GABA Receptor Activators

Santa Cruz Biotechnology now offers a broad range of GABA Receptor Activators. In the central nervous system GABA functions as the main inhibitory transmitter by increasing a Cl- conductance that inhibits neuronal firing. GABA has been shown to activate both ionotropic (GABAA) and metabotropic (GABAB) receptors as well as a third class of receptors called GABAC. GABA Receptor Activators offered by Santa Cruz activate GABA Receptor and, in some cases, other ionotropic and metabotropic receptor related proteins. View detailed GABA Receptor Activator specifications, including GABA Receptor Activator CAS number, molecular weight, molecular formula and chemical structure, by clicking on the product name.

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PRODUCT NAME/Application CAS Catalog # QUANTITY Price Citations RATING
Etomidate
A GABAA receptors agonist
33125-97-2 sc-203577
10 mg
$122.00
0
Securinine
A GABA receptor antagonist
5610-40-2 sc-220097
sc-220097A
50 mg
100 mg
$175.00
$350.00
2
(+/-)-Baclofen
A selective agonist of the GABAB receptor
1134-47-0 sc-200464
sc-200464A
1 g
5 g
$49.00
$243.00
0
4-Imidazoleacetic acid hydrochloride
A competitive antagonist at GABAC receptors
3251-69-2 sc-254684
1 g
$119.00
0
Isoguvacine HCl
An agonist of Gamma-amino butyric acid receptors
68547-97-7 sc-200451
sc-200451A
10 mg
50 mg
$25.00
$108.00
2
Indiplon
A potent GABAAreceptor positive allosteric modulator
325715-02-4 sc-204011
sc-204011A
10 mg
50 mg
$129.00
$516.00
0
R-(+)-Baclofen hydrochloride
A seelctive GABAB receptor agonist
63701-55-3 sc-203229
sc-203229A
10 mg
50 mg
$30.00
$117.00
0
GABA
An inhibitory neurotransmitter in the CNS
56-12-2 sc-203053
sc-203053A
10 g
25 g
$40.00
$82.00
1
Hispidulin
A potent benzodiazepine (BZD) receptor ligand
1447-88-7 sc-203999
10 mg
$229.00
1
Muscimol
A potent and specific GABAA receptor agonist/GABA analog
2763-96-4 sc-200460
sc-200460A
5 mg
25 mg
$96.00
$225.00
2
Valerenic acid
A positive allosteric modulator of the GABAA receptor
3569-10-6 sc-204377
sc-204377A
1 mg
10 mg
$53.00
$460.00
1
TACA
A GABAA and GABAC agonist
38090-53-8 sc-203705
sc-203705A
10 mg
50 mg
$90.00
$290.00
0
THIP hydrochloride
A GABAA receptor agonist and GABAC receptor antagonist
64603-91-4 sc-204342
50 mg
$101.00
0
ZAPA sulfate
A selective potent GABAA receptor agonist
92138-10-8 sc-200471
sc-200471A
5 mg
25 mg
$71.00
$275.00
0
SKF 97541
A very potent GABAB agonist/GABAC antagonist
127729-35-5 sc-200469
sc-200469A
5 mg
25 mg
$101.00
$450.00
0
R-(+)-Baclofen (free base)
A selective GABAB receptor agonist
69308-37-8 sc-203228
sc-203228A
10 mg
50 mg
$50.00
$195.00
0
Loreclezole hydrochloride
A subtype-selective GABAA receptor agonist
117857-45-1 sc-204061
sc-204061A
10 mg
50 mg
$195.00
$825.00
0
rac BHFF
A GABAB receptor positive allosteric modulator
123557-91-5 sc-204228
sc-204228A
5 mg
25 mg
$110.00
$420.00
0
SB 205384
A GABAA receptor modulator
160296-13-9 sc-204263
sc-204263A
10 mg
50 mg
$195.00
$825.00
0
Org 20599
A positive allosteric modulator and agonist of GABA receptors
156685-94-8 sc-204150
sc-204150A
10 mg
50 mg
$185.00
$781.00
0
U 89843A
A positive allosteric modulator of GABAA receptors
157013-85-9 sc-204361
sc-204361A
10 mg
50 mg
$125.00
$525.00
0
5-Nitro-alpha-oxo-N-(1R)-phenylethyl]-1H-indole-3-acetamide
A GABA<sub>A</sub> α2 agonist
355022-97-8 sc-358561
sc-358561A
10 mg
50 mg
$135.00
$595.00
0
DS2
A positive allosteric modulator of δ-subunit containing GABA<sub>A</sub> receptors
374084-31-8 sc-294421
sc-294421A
10 mg
25 mg
$170.00
$700.00
0
AA 29504
A positive allosteric modulator of GABAA receptors
945828-50-2 sc-361096
sc-361096A
5 mg
25 mg
$83.00
$350.00
0
(S)-Baclofen
A specific GABA-B receptor agonist
66514-99-6 sc-396081
sc-396081A
sc-396081B
sc-396081C
10 mg
25 mg
50 mg
100 mg
$250.00
$500.00
$930.00
$2,000.00
0
Allopregnanolone
A neuroactive steroid
516-54-1 sc-203813
sc-203813A
5 mg
10 mg
$162.00
$193.00
1
Chlormezanone
A compound acting at the benzodiazapine site of GABAA receptors
80-77-3 sc-203887
1 g
$67.00
0
CL 218872
A benzodiazepine agonist selective for α1 subunit-containing GABAA receptors
66548-69-4 sc-203552
sc-203552A
10 mg
50 mg
$85.00
$319.00
0
CGS 20625
A central benzodiazepine receptor partial agonist
111205-55-1 sc-203545
sc-203545A
10 mg
50 mg
$169.00
$712.00
0
Primidone
A compound that potentiates GABA receptor function
125-33-7 sc-204861
5 g
$37.00
0
Acamprosate Calcium
A GABA receptor agonist and glutamatergic systems modulator
77337-73-6 sc-210733
100 mg
$140.00
0
L-838417
A subtype-selective GABAA receptor partial agonist
286456-42-6 sc-211693
5 mg
$209.00
0
Ganaxolone
A potent stereoselective modulator of GABAA receptors
38398-32-2 sc-203586
sc-203586A
10 mg
50 mg
$129.00
$560.00
0
7-Chloro-1-methyl-5-phenyl-[1,2,4]triazolo[4,3-a]quinolin-4-amine
An impurity of alprazolam
448950-89-8 sc-396449
5 mg
$300.00
0
Bretazenil
84379-13-5 sc-252512
5 mg
$150.00
0
Safranal
A chemical responsible for Saffron smell that is also a proposed GABA A receptor agonist activity in vitro
116-26-7 sc-472985
5 g
$100.00
0
Progabide
A GABAA and GABAB receptor agonistic
62666-20-0 sc-476638
sc-476638A
100 mg
5 mg
$300.00
$20.00
0
1-Methyl-4-imidazoleacetic acid hydrochloride
A metabolite
35454-39-8 sc-222712
sc-222712A
10 mg
250 mg
$60.00
$600.00
0
5-Oxo-Zaleplon
A metabolite of Zaleplon, a selective non-benzodiazepine GABAA receptor agonist
159225-99-7 sc-478295
10 mg
$300.00
0
Baclofen-d4
A specific GABA-B receptor agonist
1189938-30-4 sc-217694
1 mg
$450.00
0
3-Aminopropylphosphonic acid
13138-33-5 sc-251943
1 g
$142.00
0

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