Histamine H1 Receptor Inhibitors

Santa Cruz Biotechnology now offers a broad range of Histamine H1 Receptor Inhibitors. Histamine is an inflammatory mediator that is ubiquitously expressed and has a broad range of pharmacologic effects. The effects of histamine are mediated by a family of G protein-coupled receptors, the Histamine H1, H2, H3 and H4 Receptors. Histamine H1 Receptor Inhibitors offered by Santa Cruz inhibit Histamine H1 Receptor and, in some cases, other inflammation and immune response related proteins. View detailed Histamine H1 Receptor Inhibitor specifications, including Histamine H1 Receptor Inhibitor CAS number, molecular weight, molecular formula and chemical structure, by clicking on the product name.

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PRODUCT NAME/Application CAS Catalog # QUANTITY Price Citations RATING
Ketotifen fumarate
A histamine H1 antagonist and mast cell growth inhibitor
34580-14-8 sc-201094
sc-201094A
1 g
100 mg
$62.00
$39.00
0
Loratadine
A peripheral histamine H1 receptor agonist
79794-75-5 sc-203117
sc-203117A
10 mg
50 mg
$105.00
$446.00
1
Chlorpromazine, Hydrochloride
An inhibitor of PDE, D2DR, NOS1, and PLA2
69-09-0 sc-202537
sc-202537A
sc-202537B
sc-202537C
sc-202537D
500 mg
5 g
25 g
100 g
250 g
$32.00
$48.00
$140.00
$480.00
$1,060.00
1
Terfenadine
A histamine H1-receptor antagonist, which blocks HERG and KIR6 channels
50679-08-8 sc-208421
5 g
$85.00
0
Astemizole
A potent and selective H1-receptor antagonist that displays antihistamine and antimalarial activity
68844-77-9 sc-201088
sc-201088A
10 mg
50 mg
$69.00
$275.00
0
Methapyrilene HCl
A specialty product for proteomics research
135-23-9 sc-257708
1 g
$83.00
0
Diphenhydramine hydrochloride
A histamine H1-receptor antagonist
147-24-0 sc-204729
sc-204729A
sc-204729B
10 g
25 g
100 g
$50.00
$80.00
$0.00
0
Meclizine Dihydrochloride
A histamine H1 receptor antagonist and pregnane X receptor (PXR) agonist
1104-22-9 sc-211779
sc-211779A
10 g
5 g
$150.00
$85.00
1
(S)-(+)-Dimethindene maleate
A subtype-selective mAChR M2 antagonist and histamine H1 receptor antagonist
121367-05-3 sc-361329
sc-361329A
10 mg
50 mg
$165.00
$700.00
0
Mepyramine maleate
A histamine H1 receptor antagonist
59-33-6 sc-203629
sc-203629A
100 mg
1 g
$65.00
$220.00
1
Fluphenazine
A dopamine receptor antagonist
69-23-8 sc-205700
sc-205700A
1 g
5 g
$136.00
$415.00
0
Lidocaine
A selective inverse peripheral histamine H1-receptor agonist
137-58-6 sc-204056
sc-204056A
50 mg
1 g
$49.00
$125.00
0
Cyproheptadine hydrochloride
A non-selective 5-HT2 antagonist
969-33-5 sc-203557
50 mg
$85.00
1
Brompheniramine Maleate
A histamine H1 receptors antagonist
980-71-2 sc-210967
sc-210967A
25 mg
250 mg
$60.00
$200.00
1
Doxepin hydrochloride
A highly potent histamine H1 antagonist with affinity to H4 receptor
1229-29-4 sc-203930
1 g
$32.00
0
Hydroxyzine Dihydrochloride
A hetercyclic H1 receptor antagonist
2192-20-3 sc-205716
sc-205716A
5 g
10 g
$53.00
$103.00
0
Antazoline hydrochloride
An anticholinergic and antihistamine agent
2508-72-7 sc-203515
sc-203515A
sc-203515B
100 mg
1 g
5 g
$65.00
$80.00
$200.00
0
Fenspiride Hydrochloride
An α adrenergic and H1 histamine receptor antaonist
5053-08-7 sc-207684
10 mg
$145.00
0
trans-Triprolidine hydrochloride
A potent H1 receptor antagonist
6138-79-0 sc-204354
1 g
$35.00
0
Clemastine fumarate
A selective histamine H1 antagonist
14976-57-9 sc-203897
100 mg
$95.00
0
Zotepine
An SR-2A and D2DR inhibitor and Histamine H1 receptor antagonist
26615-21-4 sc-360895
sc-360895A
10 mg
50 mg
$66.00
$246.00
0
Oxatomide
An H1-histamine receptor antagonist
60607-34-3 sc-208136
10 mg
$200.00
0
Azelastine HCl
An H1-receptor antagonist with antiallergic effects and disrupts TNF alpha activity
79307-93-0 sc-201096
100 mg
$92.00
0
Levocabastine Hydrochloride
A histamine H1 receptor antagonist and anti-allergic agent
79547-78-7 sc-201095
10 mg
$184.00
3
Cetirizine Dihydrochloride
A Histamine H1 receptor inverse agonist
83881-52-1 sc-202992
50 mg
$59.00
0
Mirtazapine
A potent SR-2, SR-3, and Histamine H1 receptor antagonist
85650-52-8 sc-204088
sc-204088A
10 mg
50 mg
$105.00
$409.00
0
Ebastine
An antagonist of the histamine H1-receptor
90729-43-4 sc-205663
sc-205663A
1 g
5 g
$104.00
$420.00
1
Pemirolast Potassium Salt
An inhibitor of mast cell mediator release
100299-08-9 sc-208156
10 mg
$165.00
0
Desloratadine
A potent and selective H1-receptor agonist
100643-71-8 sc-202133
sc-202133A
100 mg
500 mg
$85.00
$384.00
2
Olopatadine Hydrochloride
A dual acting histamine H1-receptor antagonist and mast cell stabilizer
140462-76-6 sc-212473
25 mg
$140.00
0
(S)-Azelastine Hydrochloride
N orally active Histamine H1 Receptor
153408-27-6 sc-208363
1 mg
$250.00
0
(R)-Azelastine Hydrochloride
An orally active Histamine H1 Receptor
153408-28-7 sc-208236
1 mg
$250.00
0
Fexofenadine HCl
An antihistamine that inhibits Cox-1, Cox-2, and is a histamine H1 receptor agonist
153439-40-8 sc-203047
sc-203047A
10 mg
50 mg
$95.00
$399.00
0
Asenapine maleate
An antagonist of noradrenalin, dopamine, 5-HT and receptors
65576-45-6 sc-361110
sc-361110A
10 mg
50 mg
$145.00
$615.00
0
Iso Loratadine
An isomer of loratadine used to prepare tricyclic amides and ureas
170727-59-0 sc-394085
5 mg
$300.00
0
4-Diphenylmethoxy-1-methylpiperidine hydrochloride
N inhibitor of Histamine H1 Receptor
132-18-3 sc-254657
10 g
$67.00
0
Mianserin hydrochloride
A non-selective 5-HT2 receptor antagonist with moderate affinity for 5-HT6
21535-47-7 sc-358986
100 mg
$49.00
0
Phenindamine Hydrochloride
A Histamine H1 receptor inhibitor
5503-08-2 sc-460196
50 mg
$280.00
0
Fexofenadine
A metabolite of of terfenadine, a H1-Histamine receptor antagonist
83799-24-0 sc-218475
100 mg
$200.00
1
Chlorpheniramine Maleate
An antagonist of the histamine H1-receptor
113-92-8 sc-204684
sc-204684A
5 g
25 g
$29.00
$49.00
0
(S)-Cetirizine Dihydrochloride
A nonsedating type histamine H1-receptor antagonist
163837-48-7 sc-208364
2.5 mg
$250.00
0
Olopatadine N-Oxide
An active metabolite of Olopatadine
203188-31-2 sc-212474
2.5 mg
$280.00
0
Fexofenadine-d6
An H1-Histamine receptor antagonist
548783-71-7 sc-211506
1 mg
$210.00
1
Doxylamine Succinate
An H1 histamine receptor antagonist
562-10-7 sc-211381
100 mg
$100.00
0
Epinastine Hydrochloride
A tetracyclic, histamine H1 receptor antagonist
108929-04-0 sc-211420
10 mg
$86.00
0
Azelastine-13C,d3
An H1-histamine receptor antagonist
58581-89-8 (unlabeled) sc-217683
1 mg
$250.00
0
Rupatadine Fumarate
A dual histamine H1 and PAF antagonist
182349-12-8 sc-212795
10 mg
$160.00
0
Diphenhydramine-d6 Hydrochloride
A labeled H1-Histamine receptor antagonist
147-24-0 (unlabeled) sc-218244
1 mg
$250.00
0
Loratadine-d4
A labelled histamine H1-receptor inhibitor
381727-27-1 sc-280929
1 mg
$300.00
0
Chlorprothixene Hydrochloride
A D2DR inhibitor
6469-93-8 sc-211077
1 g
$30.00
0
Hydroxyzine
An H1 receptor antagonist
68-88-2 sc-207748
500 mg
$240.00
0
Fluphenazine Dihydrochloride
A D1DR and D2DR inhibitor
146-56-5 sc-211531
100 mg
$110.00
0
Orphenadrine Citrate Salt
A histaminergic compound
4682-36-4 sc-212481
5 g
$45.00
0
Promethazine Hydrochloride
An antagonist of the histamine H1-receptor
58-33-3 sc-212586
100 mg
$20.00
0
rac-N-Demethyl dimethindene-d3 hydrobromide
CAS: 151562-10-6 (unlabeled free base), MF: C19H19D3N2•HBr, MW: 362.32
151562-10-6 (unlabeled free base) sc-500664
1 mg
$280.00
0
Astemizole-d3
A labeled histamine H1-receptor anatagonist
1189961-39-4 sc-217667
1 mg
$450.00
0
Cetirizine-d8, Dihydrochloride
A nonsedating type histamine H1-receptor antagonist
sc-217874
1 mg
$250.00
0
alpha-Hydroxy olopatadine
1331822-32-2 sc-489117
1 mg
$300.00
0
Hydroxyzine-d8 Dihydrochloride
An H1 receptor antagonist
sc-280807
1 mg
$300.00
0
Hydroxyzine-d8
An H1 receptor antagonist
68-88-2 (unlabeled) sc-280806
1 mg
$165.00
0
Olopatadine-d6 Hydrochloride
A labeled Olopatadine
1217229-05-4 sc-219484
1 mg
$280.00
0
Trimipramine-d3 Maleate Salt
A serotonin transport blocker that also blocks norepinephrine uptake
521-78-8 (unlabeled) sc-220342
1 mg
$200.00
0
Mebhydroline 1,5-naphthalenedisulfonate salt
An H1 histamine receptor antagonist
6153-33-9 sc-263459
1 g
$20.00
0
Desmethyl Nizatidine
A main metabolite of Nizatidine
82586-78-5 sc-391545
2.5 mg
$280.00
0
Acrivastine
A second-generation antihistamine
87848-99-5 sc-357283
sc-357283A
10 mg
50 mg
$100.00
$304.00
0
Pheniramine maleate salt
An H1 histamine receptor antagonist
132-20-7 sc-253258
5 g
$110.00
0
Bepotastine besilate
An inhibitor of Histamine H1 Receptor.
190786-44-8 sc-482068
10 mg
$79.00
0
Diphenylamine Hydrochloride
An antagonist of histamine H1 receptor
537-67-7 sc-485023
25 g
$68.00
0

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