)butanoate oxalate
Enhances acetylcholine release
sc-205983
10 mg
$60.00
0
Asoxime chloride
A cholinesterase reactivator
34433-31-3 sc-207304
50 mg
$339.00
0
(Carbethoxymethylene)triphenylphosphorane
A Wittig reagent and cholinesterase inhibitor
1099-45-2 sc-207403
50 g
$135.00
0
Choline chloride
An acyl group acceptor
67-48-1 sc-207430
sc-207430A
sc-207430B
10 mg
5 g
50 g
$15.00
$30.00
$45.00
0
Clidinium Bromide
An anticholinergic
3485-62-9 sc-207449
1 g
$47.00
0
Edrophonium chloride
116-38-1 sc-207610
sc-207610A
sc-207610B
250 mg
1 g
5 g
$48.00
$146.00
$373.00
1
Oxybutynin Chloride
An antagonist of M1, M2, & M3 muscarinic acetylcholine receptors
1508-65-2 sc-208141
2.5 g
$185.00
0
Paraoxon
A parathion metabolite and cholinesterase inhibitor
311-45-5 sc-208151
sc-208151A
sc-208151B
1 g
5 g
10 g
$400.00
$2,600.00
$5,000.00
1
Acetylthiocholine iodide
A nAChR agonist and substrate of acetylcholinesterase
1866-15-5 sc-208323
sc-208323A
sc-208323B
sc-208323C
sc-208323D
1 g
5 g
25 g
100 g
250 g
$30.00
$78.00
$350.00
$1,125.00
$2,600.00
0
Acetyl-L-carnitine chloride
A cholinergic agonist that stimulates neuronal response to serotonin and acetylcholine
5080-50-2 sc-210747
1 g
$25.00
0
D,L-Trihexyphenidyl, Hydrochloride
An anticholinergic tertiary amine
58947-95-8 sc-211201
5 g
$56.00
0
N-Butylscopolammonium Bromide
An anticholinergic and antispasmodic
149-64-4 sc-212165
10 mg
$135.00
0
(+/-)-Nicotine
An alkaloid found in tobacco with addictive and teratogenic properties
22083-74-5 sc-212379
250 mg
$217.00
1
o-Nicotine
A Nicotine analog
23950-04-1 sc-212458
sc-212458A
sc-212458B
sc-212458C
10 mg
25 mg
50 mg
100 mg
$280.00
$720.00
$1,410.00
$2,235.00
0
Obidoxime Chloride
A cholinesterase reactivator
114-90-9 sc-212467
1 g
$430.00
1
Propiverine, Hydrochloride
Used for treatment of urinary incontinence
54556-98-8 sc-212594
100 mg
$113.00
0
Solifenacin Hydrochloride
A muscarinic M3 receptor antagonist
180468-39-7 sc-212950
10 mg
$300.00
0
Succinylcholine chloride dihydrate
A cholinergic antagonist
6101-15-1 sc-212965
25 g
$79.00
0
Benzoylcholine chloride
2964-09-2 sc-214590
sc-214590A
25 g
50 g
$69.00
$226.00
0
Betaine
Researched for its role in osmoregulation and methionine biosynthesis
107-43-7 sc-214595
sc-214595A
50 g
100 g
$29.00
$37.00
0
(+)-Tubocurarine chloride pentahydrate
An inhibitor of AChR
6989-98-6 sc-216029
sc-216029A
250 mg
1 g
$91.00
$294.00
0
Acetylcholine-d9 Chloride
A deuterium labeled version of acetylcholine chloride
344298-95-9 sc-217569
sc-217569A
5 mg
10 mg
$250.00
$400.00
0
Entacapone-d10
A labeled form of the COMT inhibitor entacapone
sc-218316
1 mg
$210.00
0
Galanthamine
A selective acetylcholinesterase inhibitor
357-70-0 sc-218556
10 mg
$240.00
0
1-Benzyl-1-methyl-4-cyclopentylmethoxycarbonyl-piperidinium bromide
An acetylcholine transport inhibitor
sc-220461
5 mg
$400.00
0
alpha-NETA
A fluorescent choactase inhibitor
31059-54-8 sc-221190
sc-221190A
sc-221190B
sc-221190C
5 mg
25 mg
50 mg
100 mg
$54.00
$206.00
$195.00
$374.00
0
Methyllycaconitine Perchlorate, Delphinium sp.
An α-bungarotoxin neuronal nicotinic receptor antagonist
sc-221938
5 mg
$126.00
0
Tropanyl 2-(4-chlorophenoxy)propionate maleate
Causes an increased release of acetylcholine
sc-222373
10 mg
$200.00
0
Tropanyl 2-naphthoxypropionate maleate
Increases the release of acetylcholine
sc-222374
10 mg
$200.00
0
AF-DX 116
A selective mAChR M2 antagonist
102394-31-0 sc-223772
5 mg
$76.00
1
AB-MECA
A high affinity A3 adenosine receptor agonist
152918-26-8 sc-239176
1 mg
$84.00
0
Decamethonium bromide
A nicotinic acetylcholine receptor partial agonist
541-22-0 sc-239651
5 g
$120.00
0
Pilocarpine nitrate salt
A nonselectivce muscarinic acetylcholine receptor agonist
148-72-1 sc-250722
10 g
$174.00
0
Procyclidine hydrochloride
1508-76-5 sc-250777
1 g
$120.00
0
Bromoacetylcholine bromide
An affinity alkylating agent for nicotinic receptors
22004-27-9 sc-252517
500 mg
$290.00
0
cis-2-Methyl-5-trimethylammoniummethyl-1,3-oxathiolane iodide
76541-57-6 sc-252614
5 mg
$199.00
0
Methyllycaconitine citrate
A potent antagonist for α7-containing neuronal nicotinic receptors
112825-05-5 sc-253043
5 mg
$81.00
1
Acetyl-beta-methylcholine chloride
A metabolically stable analog of acetylcholine
62-51-1 sc-257063
sc-257063A
5 g
25 g
$45.00
$90.00
0
Acetylthiocholine chloride
A substrate for acetylcholinesterase
6050-81-3 sc-257066
sc-257066A
1 g
5 g
$65.00
$245.00
0
Lobeline sulfate
CAS: 134-64-5, MF: C44H54N2O4·H2SO4, MW: 772.99, Purity: ≥98%
134-64-5 sc-269345
1 g
$84.00
0
BQCA
A highly selective allosteric potentiator of the M1 muscarinic acetylcholine receptor (mAChR)
338747-41-4 sc-280627
sc-280627A
10 mg
50 mg
$71.00
$390.00
0
Acetylethylcholine mustard hydrochloride
An inhibitor of choactase (choline acetyl-transferase)
103994-00-9 sc-281685
sc-281685A
5 mg
25 mg
$50.00
$174.00
0
S-Butyrylthiocholine Iodide
A chromogenic substrate for cholinesterases
1866-16-6 sc-286740
5 g
$58.00
0
L-Hyoscyamine
A non-selective, competitive antagonist of the muscarinic acetylcholine receptors
101-31-5 sc-295290
sc-295290A
1 g
5 g
$86.00
$128.00
0
Procaine
A sodium channel blocker and inhibitor of a variety of processes
59-46-1 sc-296134
sc-296134A
25 g
50 g
$101.00
$180.00
0
14-Acetylvirescenine from Delphinium sp.
CAS: 71609-79-5, MF: C25H39NO7, MW: 465.58
71609-79-5 sc-297973
10 mg
$98.00
0
A-85380 dihydrochloride
sc-300146
5 mg
$849.00
0
Aminobenztropine
88097-86-3 sc-300194
50 mg
$183.00
0
(+/-)-Epibatidine dihydrochloride
CAS: 166374-43-2, MF: C11H13ClN22HCl, MW: 281.61, Purity: ≥98%
166374-43-2 sc-300512
5 mg
$150.00
0
LY2033298
An allosteric potentiator.
886047-13-8 sc-300942
5 mg
$255.00
0
N,N,N-Trimethyl-1-(4-trans-stilbenoxy)-2-propylammonium iodide
sc-301439
25 mg
$750.00
0
NDNI hydriodide
A highly selective α4β2 nicotinic receptor antagonist
244025-06-7 sc-301459
5 mg
$148.00
0
PNU-282987 hydrate
A highly selective AChR α7 agonist
123464-89-1 (anhydrous) sc-301554
10 mg
$133.00
0
R(-)-Quinuclidinyl benzilate methiodide
A nonselective muscarinic acetylcholine receptor antagonist
sc-301655
2 mg
$400.00
0
VU 0238429
1160247-92-6 sc-301975
sc-301975A
5 mg
25 mg
$74.00
$297.00
0
Xanomeline L-tartrate
MF: C14H23N3OS•xC4H6O6, MW: 281.42, Purity: ≥98%
sc-301981
5 mg
$156.00
0
VU 152100
A positive allosteric modulator of muscarinic choline receptor M4
409351-28-6 sc-311554
sc-311554A
5 mg
25 mg
$98.00
$384.00
0
Trospium Bromide
An antimuscarinic compound that blocks action at mAChR M
10405-02-4 sc-356177
100 mg
$1,575.00
0
Mepenzolate Bromide
An anticholinergic
76-90-4 sc-358272
5 g
$51.00
0
Desformylflustrabromine hydrochloride
A positive allosteric modulator of α4β2 nicotinic acetylcholine receptors
951322-11-5 sc-358800
sc-358800A
10 mg
50 mg
$145.00
$645.00
0
Bretylium Tosylate
An inhibitor of AChE
61-75-6 sc-360745
10 mg
$263.00
0
(S)-(+)-Dimethindene maleate
A subtype-selective mAChR M2 antagonist and histamine H1 receptor antagonist
121367-05-3 sc-361329
sc-361329A
10 mg
50 mg
$165.00
$700.00
0
(+)-Muscarine iodide
A muscarinic acetylcholine receptor agonist
24570-49-8 sc-362769
sc-362769A
sc-362769B
2 mg
5 mg
10 mg
$215.00
$300.00
$420.00
0
L-Cystine
A non-essential amino acid vital for human development
56-89-3 sc-394415
25 g
$42.00
0
Cyclopentolate Hydrochloride
A mydriatic
5870-29-1 sc-396350
50 mg
$240.00
0
W-84 dibromide
A potent allosteric modulator of muscarinic receptors
21093-51-6 sc-397260
10 mg
$140.00
0
Chlorisondamine diiodide
96750-66-2 sc-500792
sc-500792A
10 mg
50 mg
$127.00
$539.00
0

Santa Cruz Biotechnology, Inc. is a world leader in the development of products for the biomedical research market. Call us Toll Free at 1-800-457-3801.
Copyright © 2007-2019 Santa Cruz Biotechnology, Inc. All Rights Reserved. "Santa Cruz Biotechnology", and the Santa Cruz Biotechnology, Inc. logo, "Santa Cruz Animal Health", "San Juan Ranch", "Supplement of Champions", the San Juan Ranch logo, "Ultracruz", "Chemcruz", "Immunocruz", "Exactacruz", and "EZ Touch" are registered trademarks of Santa Cruz Biotechnology, Inc.
All trademarks are the property of their respective owners.