NPY 5RA972 CAS: 439861-56-0
MF: C21H25N3O2
NPY 5RA972 is a potent and selective NPY5-R antagonist.

NPY 5RA972 (CAS 439861-56-0)

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Nomes alternativos: N-[4-Methyl-9-(1-methylethyl)-9H-carbazol-3-yl]-4-morpholinecarboxamide
Aplicação NPY 5RA972 is a potent and selective NPY5-R antagonist
Numero VAT: 439861-56-0
Peso Molecular: 351.44
Separar por Funcao: C21H25N3O2
Para uso em exclusivo em pesquisa. Não se destina a uso em diagnostico e tratamento.
Available in US only.
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NPY 5RA972 is a potent and selective NPY5-R (neuropeptide Y) antagonist (IC50 values are 3.1, >10000, >10000 and >10000 nM for NPY5-R, NPY1-R, NPY2-R and NPY4-R respectively). This compound does not block NPY-induced feeding in vivo. NPY 5RA972 has also been shown to be a brain penetrant.


Referencias

Block et al (2002) Discovery and optimization of a series of carbazole ureas as NPY5 antagonists for the treatment of obesity. J.Med.Chem. 45 3509. Turnbull et al (2002) Selective antagonism of the NPY Y5 receptor does not have a major effect on feeding i

Estado físico :
Solid
envie :
DMSO (100mM)
Manutencao :
Store at room temperature
Para uso em exclusivo em pesquisa. Não se destina a uso em diagnostico e tratamento.
Available in US only.
Transporte :
Not available for sale outside of the United States.
PubChem CID :
SMILES :
CC1=C(C=CC2=C1C3=CC=CC=C3N2C(C)C)NC(=O)N4CCOCC4

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