Zinterol CAS: 37000-20-7
MF: C19H26N2O4S
MW: 378.48
A potent and selective β 2-adrenoceptor agonist.

Zinterol (CAS 37000-20-7)

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Application: Zinterol is a potent and selective β 2-adrenoceptor agonist
CAS Number: 37000-20-7
Molecular Weight: 378.48
Molecular Formula: C19H26N2O4S
For Research Use Only. Not Intended for Diagnostic or Therapeutic Use.
* Refer to Certificate of Analysis for lot specific data (including water content).
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Zinterol is a potent and selective β2-AR (β2-adrenoceptor) agonist (pKB values are 8.3 and < 5.7 for β 2 and β1 receptors respectively, as measured in human artery).


References

Kaumann (1997) Four b-adrenoceptor subtypes in the mammalian heart. TiPS 18 70. Arvydas Skeberdis et al (1997) Beta-2 adrenergic activation of L-type Ca2+ current in cardiac myocytes. J.Pharmacol.Exp.Ther. 283 452. Hutchinson et al (2006) Agonist effects of zinterol at the mouse and human b3-adrenoceptor. Naunyn-Schmied.Arch.Pharmacol. 373 158.

Physical State :
Solid
Solubility :
Soluble to 25 mM in Water
Storage :
Store at 4° C
Melting Point :
228.21° C (Predicted)
Boiling Point :
574.29° C at 760 mmHg (Predicted)
Density :
1.28 g/cm3 (Predicted)
Refractive Index :
n20D 1.62 (Predicted)
IC50 :
β2-AR: EC5050 = 0.05 nM (human)
pK Values :
pKa: 8.57, pKb: 9.5
For Research Use Only. Not Intended for Diagnostic or Therapeutic Use.
PubChem CID :
MDL Number :
MFCD00867031
SMILES :
CC(C)(CC1=CC=CC=C1)NCC(C2=CC(=C(C=C2)O)NS(=O)(=O)C)O

Download SDS (MSDS)

Certificate of Analysis

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