CYP Inhibitors

Santa Cruz Biotechnology now offers a broad range of CYP Inhibitors. Cytochrome P450 (CYP) proteins are heme-thiolate monooxygenases that mediate NADPH-dependent electron transport and function to oxidize a variety of structurally unrelated compounds, including steroids, fatty acids and xenobiotics. Cytochrome P450s are responsible for metabolizing arachidonic acid (AA) to hydroxyeicosatetraenoic acid (a regulator of blood pressure) and epoxyeicosatrienoic acid (a molecule involved in signaling events). CYP Inhibitors offered by Santa Cruz inhibit CYP and, in some cases, other NADPH-dependent electron transport and oxidation related proteins. View detailed CYP Inhibitor specifications, including CYP Inhibitor CAS number, molecular weight, molecular formula and chemical structure, by clicking on the product name.

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PRODUCT NAME/Application CAS Catalog # QUANTITY Price Citations RATING
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Furafylline
An inhibitor of Cytochrome P450 (CYP1A2) and phosphodiesterase (PDE)
80288-49-9 sc-215061
5 mg
$278.00
0
PPOH
An inhibitor of CYP epoxidase activity on arachadonic acid
206052-01-9 sc-205442
sc-205442A
1 mg
5 mg
$21.00
$95.00
0
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Troleandomycin
A macrolide antibiotic and an inhibitor of CYP
2751-09-9 sc-200747
sc-200747A
10 mg
50 mg
$87.00
$374.00
3
NDGA (Nordihydroguaiaretic acid)
An antioxidant and lipoxygenase inhibitor
500-38-9 sc-200487
1 g
$80.00
0
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17-ODYA (17-Octadecynoic acid)
A potent suicide inhibitor of LTB4 ω-oxidase
34450-18-5 sc-200488
sc-200488A
1 mg
10 mg
$45.00
$139.00
7
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7-Ethoxyresorufin
A fluorometric inhibitor of vasorelaxant responses
5725-91-7 sc-200606
sc-200606A
2 mg
10 mg
$120.00
$196.00
1
Roquefortine C
A potent neurotoxin produced most notably by Penicillium species
58735-64-1 sc-202323
500 µg
$350.00
4
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Ketoconazole-d8
An inhibitor of cytochrome P-450 dependent steps in the biosynthesis of steroid hormones in vivo
sc-280876
2.5 mg
$350.00
0
HET-0016
A potent and selective inhibitor of the biosynthesis of 20-HETE
339068-25-6 sc-200673
sc-200673A
5 mg
25 mg
$84.00
$325.00
2
Triadimefon
An antifungal cytochrome P450 inhibitor
43121-43-3 sc-204923
sc-204923A
5 g
10 g
$94.00
$150.00
0
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ETYA
A Cox, LO, and PLA2 inhibitor
1191-85-1 sc-200764
sc-200764A
20 mg
100 mg
$67.00
$284.00
1
Silybin
A major active constituent of silymarin which inhibits mitogen-activated protein kinase (MAPK)
22888-70-6 sc-202812
sc-202812A
1 g
5 g
$30.00
$50.00
2
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Cylindrospermopsin
A cyanotoxin inhibitor of protein synthesis
143545-90-8 sc-203014
sc-203014A
25 µg
100 µg
$161.00
$239.00
0
Ketoconazole
An inhibitor of CYP proteins, thromboxane synthetase, and 5-LO
65277-42-1 sc-200496
sc-200496A
50 mg
500 mg
$54.00
$249.00
12
Methoxsalen (8-Methoxypsoralen)
A potent suicide inhibitor of cytochrome P-450
298-81-7 sc-200505
1 g
$35.00
1
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Metyrapone
An inhibitor of cytochrome P450-mediated ω/ω-1 hydroxylase activity and CYP11B1
54-36-4 sc-200597
200 mg
$20.00
0
Proadifen hydrochloride
An inhibitor of NOS1, AChR, cytochrome P-450, and KIR6.1
62-68-0 sc-200492
sc-200492A
250 mg
1 g
$79.00
$235.00
0
Rhapontigenin
a natural analog of resveratrol and an inhibitor of CYP1A1
500-65-2 sc-296263
sc-296263A
1 mg
5 mg
$144.00
$578.00
0
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Omeprazole
A selective proton pump and CYP inhibitor
73590-58-6 sc-202265
50 mg
$65.00
2
Exemestane
A CYP19 (aromatase) inhibitor
107868-30-4 sc-203045
sc-203045A
25 mg
100 mg
$128.00
$395.00
0
Naringin
A citrus bioflavonoid reported to inhibit cytochrom P450 monooxygenase activity
10236-47-2 sc-203443
sc-203443A
25 g
50 g
$38.00
$92.00
1
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1-Aminobenzotriazole
A suicide substrate for CYP-450 and chloroperoxidase
1614-12-6 sc-200600
sc-200600A
50 mg
100 mg
$45.00
$119.00
5
TMS
An inhibitor of cytochrome P450 1B1 and cancer cell growth
24144-92-1 sc-203708
sc-203708A
10 mg
50 mg
$159.00
$409.00
0
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Liarozole hydrochloride
A Imidazole-containing compound that inhibits the cytochrome P450-dependent metabolism
145858-50-0 sc-204055
sc-204055A
10 mg
50 mg
$159.00
$670.00
0
Xanthohumol from hop (Humulus lupulus)
An inhibitor of cytochrome P450 enzymes
6754-58-1 sc-301982
5 mg
$201.00
0
BVT 948
A non-competitive protein tyrosine phosphatase inhibitor
39674-97-0 sc-203536
sc-203536A
10 mg
50 mg
$139.00
$585.00
0
Ticrynafen
A cytochrome P450 inhibitor
40180-04-9 sc-220253
10 mg
$196.00
0
Tioconazole
A cytochrome-P450 inhibitor
65899-73-2 sc-205864
sc-205864A
1 g
5 g
$75.00
$118.00
0
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Atipamezole hydrochloride
A selective α2-adrenergic receptor antagonist
104075-48-1 sc-291914
sc-291914A
10 mg
50 mg
$140.00
$592.00
0
PF 4981517
A potent and selective inhibitor of CYP3A4
1390637-82-7 sc-364347
sc-364347A
10 mg
50 mg
$245.00
$1,030.00
0
Abiraterone Acetate - Labeled d4
Abiraterone acetate-d4 binds and inhibits both wild type and mutant androgen receptors (AR). Adittionally, abiraterone is an inhibitor of the cytochrome p450 group of enzymes, which are responsible for a variety of oxidative metabolic reactions.
154229-18-2 (unlabeled) sc-352989
10 mg
$3,775.00
0
Naringenin-4prime-O-beta-D-Glucuronide
An inhibitor of cytochrome P450 isoform CYP1A2
158196-35-1 sc-295905
sc-295905A
500 µg
1 mg
$222.00
$885.00
0
Clotrimazole-d5
A deuterium labeled antifungal CYP inhibitor
sc-217942
1 mg
$250.00
0
2,3-dihydrothieno-Thiadiazole Carboxylate
An inhibitor of CYP2E1 and CYP2B4
sc-220770
sc-220770A
50 mg
100 mg
$20.00
$37.00
0
Cytochrome P450 14a-demethylase inhibitor 1F
An antifungal compound and a CYP inhibitor
sc-364340
sc-364340A
5 mg
10 mg
$305.00
$480.00
0
12(S)-hydroxy-16-Heptadecynoic Acid
A mechanism-based inhibitor of CYP ω hydroxylation
148019-74-3 sc-223157
sc-223157A
1 mg
5 mg
$76.00
$344.00
0
Avasimibe
A cholesterol reducing compound that also inhibits CYP
166518-60-1 sc-364315
sc-364315A
10 mg
50 mg
$105.00
$405.00
0
Cytochrome P450 14a-demethylase inhibitor 1A
An antifungal CYP inhibitor
1155360-99-8 sc-364335
sc-364335A
5 mg
10 mg
$305.00
$480.00
0
Cytochrome P450 14a-demethylase inhibitor 1B
An antifungal compound that inhibits cytochrome P450 isoenzymes
1155361-00-4 sc-364336
sc-364336A
5 mg
10 mg
$305.00
$480.00
0
Cytochrome P450 14a-demethylase inhibitor 1C
An antifungal compound and CYP inhibitor
1155361-01-5 sc-364337
sc-364337A
5 mg
10 mg
$305.00
$480.00
0
Galeterone
An antagonist to LNCaP AR
851983-85-2 sc-364495
sc-364495A
5 mg
25 mg
$244.00
$550.00
0
Cytochrome P450 14a-demethylase inhibitor 1D
An antifungal compound and cytochrome P450 inhibitor
1155361-02-6 sc-364338
sc-364338A
5 mg
10 mg
$305.00
$480.00
0
Letrozole
A CYP19 (aromatase) inhibitor
112809-51-5 sc-204791
sc-204791A
25 mg
50 mg
$77.00
$135.00
0
4,5-diphenyl-1,2,3-Thiadiazole
An antibiotic compound with CYP450 inhibitory properties
5393-99-7 sc-205127
sc-205127A
250 mg
500 mg
$20.00
$33.00
0
6prime,7prime-dihydroxy Bergamottin
A potent CYP3A4 inhibitor
145414-76-2 sc-205162
sc-205162A
1 mg
10 mg
$100.00
$600.00
0
MS-PPOH
A selective inhibitor of the epoxygenation reactions catalyzed by specific CYP450 isozymes
206052-02-0 sc-205392
sc-205392A
1 mg
5 mg
$35.00
$154.00
1
Clarithromycin
A macrolide antibiotic and protein synthesis inhibitor
81103-11-9 sc-205634
sc-205634A
100 mg
250 mg
$69.00
$113.00
0
Cytochrome P450 14a-demethylase inhibitor 1E
A potent antifungal compound that is also an inhibitor of CYP
1155361-03-7 sc-364339
sc-364339A
5 mg
10 mg
$305.00
$480.00
0
Isoniazid
An antituberculosis agent and an inhibitor/activator of CYP isoenzymes
54-85-3 sc-205722
sc-205722A
5 g
50 g
$20.00
$25.00
0
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Abiraterone Acetate
A steroidal inhibitor of CYP17A1 in androgen biosynthesis
154229-18-2 sc-207240
5 mg
$255.00
0
Aminoglutethimide
A CYP19 (aromatase) inhibitor
125-84-8 sc-207280
1 g
$160.00
0
Voriconazole
An antifungal CYP2C9 inhibitor
137234-62-9 sc-208487
10 mg
$125.00
0
Abiraterone Acetate-d4
A steroidal cytochrome p450 inhibitor
154229-18-2 (unlabeled) sc-217550
1 mg
$300.00
0
Cytochrome P450 14a-demethylase inhibitor 1G
An antifungal compound and CYP inhibitor
1155361-05-9 sc-364341
sc-364341A
5 mg
10 mg
$305.00
$480.00
0
Anastrozole
A CYP19 (aromatase) inhibitor
120511-73-1 sc-217647
10 mg
$70.00
0
Anastrozole-d12
A deuterium labeled CYP19 (aromatase) inhibitor
120511-73-1 (unlabeled) sc-217649
1 mg
$250.00
0
Clarithromycin-N-methyl-d3 (contains 2% d0)
A deuterium-labeled clarithromycin derivative and a CYP4A inhibitor and substrate
sc-217926
5 mg
$280.00
0
Exemestane-19-d3
A deuterium-labeled analog of exemestane
sc-218454
1 mg
$500.00
0
Isoniazid-d4
An inhibitor and an inducer of various isoforms of CYP450
774596-24-6 sc-218611
1 mg
$300.00
0
Cytochrome P450 14a-demethylase inhibitor 1H
An antifungal compound and an inhibitor of CYP
1155361-06-0 sc-364342
sc-364342A
5 mg
10 mg
$305.00
$480.00
0
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Voriconazole-d3
A labeled Ergosterol Biosynthesis inhibitor
137234-62-9 unlabeled sc-220387
1 mg
$300.00
1
alpha-Asarone
An inhibitor of HMG-CoA reductase and CYP isoenzymes
2883-98-9 sc-239153
1 g
$55.00
0
Naringin dihydrochalcone
A citrus bioflavonoid that is also an inhibitor of CYP enzymes
18916-17-1 sc-279909
sc-279909A
10 g
25 g
$200.00
$315.00
0
Letrozole-d4
A deuterated version of Letrozole, a nonsteroidal aromatase (CYP19) inhibitor
sc-280910
1 mg
$250.00
0
Clotrimazole
An antifungal compound and CYP inhibitor
23593-75-1 sc-3583
sc-3583A
100 mg
1 g
$35.00
$50.00
4
Cytochrome P450 14a-demethylase inhibitor 1I
An inhibitor of CYP and an antifungal compound
1155361-07-1 sc-364343
sc-364343A
5 mg
10 mg
$305.00
$480.00
0
Cytochrome P450 14a-demethylase inhibitor 1J
An inhibitor of CYP isoenzymes and an antifungal agent
1155361-08-2 sc-364344
sc-364344A
5 mg
10 mg
$305.00
$480.00
0
No data available
Tenofovir
A selective HIV reverse transcriptase (HIV-1 RT) inhibitor
147127-20-6 sc-204335
sc-204335A
10 mg
50 mg
$145.00
$615.00
8

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